Sfoglia per Autore
Design and synthesis of small libraries of peptidomimetics based on a thiazolidine moiety
2006-01-01 Campiglia, Pietro; GOMEZ MONTERREY, Isabel; Carotenuto, Alfonso; Lama, Teresa; DIURNO MARIA, V; Bertamino, Alessia; Mazzoni, Orazio; Sala, Marina; Novellino, Ettore; Grieco, Paolo
Design, Synthesis, and Cytotoxic Evaluation of a New Series of 3-Substituted Spiro[(dihydropyrazine-2,5-dione)-6,3‘-(2‘,3‘-dihydrothieno[2,3-b]naphtho-4‘,9‘-dione)] Derivatives
2007-01-01 Isabel Gomez, Monterrey; Campiglia, Pietro; Alfonso, Carotenuto; Daniela, Califano; Claudio, Pisano; Loredana, Vesci; Teresa, Lama; Bertamino, Alessia; Sala, Marina; Antonio Mazzella di, Bosco; Paolo, Grieco; Ettore, Novellino
A beta 16-35 peptide: structural features in membrane mimicking systems.
2008-01-01 Scrima, Mario; Grimaldi, Manuela; Esposito, Cinzia; Tedesco, A.; D'Errico, G.; Sala, Marina; Campiglia, Pietro; D'Ursi, Anna Maria
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1.
2008-01-01 Castellano, Sabrina; Kuck, D; Sala, Marina; Novellino, E; Lyko, F; Sbardella, Gianluca
Spiro[(dihydropyrazin-2,5-dione)-6,3′-(2′,3′- dihydrothieno[2,3-b]naphtho-4′,9′-dione)]-based cytotoxic agents: Structure-activity relationship studies on the substituent at N4-position of the diketopiperazine domain
2008-01-01 Gomez Monterrey, Isabel; Campiglia, Pietro; Carotenuto, Alfonso; Stiuso, Paola; Bertamino, Alessia; Sala, Marina; Aquino, Claudio; Grieco, Paolo; Morello, Silvana; Pinto, Aldo; Iannelli, Pio; Novellino, Ettore
Synthesis of novel indole-based ring systems by acid-catalysed condensation from α -amino aldehydes and L-Trp-OMe
2008-01-01 GOMEZ MONTERREY ISABEL, M; Campiglia, Pietro; Bertamino, Alessia; Aquino, Claudio; Mazzoni, Orazio; DIURNO MARIA, V; Iacovino, Rosa; Saviano, Michele; Sala, Marina; Novellino, Ettore; Grieco, Paolo
Novel route in the synthesis of ψ[CH2NH] amide bond surrogate
2008-01-01 Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Sala, Marina; Isabel M., Gomez Monterrey; Ettore, Novellino; Paolo, Grieco
A New Series of 1,3-Dihidro-Imidazo[1,5-c]thiazole-5,7-Dione Derivatives: Synthesis and Interaction with Aβ(25-35) Amyloid Peptide
2009-01-01 Campiglia, Pietro; Scrima, Mario; Grimaldi, Manuela; Cioffi, Giuseppina; Bertamino, Alessia; Sala, Marina; Claudio, Aquino; Isabel Gomez, Monterrey; Paolo, Grieco; Ettore, Novellino; D'Ursi, Anna Maria
New Insight into the Binding Mode of Peptide Ligands at Urotensin-II Receptor: Structure−Activity Relationships Study on P5U and Urantide
2009-01-01 Paolo, Grieco; Alfonso, Carotenuto; Campiglia, Pietro; Isabel Gomez, Monterrey; Luigia, Auriemma; Sala, Marina; Cristina, Marcozzi; Roberta d’Emmanuele di Villa, Bianca; Diego, Brancaccio; Paolo, Rovero; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Ettore, Novellino
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters
