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Phenol-derived CVFM analog inhibitors of ras farnesyltransferase possessing cellular in vitro activity. 1-gen-1998 Caliendo, G; Fiorino, F; Grieco, P; Perissutti, E; Ramunno, Anna; Santagada, V; Albrizio, S; Califano, D; Giuliano, A; Santelli, G.
Pyrrolobenzoxazepinone derivatives as non-nucleoside HIV-1 RT inhibitors: Further structure-activity relationship studies and identification of more potent broad-spectrum HIV-1 RT inhibitors with antiviral activity. 1-gen-1999 Campiani, G; Morelli, E; Fabbrini, M; Nacci, V; Greco, G; Novellino, E; Ramunno, Anna; Maga, G; Spadari, S; Caliendo, G; Bergamini, A; Faggioli, E; Uccella, I; Bolacchi, F; Marini, S; Coletta, M; Nacca, A; Caccia, S.
Characterization of the 1H-cyclopentapyrimidine-2,4(1H,3H)-dione derivative (S)-CPW399 as a novel, potent, and subtype-selective AMPA receptor full agonist with partial desensitization properties. 1-gen-2001 Campiani, G; Morelli, E; Nacci, V; Fattorusso, C; Ramunno, Anna; Novellino, E; Greenwood, J; Liljefors, T; Griffiths, R; Sinclair, C; Reavy, H; Kristensen, A. S.; Pickering, D. S.; Schousboe, A; Cagnotto, A; Fumagalli, E; Mennini, T.
Pyrrolo-1,5-benzoxazepines induce apoptosis in chronic myelogenous leukemia (CML) cells by bypassing the apoptotic suppressor Bcr-Abl. 1-gen-2001 MC GEE, M. M.; Campiani, G; Ramunno, Anna; Fattorusso, C; Nacci, V; Lawler, M; Williams, D. C.; Zisterer, D. M.
Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent. 1-gen-2001 Campiani, G; Aiello, F; Fabbrini, M; Morelli, E; Ramunno, Anna; Armaroli, S; Nacci, V; Garofalo, A; Greco, G; Novellino, E; Maga, G; Spadari, S; Bergamini, A; Ventura, L; Bongiovanni, B; Capozzi, M; Bolacchi, F; Marini, S; Coletta, M; Guiso, G; Caccia, S.
Pyrrolo-1,5-benzoxazepines: a new class of apoptotic agents. 1-gen-2001 ZISTERER D., M; MCGEE M., M; Campiani, G; Ramunno, Anna; Fattorusso, C; Nacci, V; Lawler, M; Williams, D. C.
The stereoselective targeting of a specific enzyme-substrate complex is the molecular mechanism for the synergic inhibition of HIV-1 reverse transcriptase by (R)-(-)-PPO464. A novel generation of nonnucleoside inhibitors. 1-gen-2001 Maga, G; Ramunno, Anna; Nacci, V; Locatelli, G; Spadari, S; Fiorini, I; Baldanti, F; Paolucci, S; Zavattoni, M; Bergamini, A; Galletti, B; Muck, S; Hubscher, U; Giorgi, G; Guiso, G; Caccia, S; Campiani, G.
A rational approach to the design of selective substrates and potent nontransportable inhibitors of the excitatory amino acid transporter EAAC1 (EAAT3). new glutamate and aspartate analogues as potential neuroprotective agents. 1-gen-2001 Campiani, G; DE ANGELIS, M; Armaroli, S; Fattorusso, C; Catalanotti, B; Ramunno, Anna; Nacci, V; Novellino, E; Grewer, C; Ionescu, D; Rauen, T; Griffiths, R; Sinclair, C; Fumagalli, E; Mennini, T.
Non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors: Past, present, and future perspectives. 1-gen-2002 Campiani, G; Ramunno, Anna; Maga, G; Nacci, V; Fattorusso, C; Catalanotti, B; Morelli, E; Novellino, E.
Caspase-3 is not essential for DNA fragmentation in MCF-7 cells during apoptosis induced by the pyrrolo-1,5-benzoxazepine, PBOX-6. 1-gen-2002 Mcgee, M. M.; Hyland, E; Campiani, G; Ramunno, Anna; Nacci, V; Zisterer, D. M.
