BALZANO, AMODIO LUCA
BALZANO, AMODIO LUCA
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach
2015-01-01 Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy
2017-01-01 Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY
2016-01-01 Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca
The emerging role of lysine methyltransferase SETD8 in human diseases
2016-01-01 Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca
Titolo | Data di pubblicazione | Autore(i) | File |
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A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy | 1-gen-2017 | Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca | |
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY | 1-gen-2016 | Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca | |
The emerging role of lysine methyltransferase SETD8 in human diseases | 1-gen-2016 | Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca |