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The Binding Mode of Petrosaspongiolide M to the Human Group IIA Phospholipase A2: Exploring the Role of Covalent and Noncovalent Interactions in the Inhibition Process 1-gen-2009 Monti, Maria Chiara; Casapullo, Agostino; CLAUDIO N., Cavasotto; Tosco, Alessandra; DAL PIAZ, Fabrizio; Arturas, Ziemys; Margarucci, Luigi; Riccio, Raffaele
Effects of Petrosapongiolide R on the Surface Topology of bee venom PLA2: a Limited Proteolysis and Mass Spectrometry Analysis 1-gen-2009 Monti, Maria Chiara; Riccio, Raffaele; Casapullo, Agostino
Perthamides C and D, two new potent anti-inflammatory cyclopeptides from a Solomon Lithistid sponge Theonella swinhoei 1-gen-2009 Carmen, Festa; Simona De, Marino; Valentina, Sepe; Monti, Maria Chiara; Paolo, Luciano; Maria Valeria, D'Auria; Cecile, Débitus; Mariarosaria, Bucci; Valentina, Vellecco; Angela, Zampella
Chemical Proteomics as a Tool in Target Discovery of BioactiveSmall Molecules 1-gen-2010 Margarucci, Luigi; Monti, Maria Chiara; Riccio, Raffaele; Casapullo, Agostino
Copper binds the carboxy-terminus of trefoil protein 1 (TFF1), favoring its homodimerization and motogenic activity 1-gen-2010 Tosco, Alessandra; Monti, Maria Chiara; Fontanella, Bianca; S., Montefusco; L., D'Andrea; B., Ziaco; Baldantoni, Daniela; M. C., Rio; Marzullo, Liberato
Bolinaquinone, a New Clathrin-Mediated Endocytosis Inhibitorby Chemical Proteomics 1-gen-2010 Margarucci, Luigi; Monti, Maria Chiara; Bianca, Fontanella; Riccio, Raffaele; Casapullo, Agostino
Chemical Proteomics Discloses Petrosapongiolide M, an Anti-Inflammatory Marine Sesterterpene, as a Proteasome Inhibitor 1-gen-2010 Margarucci, Luigi; Monti, Maria Chiara; Tosco, Alessandra; Riccio, Raffaele; Casapullo, Agostino
Structure-Based Design, Synthesis and Preliminary Anti-inflammatory Activity of Bolinaquinone Analogues 1-gen-2011 Petronzi, Carmen; R., Filosa; Peduto, Antonella; Monti, Maria Chiara; Margarucci, Luigi; Massa, Antonio; Ercolino, Simona Francesca; Bizzarro, Valentina; Parente, Luca; Riccio, Raffaele; DE CAPRARIIS, Paolo
Native mass spectrometry provides direct evidence for DNA mismatch-induced regulation of asymmetric nucleotide binding in mismatch repair protein MutS 1-gen-2011 Monti, Maria Chiara; S. X., Cohen; A., Fish; H. H. K., Winterwerp; A., Barendregt; P., Friedhoff; A., Perrakis; A. J. R., Heck; T. K., Sixma; R. H. H., van den Heuvel; J. H. G., Lebbink
The nuclear receptor FXR regulates hepatic transport and metabolism of glutamine and glutamate BBA molecular basis of diseases 1-gen-2011 Barbara, Renga; Andrea, Mencarelli; Sabrina, Cipriani; Claudio, D’Amore; Angela, Zampella; Monti, Maria Chiara; Eleonora, Distrutti; Stefano, Fiorucci
The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2. 1-gen-2011 Monti, Maria Chiara; Chini, MARIA GIOVANNA; Margarucci, Luigi; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Chemical Proteomics Reveals Bolinaquinone as a Clathrin-Mediated Endocytosis Inhibitor 1-gen-2011 Margarucci, Luigi; Monti, Maria Chiara; Fontanella, Bianca; Riccio, Raffaele; Casapullo, Agostino
New insights on the interaction mechanism between tau protein and oleocanthal, an extra-virgin olive-oil bioactive component. 1-gen-2011 Monti, Maria Chiara; Margarucci, Luigi; Tosco, Alessandra; Riccio, Raffaele; Casapullo, Agostino
The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial 1-gen-2012 Margarucci, Luigi; Monti, Maria Chiara; Chini, MARIA GIOVANNA; Tosco, Alessandra; Riccio, Raffaele; Bifulco, Giuseppe; Casapullo, Agostino
Anti-inflammatory cyclopeptides from the marine sponge Theonella swinhoei 1-gen-2012 Carmen, Festa; Simona De, Marino; Maria Valeria, D’Auria; Monti, Maria Chiara; Mariarosaria, Bucci; Valentina, Vellecco; Cécile, Debitus; Angela, Zampella
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 1-gen-2012 Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela
Heat shock proteins as key biological targets of the marine natural cyclopeptide perthamide C 1-gen-2012 Margarucci, Luigi; Monti, Maria Chiara; Andrea, Mencarelli; Cassiano, Chiara; Stefano, Fiorucci; Riccio, Raffaele; Angela, Zampella; Casapullo, Agostino
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis 1-gen-2012 Barbara, Renga; Andrea, Mencarelli; Claudio, D'Amore; Sabrina, Cipriani; Maria Valeria, D'Auria; Valentina, Sepe; Chini, MARIA GIOVANNA; Monti, Maria Chiara; Bifulco, Giuseppe; Angela, Zampella; Stefano, Fiorucci
Modulation of Proteasome Machinery by Natural and Synthetic Analogues of the Marine Bioactive Compound Petrosaspongiolide M 1-gen-2012 Margarucci, Luigi; Tosco, Alessandra; Rosa De, Simone; Riccio, Raffaele; Monti, Maria Chiara; Casapullo, Agostino
Chemical Proteomics Reveals Heat Shock Protein 60 To Be the Main Cellular Target of the Marine Bioactive Sesterterpene Suvanine 1-gen-2012 Cassiano, Chiara; Monti, Maria Chiara; Carmen, Festa; Angela, Zampella; Riccio, Raffaele; Casapullo, Agostino
Mostrati risultati da 21 a 40 di 132
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