Sfoglia per Autore
Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery
2006-01-01 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi
Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives
2007-01-01 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate.
2007-01-01 Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B.
Synthesis of b-hydroxymalonates: the direct aldol addition of malonates to aldehydes in the presence of SiCl4 and i-Pr2EtN
2009-01-01 Massa, Antonio; Scettri, Arrigo; Filosa, Rosanna; Laura, Capozzolo
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride
2009-01-01 Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-basedx-acidic amino acids as glutamate receptors ligands
2009-01-01 Filosa, Rosanna; M., Carmela Fulco; Maura, Marinozzi; Nicola, Giacchè; Antonio, Macchiarulo; Peduto, Antonella; Massa, Antonio; DE CAPRARIIS, Paolo; Christian, Thomsen; Claus T., Christoffersen; Roberto, Pellicciari
Design, synthesis, biophysical and biological studies of trisubstitutednaphthalimides as G-quadruplex ligands
2011-01-01 Peduto, Antonella; Bruno, Pagano; Carmen, Petronzi; Massa, Antonio; Veronica, Esposito; Antonella, Virgilio; Francesco, Paduano; Francesco, Trapasso; Filomena, Fiorito; Salvatore, Florio; Concetta, Giancola; Aldo, Galeone; Filosa, Rosanna
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones
2011-01-01 Vijaykumar, More; DI MOLA, Antonia; Milena, Perillo; DE CAPRARIIS, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio
Multi-component, regio-selective aldol addition of b-ketoesters to aldehydes: scope and applications
2011-01-01 Vijaykumar, More; DI MOLA, Antonia; Gianluca, Croce; Tedesco, Consiglia; Carmen, Petronzi; Peduto, Antonella; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio
2,3-Dihydro-1,2-Diphenyl-substituted 4HPyridinone Derivatives as New Anti Flaviviridae Inhibitors
2011-01-01 Peduto, Antonella; Massa, Antonio; DI MOLA, Antonia; DE CAPRARIIS, Paolo; Paolo La, Colla; Roberta, Loddo; Sergio, Altamura; Giovanni, Maga; Filosa, Rosanna
Active methylene compounds in a very effective approach to 3-substitutedisobenzofuranones through tandem aldol/lactonization reactions
2012-01-01 Antonia Di, Mola; Gianluca, Croce; Vijaykumar, More; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio
Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures
2012-01-01 Carmen, Petronzi; Selene, Collarile; Gianluca, Croce; Filosa, Rosanna; DE CAPRARIIS, Paolo; Peduto, Antonella; Palombi, Laura; Valentina, Intintoli; Antonia Di, Mola; Massa, Antonio
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase
2013-01-01 Filosa, Rosanna; Peduto, Antonella; Polamarasetty, Aparoy; Anja M., Schaible; Susann, Luderer; Verena, Krauth; Carmen, Petronzi; Massa, Antonio; Mario de, Rosa; Pallu, Reddanna; Oliver, Werz
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series
2013-01-01 Virginia, Brancato; Peduto, Antonella; Stephen, Wharton; Stephen, Martin; Vijaykumar, More; DI MOLA, Antonia; Massa, Antonio; Brunella, Perfetto; Giovanna, Donnarumma; Chiara, Schiraldi; Maria Antonietta, Tufano; Mario de, Rosa; Filosa, Rosanna; Alan, Hay
3-Carboxylate Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions
2015-01-01 Scorzelli, Francesco; DI MOLA, Antonia; Palombi, Laura; Filosa, Rosanna; Massa, Antonio
Bifunctional Phase Transfer Catalysis in the Asymmetric Synthesis of Biologically Active Isoindolinones
2015-01-01 DI MOLA, Antonia; Tiffner, Maximilliam; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; DE CAPRARIIS, Paolo; Waser, Mario; Massa, Antonio
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture
2016-01-01 DI MOLA, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; DE CAPRARIIS, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna
Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication
2017-01-01 Scuotto, M.; Abdelnabi, R.; Collarile, Selene; Schiraldi, C.; Delang, L.; Massa, Antonio; Ferla, S.; Brancale, A.; Leyssen, P.; Neyts, J.; Filosa, Rosanna
Phenolics from Castanea sativa leaves and their effects on UVB-induced damage
2017-01-01 Cerulli, Antonietta; Masullo, Milena; Mari, Angela; Balato, Anna; Filosa, Rosanna; Lembo, Serena; Napolitano, Assunta; Piacente, Sonia
A systematic study on the use of different organocatalytic activation modes for asymmetric conjugated addition reactions of isoindolinones
2017-01-01 Scorzelli, Francesco; DI MOLA, Antonia; De Piano, F.; Tedesco, Consiglia; Palombi, Laura; Filosa, Rosanna; Waser, M.; Massa, Antonio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery | 1-gen-2006 | Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi | |
Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives | 1-gen-2007 | Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina | |
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate. | 1-gen-2007 | Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B. | |
Synthesis of b-hydroxymalonates: the direct aldol addition of malonates to aldehydes in the presence of SiCl4 and i-Pr2EtN | 1-gen-2009 | Massa, Antonio; Scettri, Arrigo; Filosa, Rosanna; Laura, Capozzolo | |
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride | 1-gen-2009 | Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo | |
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-basedx-acidic amino acids as glutamate receptors ligands | 1-gen-2009 | Filosa, Rosanna; M., Carmela Fulco; Maura, Marinozzi; Nicola, Giacchè; Antonio, Macchiarulo; Peduto, Antonella; Massa, Antonio; DE CAPRARIIS, Paolo; Christian, Thomsen; Claus T., Christoffersen; Roberto, Pellicciari | |
Design, synthesis, biophysical and biological studies of trisubstitutednaphthalimides as G-quadruplex ligands | 1-gen-2011 | Peduto, Antonella; Bruno, Pagano; Carmen, Petronzi; Massa, Antonio; Veronica, Esposito; Antonella, Virgilio; Francesco, Paduano; Francesco, Trapasso; Filomena, Fiorito; Salvatore, Florio; Concetta, Giancola; Aldo, Galeone; Filosa, Rosanna | |
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones | 1-gen-2011 | Vijaykumar, More; DI MOLA, Antonia; Milena, Perillo; DE CAPRARIIS, Paolo; Filosa, Rosanna; Peduto, Antonella; Massa, Antonio | |
Multi-component, regio-selective aldol addition of b-ketoesters to aldehydes: scope and applications | 1-gen-2011 | Vijaykumar, More; DI MOLA, Antonia; Gianluca, Croce; Tedesco, Consiglia; Carmen, Petronzi; Peduto, Antonella; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio | |
2,3-Dihydro-1,2-Diphenyl-substituted 4HPyridinone Derivatives as New Anti Flaviviridae Inhibitors | 1-gen-2011 | Peduto, Antonella; Massa, Antonio; DI MOLA, Antonia; DE CAPRARIIS, Paolo; Paolo La, Colla; Roberta, Loddo; Sergio, Altamura; Giovanni, Maga; Filosa, Rosanna | |
Active methylene compounds in a very effective approach to 3-substitutedisobenzofuranones through tandem aldol/lactonization reactions | 1-gen-2012 | Antonia Di, Mola; Gianluca, Croce; Vijaykumar, More; DE CAPRARIIS, Paolo; Filosa, Rosanna; Massa, Antonio | |
Synthesis and Reactivity of the 3-Substituted Isoindolinone Framework to Assemble Highly Functionalized Related Structures | 1-gen-2012 | Carmen, Petronzi; Selene, Collarile; Gianluca, Croce; Filosa, Rosanna; DE CAPRARIIS, Paolo; Peduto, Antonella; Palombi, Laura; Valentina, Intintoli; Antonia Di, Mola; Massa, Antonio | |
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase | 1-gen-2013 | Filosa, Rosanna; Peduto, Antonella; Polamarasetty, Aparoy; Anja M., Schaible; Susann, Luderer; Verena, Krauth; Carmen, Petronzi; Massa, Antonio; Mario de, Rosa; Pallu, Reddanna; Oliver, Werz | |
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series | 1-gen-2013 | Virginia, Brancato; Peduto, Antonella; Stephen, Wharton; Stephen, Martin; Vijaykumar, More; DI MOLA, Antonia; Massa, Antonio; Brunella, Perfetto; Giovanna, Donnarumma; Chiara, Schiraldi; Maria Antonietta, Tufano; Mario de, Rosa; Filosa, Rosanna; Alan, Hay | |
3-Carboxylate Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions | 1-gen-2015 | Scorzelli, Francesco; DI MOLA, Antonia; Palombi, Laura; Filosa, Rosanna; Massa, Antonio | |
Bifunctional Phase Transfer Catalysis in the Asymmetric Synthesis of Biologically Active Isoindolinones | 1-gen-2015 | DI MOLA, Antonia; Tiffner, Maximilliam; Scorzelli, Francesco; Palombi, Laura; Filosa, Rosanna; DE CAPRARIIS, Paolo; Waser, Mario; Massa, Antonio | |
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture | 1-gen-2016 | DI MOLA, Antonia; Gatta, Elena; Petronzi, Carmen; Cupello, Aroldo; DE CAPRARIIS, Paolo; Robello, Mauro; Massa, Antonio; Filosa, Rosanna | |
Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication | 1-gen-2017 | Scuotto, M.; Abdelnabi, R.; Collarile, Selene; Schiraldi, C.; Delang, L.; Massa, Antonio; Ferla, S.; Brancale, A.; Leyssen, P.; Neyts, J.; Filosa, Rosanna | |
Phenolics from Castanea sativa leaves and their effects on UVB-induced damage | 1-gen-2017 | Cerulli, Antonietta; Masullo, Milena; Mari, Angela; Balato, Anna; Filosa, Rosanna; Lembo, Serena; Napolitano, Assunta; Piacente, Sonia | |
A systematic study on the use of different organocatalytic activation modes for asymmetric conjugated addition reactions of isoindolinones | 1-gen-2017 | Scorzelli, Francesco; DI MOLA, Antonia; De Piano, F.; Tedesco, Consiglia; Palombi, Laura; Filosa, Rosanna; Waser, M.; Massa, Antonio |
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