Sfoglia per Autore
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1)
2014-01-01 Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe
Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold
2015-01-01 Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors
2015-01-01 Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain
2015-01-01 Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis
Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) | 1-gen-2014 | Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold | 1-gen-2015 | Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors | 1-gen-2015 | Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain | 1-gen-2015 | Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines |
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