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Synthesis, Conformational Analysis, and Cytotoxicity of New Analogues of the Natural Cyclodepsipeptide Jaspamide 1-gen-2004 Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Copper Jean, E.; Smith Charles, D.; GOMEZ PALOMA, Luigi; Riccio, Raffaele
Critical Surveys Covering the Year 2004:Total Synthesis of Natural Products 1-gen-2005 Bruno, Ines; P., Dambruoso; Terracciano, Stefania; Bifulco, Giuseppe
Synthesis, solution structure, and bioactivity of six new simplified analogues of the natural cyclodepsipeptide jaspamide 1-gen-2005 Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; E., Avallone; C. D., Smith; L., GOMEZ PALOMA; Riccio, Raffaele
Chemistry and Biology of Anti-Inflammatory Marine Natural Products.Phospholipase A2 Inhibitors 1-gen-2005 Luigi Gomez, Paloma; Monti, Maria Chiara; Terracciano, Stefania; Casapullo, Agostino; Riccio, Raffaele
Chemistry and biology of anti-inflammatory marine natural products: molecules interfering with cyclooxygenase, NF-κB and other unidentified targets 1-gen-2006 Terracciano, Stefania; Aquino, Maurizio; Rodriquez, Manuela; Monti, Maria Chiara; Casapullo, Agostino; Riccio, Raffaele; Gomez Paloma, Luigi
Total Synthesis, NMR Solution Structure, and Binding Model of the Potent Histone Deacetylase Inhibitor FR235222 1-gen-2006 Rodriquez, Manuela; Terracciano, Stefania; E., Cini; G., Settembrini; Bruno, Ines; Bifulco, Giuseppe; M., Taddei; L., GOMEZ PALOMA
Design and Synthesis of cyclopeptide analogues of the potent Histone deacetylase inhibitor FR235222 1-gen-2007 LUIGI GOMEZ, Paloma; Bruno, Ines; Elena, Cini; Saadi, Khochbin; Rodriquez, Manuela; Maurizio, Taddei; Terracciano, Stefania; AND KARIN, Sadoul
Synthetic and pharmacological studies on new simplified analogues of the potent actin-targeting Jaspamide 1-gen-2008 Terracciano, Stefania; Bruno, Ines; Elisabetta, D’Amico; Bifulco, Giuseppe; Angela, Zampella; Valentina, Sepe; Charles D., Smith; Riccio, Raffaele
Molecular modeling studies toward the structural optimization of new cyclopeptide-based HDAC inhibitors modeled on the natural product FR235222 1-gen-2008 DI MICCO, S; Terracciano, Stefania; Bruno, Ines; Rodriquez, Manuela; Riccio, Raffaele; Taddei, M; Bifulco, Giuseppe
Effects of FR235222, a novel HDAC inhibitor, in proliferation and apoptosis of human leukaemia cell lines: role of annexin A1 1-gen-2008 Petrella, Antonello; D'Acunto, Cw; Rodriquez, Manuela; Festa, M; Tosco, Alessandra; Bruno, Ines; Terracciano, Stefania; Taddei, M; Paloma, Lg; Parente, Luca
Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222 1-gen-2010 Terracciano, Stefania; DI MICCO, Simone; Bifulco, Giuseppe; Gallinari, P; Riccio, Raffaele; Bruno, Ines
Conformationally locked calixarene-based histone deacetylase inhibitors 1-gen-2010 Chini, MARIA GIOVANNA; Terracciano, Stefania; Riccio, Raffaele; Bifulco, Giuseppe; Ciao, Roberta; Gaeta, Carmine; Troisi, Francesco; Neri, Placido
Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors 1-gen-2010 Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors 1-gen-2012 Terracciano, Stefania; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors 1-gen-2013 Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Structural basis for the design and synthesis of selective HDAC inhibitors 1-gen-2013 DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
Design,virtual Screening and Synthesis of Potential Microsomal Prostaglandine E2 Synthase-1 (mPGES-1)Inhibitors 1-gen-2014 Foglia, Antonio; Simone Di, Micco; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 1-gen-2014 Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 1-gen-2015 Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
40 th "A. Corbella" International Summer School on Organic Synthesis - ISOS 2015 1-gen-2015 Foglia, Antonio; Di Micco, Simone; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Oppermann, Udo; Bifulco, Giuseppe; Bruno, Ines
Mostrati risultati da 1 a 20 di 53
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