Synthesis of New Molecular Probes for Investigation of Steroid Biosynthesis Induced by Selective Interaction with Peripheral Type Benzodiazepine Receptors (PBR). 1-gen-2002 Campiani, G; Ramunno, Anna; Fiorini, I; Nacci, V; Morelli, E; Novellino, E; Goegan, M; Mennini, T; Sullivan, S; ZISTERER D., M; Williams, C. D.
Activation of the c-Jun N-terminal kinase (JNK) signaling pathway is essential during PBOX-6-induced apoptosis in chronic myelogenous leukemia (CML) cells. 1-gen-2002 MC GEE, M. M.; Campiani, G; Ramunno, Anna; Nacci, V; Lawler, M; Williams, D. C.; Zisterer, D. M.
Inhibition of G1 cyclin-dependent kinase activity during growth arrest of human astrocytoma cells by the pyrrolo-1,5-benzoxazepine, PBOX-21. 1-gen-2003 Mulligan, J. M.; Campiani, G; Ramunno, Anna; Nacci, V; Zisterer, D. M.
Effects of drug resistance mutations L100I and V106A on the binding of pyrrolobenzoxazepinone nonnucleoside inhibitors to the human immunodeficiency virus type 1 reverse transcriptase catalytic complex. 1-gen-2004 Locatelli, Ga; Campiani, G; Cancio, R; Morelli, E; Ramunno, Anna; Gemma, S; Huebscher, U; Spadari, S; Maga, G.
3-(2-Aminoethyl)pyridine analogs as a4b2 nicotinic cholinergic receptor ligands. 1-gen-2005 Dukat, M; Ramunno, Anna; Banzi, R; Damaj, M. I.; Martin, B; Glennon, R. A.
Pyrrolo[1,5]benzoxa(thia)zepines as a New Class of Potent Apoptotic Agents. Biological Studies and Identification of an Intracellular Location of Their Drug Target. 1-gen-2005 Mcgee, ; Margaret, M.; Gemma, Sandra; Butini, Stefania; Ramunno, Anna; Zisterer, ; Daniela, M.; Fattorusso, Caterina; Catalanotti, Bruno; Kukreja, Gagan; Fiorini, Isabella; Pisano, Claudio; Cucco, Carla; Novellino, Ettore; Nacci, Vito; Williams, ; D., Clive; Campiani, Giuseppe
Specific Targeting Highly Conserved Residues in the HIV-1 Reverse Transcriptase Primer Grip Region. Design, Synthesis, and Biological Evaluation of Novel, Potent, and Broad Spectrum NNRTIs with Antiviral Activity 1-gen-2005 Fattorusso, Caterina; Gemma, Sandra; Butini, Stefania; Huleatt, Paul; Catalanotti, Bruno; Persico, Marco; De Angelis, Meri; Fiorini, Isabella; Nacci, Vito; Ramunno, Anna; Rodriquez, Manuela; Greco, Giovanni; Novellino, Ettore; Bergamini, Alberto; Marini, Stefano; Coletta, Massimo; Maga, Giovanni; Spadari, Silvio; Campiani, Giuseppe
6-(2-Phenylethyl)nicotine: A novel nicotinic cholinergic receptor ligand. 1-gen-2005 Ramunno, Anna; Dukat, M; Lee, M; Young, R; EL ZAHABI, M; Damaj, M. I.; Martin, B; Glennon, R. A.
Effect of flavonoids on A beta(25-35)/DLPC vesicle interaction. 1-gen-2008 D'Ursi, Anna Maria; Tedeschi, A.; Esposito, Cinzia; Scrima, Mario; Ramunno, Anna; D'Errico, G.; Lauro, M. R.; Aquino, R. P.
Antioxidant activity of diphenylpropionamide derivatives: synthesis, biologicalevaluation and computational analysis. 1-gen-2008 Urbani, P; Ramunno, Anna; Filosa, R; Pinto, Aldo; Popolo, Ada; Bianchino, E; PIOTTO PIOTTO, Stefano; Saturnino, Carmela; DE PRISCO, R; Nicolaus, B; Tommonaro, G.
Mostrati risultati da 1 a 20 di 48
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