Sfoglia per Autore
Molecular Insights into Azumamide E Histone Deacetylases Inhibitory Activity
2007-01-01 Maulucci, N; Chini, MARIA GIOVANNA; DI MICCO, Simone; Izzo, Irene; Cafaro, E; Russo, A; Gallinari, P; Paolini, C; Nardi, M. C; Casapullo, Agostino; Riccio, Raffaele; Bifulco, Giuseppe; DE RICCARDIS, Francesco
Fibril aggregation inhibitory activity of the β-sheet breaker peptides: a molecular docking approach
2009-01-01 Chini, MARIA GIOVANNA; Scrima, Mario; D'Ursi, Anna Maria; Bifulco, Giuseppe
The molecular mechanism of human group IIA phospholipase A2 inactivation by bolinaquinone
2009-01-01 Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Conformationally locked calixarene-based histone deacetylase inhibitors
2010-01-01 Chini, MARIA GIOVANNA; Terracciano, Stefania; Riccio, Raffaele; Bifulco, Giuseppe; Ciao, Roberta; Gaeta, Carmine; Troisi, Francesco; Neri, Placido
A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry
2010-01-01 G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani
Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors
2010-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines
Quantum Mechanical Calculation of NMR Parameters in the Stereostructural Determination of Natural Products
2010-01-01 DI MICCO, Simone; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe
The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2.
2011-01-01 Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Theonellasterols and Conicasterols from Theonella swinhoei. Novel Marine Natural Ligands for Human Nuclear Receptors
2011-01-01 S., De Marino; R., Ummarino; M. V., D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; B., Renga; C., D’Amore; S., Fiorucci; C., Debitus; A., Zampella
Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents
2011-01-01 R., De Simone; Chini, MARIA GIOVANNA; Bruno, Ines; Riccio, Raffaele; D., Mueller; O., Werz; Bifulco, Giuseppe
The bile acid receptor GPBAR-1 (TGR5) modulates integrity of intestinal barrier and immune response to experimental Colitis.
2011-01-01 S., Cipriani; A., Mencarelli; Chini, MARIA GIOVANNA; E., Distrutti; B., Renga; Bifulco, Giuseppe; F., Baldelli; A., Donini; S., Fiorucci
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis
2012-01-01 Barbara, Renga; Andrea, Mencarelli; Claudio, D'Amore; Sabrina, Cipriani; Maria Valeria, D'Auria; Valentina, Sepe; Chini, MARIA GIOVANNA; Monti, Maria Chiara; Bifulco, Giuseppe; Angela, Zampella; Stefano, Fiorucci
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei
2012-01-01 Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Barbara, Renga; Claudio, D’Amore; Cécile, Debitus; Stefano, Fiorucci; Angela, Zampella
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity
2012-01-01 Simona De, Marino; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Claudio, D’Amore; Barbara, Renga; Andrea, Mencarelli; Sylvain, Petek; Stefano, Fiorucci; Angela, Zampella
Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90
2012-01-01 DAL PIAZ, Fabrizio; Vassallo, Antonio; Chini, MARIA GIOVANNA; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; Brandi, Alberto
Quantitative NMR-Derived Interproton Distances Combined with Quantum Mechanical Calculations of13C Chemical Shifts in the Stereochemical Determination of Conicasterol F, a Nuclear Receptor Ligand fromTheonella swinhoei
2012-01-01 Chini, MARIA GIOVANNA; Catharine R., Jones; Angela, Zampella; Maria Valeria, D’Auria; Barbara, Renga; Stefano, Fiorucci; Craig P., Butts; Bifulco, Giuseppe
Preliminary Structure-Activity Relationship on Theonellasterol, a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei
2012-01-01 Valentina, Sepe; Raffaella, Ummarino; Maria, D'Auria; Orazio Taglialatela, Scafati; Simona, Marino; Claudio, D'Amore; Barbara, Renga; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Yoichi, Nakao; Nobuhiro, Fusetani; Stefano, Fiorucci; Angela, Zampella
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors
2012-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial
2012-01-01 Margarucci, Luigi; Monti, Maria Chiara; Chini, MARIA GIOVANNA; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors
2012-01-01 Chini, MARIA GIOVANNA; Rosa De, Simone; Bruno, Ines; Riccio, Raffaele; Friederike, Dehm; Christina, Weinigel; Dagmar, Barz; Oliver, Werz; Bifulco, Giuseppe