2010-01-01 Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Nicoletta De, Simone; Sala, Marina; Castellano, Sabrina; Marisabella, Santoriello; Paolo, Grieco; Ettore, Novellino; Isabel Maria Gomez, Monterrey
A novel quinone-based derivative (DTNQ-Pro) induces apoptotic death via modulation of heat shock protein expression in Caco-2 cells
2010-01-01 Gomez Monterrey, Isabe; Campiglia, Pietro; Bertamino, Alessia; Aquino, Claudio; Sala, Marina; Grieco, Paolo; Dicitore, Alessandra; Vanacore, Daniela; Porta, Amalia; Maresca, Bruno; Novellino, Ettore; Stiuso, Paola
Design and synthesis of spirotryprostatin-inspired diketopiperazine systems from prolyl spirooxoindolethiazolidine derivatives
2010-01-01 Bertamino, Alessia; Claudio, Aquino; Sala, Marina; Nicoletta de, Simone; Mattia, Carlo; Loredana, Erra; Musella, Simona; Iannelli, Pio; Alfonso, Carotenuto; Paolo, Grieco; Ettore, Novellino; Campiglia, Pietro; Isabel Gomez, Monterrey
Identification of the Spiro(oxindole-3,3 '-thiazolidine)-Based Derivatives as Potential p53 Activity Modulators
2010-01-01 Isabel Gomez, Monterrey; Bertamino, Alessia; Porta, Amalia; Alfonso, Carotenuto; Musella, Simona; Claudio, Aquino; Granata, Ilaria; Sala, Marina; Diego, Brancaccio; Delia, Picone; Carmine, Ercole; Paola, Stiuso; Campiglia, Pietro; Paolo, Grieco; Iannelli, Pio; Maresca, Bruno; Ettore, Novellino
Antiproliferative Activity of "Lycopersicon Esculentum" Leaves (var.Paul Robenson)Preliminary study
2011-01-01 Saturnino, Carmela; Popolo, Ada; Annalisa, Spagnuolo; Sirignano, Esther; Botta, Antonio; Sala, Marina; Giuseppina, Tommonaro; Maria Stefania, Sinicropi
Design,Synthesis and Biological Evaluation of New 4-Thiazolidinone Derivatives in Breast Cancer Cells
2012-01-01 Sala, Marina; Vernieri, Ermelinda; I. M., Gomez Monterrey; M. S., Sinicropi; V., Pezzi; A., Chimento; P., Tortorella; Saturnino, Carmela; E., Novellino; Campiglia, Pietro
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1
2012-01-01 Castellano, Sabrina; Spannhoff, Astrid; Milite, Ciro; DAL PIAZ, Fabrizio; Cheng, Donghang; Tosco, Alessandra; Viviano, Monica; Yamani, Abdellah; Cianciulli, Agostino; Sala, Marina; Cura, Vincent; Cavarelli, Jean; Novellino, Ettore; Mai, Antonello; Bedford, Mark T.; Sbardella, Gianluca
Isolation and Functional Characterization of Peptide Agonists of PTPRJ, a Tyrosine Phosphatase Receptor Endowed with Tumor Suppressor Activity
2012-01-01 Francesco, Paduano; Francesco, Ortuso; Campiglia, Pietro; Cinzia, Raso; Enrico, Iaccino; Marco, Gaspari; Gaudio, ; Graziella, Mangone; Alfonso, Carotenuto; Anna, Bilotta; Domenico, Narciso; Camillo, Palmieri; Valter, Agosti; Anna, Artese; Isabel Gomez, Monterrey; Sala, Marina; Giovanni, Cuda; Rodolfo, Iuliano; Nicola, Perrotti; Giuseppe, Scala; Giuseppe, Viglietto; Stefano, Alcaro; Carlo M., Croce; Ettore, Novellino; Alfredo, Fusco; Francesco, Trapasso
Heat Shock Protein 90 Inhibitors as Therapeutic Agents.
2012-01-01 Gomez Monterrey, I; Sala, Marina; Musella, S; Campiglia, Pietro
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors
2013-01-01 Vernieri, Ermelinda; Isabel Gomez, Monterrey; Milite, Ciro; Paolo, Grieco; Musella, Simona; Bertamino, Alessia; Ilaria, Scognamiglio; Stefano, Alcaro; Anna, Artese; Francesco, Ortuso; Ettore, Novellino; Sala, Marina; Campiglia, Pietro
Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2'-thiazolidine]-Based p53 Modulators
2013-01-01 Bertamino, Alessia; Maria, Soprano; Musella, Simona; Maria Rosaria, Rusciano; Sala, Marina; Vernieri, Ermelinda; DI SARNO, Veronica; Antonio, Limatola; Alfonso, Carotenuto; Sandro, Cosconati; Paolo, Grieco; Ettore, Novellino; Maddalena, Illario; Campiglia, Pietro; Isabel Gomez, Monterrey
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design and synthesis of small libraries of peptidomimetics based on a thiazolidine moiety | 1-gen-2006 | Campiglia, Pietro; GOMEZ MONTERREY, Isabel; Carotenuto, Alfonso; Lama, Teresa; DIURNO MARIA, V; Bertamino, Alessia; Mazzoni, Orazio; Sala, Marina; Novellino, Ettore; Grieco, Paolo | |
Design, Synthesis, and Cytotoxic Evaluation of a New Series of 3-Substituted Spiro[(dihydropyrazine-2,5-dione)-6,3‘-(2‘,3‘-dihydrothieno[2,3-b]naphtho-4‘,9‘-dione)] Derivatives | 1-gen-2007 | Isabel Gomez, Monterrey; Campiglia, Pietro; Alfonso, Carotenuto; Daniela, Califano; Claudio, Pisano; Loredana, Vesci; Teresa, Lama; Bertamino, Alessia; Sala, Marina; Antonio Mazzella di, Bosco; Paolo, Grieco; Ettore, Novellino | |
A beta 16-35 peptide: structural features in membrane mimicking systems. | 1-gen-2008 | Scrima, Mario; Grimaldi, Manuela; Esposito, Cinzia; Tedesco, A.; D'Errico, G.; Sala, Marina; Campiglia, Pietro; D'Ursi, Anna Maria | |
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. | 1-gen-2008 | Castellano, Sabrina; Kuck, D; Sala, Marina; Novellino, E; Lyko, F; Sbardella, Gianluca | |
Spiro[(dihydropyrazin-2,5-dione)-6,3′-(2′,3′- dihydrothieno[2,3-b]naphtho-4′,9′-dione)]-based cytotoxic agents: Structure-activity relationship studies on the substituent at N4-position of the diketopiperazine domain | 1-gen-2008 | Gomez Monterrey, Isabel; Campiglia, Pietro; Carotenuto, Alfonso; Stiuso, Paola; Bertamino, Alessia; Sala, Marina; Aquino, Claudio; Grieco, Paolo; Morello, Silvana; Pinto, Aldo; Iannelli, Pio; Novellino, Ettore | |
Synthesis of novel indole-based ring systems by acid-catalysed condensation from α -amino aldehydes and L-Trp-OMe | 1-gen-2008 | GOMEZ MONTERREY ISABEL, M; Campiglia, Pietro; Bertamino, Alessia; Aquino, Claudio; Mazzoni, Orazio; DIURNO MARIA, V; Iacovino, Rosa; Saviano, Michele; Sala, Marina; Novellino, Ettore; Grieco, Paolo | |
Novel route in the synthesis of ψ[CH2NH] amide bond surrogate | 1-gen-2008 | Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Sala, Marina; Isabel M., Gomez Monterrey; Ettore, Novellino; Paolo, Grieco | |
A New Series of 1,3-Dihidro-Imidazo[1,5-c]thiazole-5,7-Dione Derivatives: Synthesis and Interaction with Aβ(25-35) Amyloid Peptide | 1-gen-2009 | Campiglia, Pietro; Scrima, Mario; Grimaldi, Manuela; Cioffi, Giuseppina; Bertamino, Alessia; Sala, Marina; Claudio, Aquino; Isabel Gomez, Monterrey; Paolo, Grieco; Ettore, Novellino; D'Ursi, Anna Maria | |
New Insight into the Binding Mode of Peptide Ligands at Urotensin-II Receptor: Structure−Activity Relationships Study on P5U and Urantide | 1-gen-2009 | Paolo, Grieco; Alfonso, Carotenuto; Campiglia, Pietro; Isabel Gomez, Monterrey; Luigia, Auriemma; Sala, Marina; Cristina, Marcozzi; Roberta d’Emmanuele di Villa, Bianca; Diego, Brancaccio; Paolo, Rovero; Paolo, Santicioli; Stefania, Meini; Carlo A., Maggi; Ettore, Novellino | |
