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Mostrati risultati da 1 a 20 di 57
Titolo Data di pubblicazione Autore(i) File
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 1-gen-2007 Castellano, Sabrina; Milite, Ciro; Campiglia, Pietro; Sbardella, Gianluca
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 1-gen-2010 Tommy, Bui; Gloria Hernández, Torres; Milite, Ciro; Carlos F., Barbas
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 1-gen-2010 Castellano, Sabrina; Milite, Ciro; Ragno, R; Simeoni, S; Mai, A; Limongelli, V; Novellino, E; Bauer, I; Brosch, G; Spannhoff, A; Cheng, Dh; Bedford, Mt; Sbardella, Gianluca
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 1-gen-2011 Sbardella, Gianluca; Mai, Antonello; Bartolini, Sara; Castellano, Sabrina; Cirilli, Roberto; Rotili, Dante; Milite, Ciro; Santoriello, Marisabella; Orlando, Serena; Sciamanna, Ilaria; Serafino, Annalucia; Lavia, Patrizia; Spadafora, Corrado
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 1-gen-2011 Milite, Ciro; Castellano, Sabrina; Benedetti, Rosaria; Tosco, Alessandra; Ciliberti, Carmen; Vicidomini, Caterina; Boully, Ludovic; Franci, Gianluigi; Altucci, Lucia; Mai, Antonello; Sbardella, Gianluca
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 1-gen-2012 Castellano, Sabrina; Spannhoff, Astrid; Milite, Ciro; DAL PIAZ, Fabrizio; Cheng, Donghang; Tosco, Alessandra; Viviano, Monica; Yamani, Abdellah; Cianciulli, Agostino; Sala, Marina; Cura, Vincent; Cavarelli, Jean; Novellino, Ettore; Mai, Antonello; Bedford, Mark T.; Sbardella, Gianluca
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 1-gen-2012 Castellano, Sabrina; Sabrina, Taliani; Milite, Ciro; Isabella, Pugliesi; Eleonora Da, Pozzo; Elisa, Rizzetto; Sara, Bendinelli; Barbara, Costa; Sandro, Cosconati; Giovanni, Greco; Ettore, Novellino; Sbardella, Gianluca; Giorgio, Stefancich; Claudia, Martini; Federico Da, Settimo
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 1-gen-2012 Wei, Wei; Coelho, Carlos M.; Li, Xiang; Marek, Roger; Yan, Shanzhi; Anderson, Shawn; Meyers, David; Mukherjee, Chandrani; Sbardella, Gianluca; Castellano, Sabrina; Milite, Ciro; Rotili, Dante; Mai, Antonello; Cole, Philip A.; Sah, Pankaj; Kobor, Michael S.; Bredy, Timothy W.
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 1-gen-2012 De Nisco, Mauro; Manfra, Michele; Bolognese, Adele; Sofo, Adriano; Scopa, Antonio; Carlo Tenore, Gian; Pagano, Francesco; Milite, Ciro; Teresa Russo, Maria
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 1-gen-2012 Milite, Ciro; Viviano, Monica; Marisabella, Santoriello; Fabio, Arico`; Sbardella, Gianluca; Castellano, Sabrina
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 1-gen-2013 Vernieri, Ermelinda; Isabel Gomez, Monterrey; Milite, Ciro; Paolo, Grieco; Musella, Simona; Bertamino, Alessia; Ilaria, Scognamiglio; Stefano, Alcaro; Anna, Artese; Francesco, Ortuso; Ettore, Novellino; Sala, Marina; Campiglia, Pietro
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 1-gen-2013 Calabrese, ELENA CONCETTA; Castellano, Sabrina; M., Santoriello; C., Sgherri; M. F., Quartacci; L., Calucci; A. G. S., Warrilow; D. C., Lamb; S. L., Kelly; Milite, Ciro; Granata, Ilaria; Sbardella, Gianluca; G., Stefancich; Maresca, Bruno; Porta, Amalia
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 1-gen-2013 Sala, Marina; Adele, Chimento; Saturnino, Carmela; Isabel M., Gomez Monterrey; Musella, Simona; Bertamino, Alessia; Milite, Ciro; Maria Stefania, Sinicropi; Anna, Caruso; Rosa, Sirianni; Paolo, Tortorella; Ettore, Novellino; Campiglia, Pietro; Vincenzo, Pezzi
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 1-gen-2013 Yi, Zhang; Paolo Zanotti, Fregonara; Kimberly, Jenko; Robert L., Gladding; Sami S., Zoghbi; Masahiro, Fujita; Milite, Ciro; Castellano, Sabrina; Sabrina, Taliani; Claudia, Martini; Robert B., Innis; Federico Da, Settimo; Victor W., Pike
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 1-gen-2014 Milite, Ciro; Castellano, Sabrina; Feoli, Alessandra; La Pietra, Valeria; Cosconati, Sandro; Mai, Antonello; Sasaki, Kazuki; Yoshida, Minoru; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 1-gen-2014 Castellano, Sabrina; Sabrina, Taliani; Viviano, Monica; Milite, Ciro; Eleonora Da, Pozzo; Barbara, Costa; Elisabetta, Barresi; Agostino, Bruno; Sandro, Cosconati; Luciana, Marinelli; Giovanni, Greco; Ettore, Novellino; Sbardella, Gianluca; Federico Da, Settimo; Claudia, Martini
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 1-gen-2015 Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 1-gen-2015 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 1-gen-2015 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 1-gen-2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Mostrati risultati da 1 a 20 di 57
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