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Molecular Insights into Azumamide E Histone Deacetylases Inhibitory Activity | 1-gen-2007 | Maulucci, N; Chini, MARIA GIOVANNA; DI MICCO, Simone; Izzo, Irene; Cafaro, E; Russo, A; Gallinari, P; Paolini, C; Nardi, M. C; Casapullo, Agostino; Riccio, Raffaele; Bifulco, Giuseppe; DE RICCARDIS, Francesco | |
Fibril aggregation inhibitory activity of the β-sheet breaker peptides: a molecular docking approach | 1-gen-2009 | Chini, MARIA GIOVANNA; Scrima, Mario; D'Ursi, Anna Maria; Bifulco, Giuseppe | |
The molecular mechanism of human group IIA phospholipase A2 inactivation by bolinaquinone | 1-gen-2009 | Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino | |
Conformationally locked calixarene-based histone deacetylase inhibitors | 1-gen-2010 | Chini, MARIA GIOVANNA; Terracciano, Stefania; Riccio, Raffaele; Bifulco, Giuseppe; Ciao, Roberta; Gaeta, Carmine; Troisi, Francesco; Neri, Placido | |
A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry | 1-gen-2010 | G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani | |
Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors | 1-gen-2010 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines | |
Quantum Mechanical Calculation of NMR Parameters in the Stereostructural Determination of Natural Products | 1-gen-2010 | DI MICCO, Simone; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe | |
The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2. | 1-gen-2011 | Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino | |
Theonellasterols and Conicasterols from Theonella swinhoei. Novel Marine Natural Ligands for Human Nuclear Receptors | 1-gen-2011 | S., De Marino; R., Ummarino; M. V., D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; B., Renga; C., D’Amore; S., Fiorucci; C., Debitus; A., Zampella | |
Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents | 1-gen-2011 | R., De Simone; Chini, MARIA GIOVANNA; Bruno, Ines; Riccio, Raffaele; D., Mueller; O., Werz; Bifulco, Giuseppe | |
The bile acid receptor GPBAR-1 (TGR5) modulates integrity of intestinal barrier and immune response to experimental Colitis. | 1-gen-2011 | S., Cipriani; A., Mencarelli; Chini, MARIA GIOVANNA; E., Distrutti; B., Renga; Bifulco, Giuseppe; F., Baldelli; A., Donini; S., Fiorucci | |
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis | 1-gen-2012 | Barbara, Renga; Andrea, Mencarelli; Claudio, D'Amore; Sabrina, Cipriani; Maria Valeria, D'Auria; Valentina, Sepe; Chini, MARIA GIOVANNA; Monti, Maria Chiara; Bifulco, Giuseppe; Angela, Zampella; Stefano, Fiorucci | |
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei | 1-gen-2012 | Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Barbara, Renga; Claudio, D’Amore; Cécile, Debitus; Stefano, Fiorucci; Angela, Zampella | |
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity | 1-gen-2012 | Simona De, Marino; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Claudio, D’Amore; Barbara, Renga; Andrea, Mencarelli; Sylvain, Petek; Stefano, Fiorucci; Angela, Zampella | |
Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90 | 1-gen-2012 | DAL PIAZ, Fabrizio; Vassallo, Antonio; Chini, MARIA GIOVANNA; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; Brandi, Alberto | |
Quantitative NMR-Derived Interproton Distances Combined with Quantum Mechanical Calculations of13C Chemical Shifts in the Stereochemical Determination of Conicasterol F, a Nuclear Receptor Ligand fromTheonella swinhoei | 1-gen-2012 | Chini, MARIA GIOVANNA; Catharine R., Jones; Angela, Zampella; Maria Valeria, D’Auria; Barbara, Renga; Stefano, Fiorucci; Craig P., Butts; Bifulco, Giuseppe | |
Preliminary Structure-Activity Relationship on Theonellasterol, a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei | 1-gen-2012 | Valentina, Sepe; Raffaella, Ummarino; Maria, D'Auria; Orazio Taglialatela, Scafati; Simona, Marino; Claudio, D'Amore; Barbara, Renga; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Yoichi, Nakao; Nobuhiro, Fusetani; Stefano, Fiorucci; Angela, Zampella | |
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors | 1-gen-2012 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial | 1-gen-2012 | Margarucci, Luigi; Monti, Maria Chiara; Chini, MARIA GIOVANNA; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino | |
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors | 1-gen-2012 | Chini, MARIA GIOVANNA; Rosa De, Simone; Bruno, Ines; Riccio, Raffaele; Friederike, Dehm; Christina, Weinigel; Dagmar, Barz; Oliver, Werz; Bifulco, Giuseppe |
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