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters | 1-gen-2010 | Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Nicoletta De, Simone; Sala, Marina; Castellano, Sabrina; Marisabella, Santoriello; Paolo, Grieco; Ettore, Novellino; Isabel Maria Gomez, Monterrey | |
A novel quinone-based derivative (DTNQ-Pro) induces apoptotic death via modulation of heat shock protein expression in Caco-2 cells | 1-gen-2010 | Gomez Monterrey, Isabe; Campiglia, Pietro; Bertamino, Alessia; Aquino, Claudio; Sala, Marina; Grieco, Paolo; Dicitore, Alessandra; Vanacore, Daniela; Porta, Amalia; Maresca, Bruno; Novellino, Ettore; Stiuso, Paola | |
Design and synthesis of spirotryprostatin-inspired diketopiperazine systems from prolyl spirooxoindolethiazolidine derivatives | 1-gen-2010 | Bertamino, Alessia; Claudio, Aquino; Sala, Marina; Nicoletta de, Simone; Mattia, Carlo; Loredana, Erra; Musella, Simona; Iannelli, Pio; Alfonso, Carotenuto; Paolo, Grieco; Ettore, Novellino; Campiglia, Pietro; Isabel Gomez, Monterrey | |
Identification of the Spiro(oxindole-3,3 '-thiazolidine)-Based Derivatives as Potential p53 Activity Modulators | 1-gen-2010 | Isabel Gomez, Monterrey; Bertamino, Alessia; Porta, Amalia; Alfonso, Carotenuto; Musella, Simona; Claudio, Aquino; Granata, Ilaria; Sala, Marina; Diego, Brancaccio; Delia, Picone; Carmine, Ercole; Paola, Stiuso; Campiglia, Pietro; Paolo, Grieco; Iannelli, Pio; Maresca, Bruno; Ettore, Novellino | |
Antiproliferative Activity of "Lycopersicon Esculentum" Leaves (var.Paul Robenson)Preliminary study | 1-gen-2011 | Saturnino, Carmela; Popolo, Ada; Annalisa, Spagnuolo; Sirignano, Esther; Botta, Antonio; Sala, Marina; Giuseppina, Tommonaro; Maria Stefania, Sinicropi | |
Design,Synthesis and Biological Evaluation of New 4-Thiazolidinone Derivatives in Breast Cancer Cells | 1-gen-2012 | Sala, Marina; Vernieri, Ermelinda; I. M., Gomez Monterrey; M. S., Sinicropi; V., Pezzi; A., Chimento; P., Tortorella; Saturnino, Carmela; E., Novellino; Campiglia, Pietro | |
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 | 1-gen-2012 | Castellano, Sabrina; Spannhoff, Astrid; Milite, Ciro; DAL PIAZ, Fabrizio; Cheng, Donghang; Tosco, Alessandra; Viviano, Monica; Yamani, Abdellah; Cianciulli, Agostino; Sala, Marina; Cura, Vincent; Cavarelli, Jean; Novellino, Ettore; Mai, Antonello; Bedford, Mark T.; Sbardella, Gianluca | |
Isolation and Functional Characterization of Peptide Agonists of PTPRJ, a Tyrosine Phosphatase Receptor Endowed with Tumor Suppressor Activity | 1-gen-2012 | Francesco, Paduano; Francesco, Ortuso; Campiglia, Pietro; Cinzia, Raso; Enrico, Iaccino; Marco, Gaspari; Gaudio, ; Graziella, Mangone; Alfonso, Carotenuto; Anna, Bilotta; Domenico, Narciso; Camillo, Palmieri; Valter, Agosti; Anna, Artese; Isabel Gomez, Monterrey; Sala, Marina; Giovanni, Cuda; Rodolfo, Iuliano; Nicola, Perrotti; Giuseppe, Scala; Giuseppe, Viglietto; Stefano, Alcaro; Carlo M., Croce; Ettore, Novellino; Alfredo, Fusco; Francesco, Trapasso | |
Heat Shock Protein 90 Inhibitors as Therapeutic Agents. | 1-gen-2012 | Gomez Monterrey, I; Sala, Marina; Musella, S; Campiglia, Pietro | |
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors | 1-gen-2013 | Vernieri, Ermelinda; Isabel Gomez, Monterrey; Milite, Ciro; Paolo, Grieco; Musella, Simona; Bertamino, Alessia; Ilaria, Scognamiglio; Stefano, Alcaro; Anna, Artese; Francesco, Ortuso; Ettore, Novellino; Sala, Marina; Campiglia, Pietro | |
Synthesis, in Vitro, and in Cell Studies of a New Series of [Indoline-3,2'-thiazolidine]-Based p53 Modulators | 1-gen-2013 | Bertamino, Alessia; Maria, Soprano; Musella, Simona; Maria Rosaria, Rusciano; Sala, Marina; Vernieri, Ermelinda; DI SARNO, Veronica; Antonio, Limatola; Alfonso, Carotenuto; Sandro, Cosconati; Paolo, Grieco; Ettore, Novellino; Maddalena, Illario; Campiglia, Pietro; Isabel Gomez, Monterrey |
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