GIORDANO, Assunta
GIORDANO, Assunta
Dipartimento di Farmacia/DIFARMA
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
2022-01-01 Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
An Alternative Approach to the Construction of N-Isoprenyl-Indole Moiety: a Novel Synthesis of Two Antifungal Indole Alkaloids
2002-01-01 Capozzo, D; DELLA SALA, Giorgio; Giordano, Assunta; Izzo, Irene; Spinella, Aldo
Discovery of new erbB4 inhibitors: Repositioning an orphan chemical library by inverse virtual screening
2018-01-01 Giordano, Assunta; Forte, Giovanni; Massimo, Luigia; Riccio, Raffaele; Bifulco, Giuseppe; Di Micco, Simone
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
2023-01-01 Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi
Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition
2019-01-01 Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C.; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH)
2024-01-01 Gazzillo, E.; Colarusso, E.; Giordano, A.; Chini, M. G.; Potenza, M.; Hofstetter, R. K.; Iorizzi, M.; Werz, O.; Lauro, G.; Bifulco, G.
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways
2021-01-01 Potenza, M.; Sciarretta, M.; Chini, M. G.; Saviano, A.; Maione, F.; D'Auria, M. V.; De Marino, S.; Giordano, A.; Hofstetter, R. K.; Festa, C.; Werz, O.; Bifulco, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis | 1-gen-2022 | Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G | |
An Alternative Approach to the Construction of N-Isoprenyl-Indole Moiety: a Novel Synthesis of Two Antifungal Indole Alkaloids | 1-gen-2002 | Capozzo, D; DELLA SALA, Giorgio; Giordano, Assunta; Izzo, Irene; Spinella, Aldo | |
Discovery of new erbB4 inhibitors: Repositioning an orphan chemical library by inverse virtual screening | 1-gen-2018 | Giordano, Assunta; Forte, Giovanni; Massimo, Luigia; Riccio, Raffaele; Bifulco, Giuseppe; Di Micco, Simone | |
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders | 1-gen-2023 | Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi | |
Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition | 1-gen-2019 | Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C.; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone | |
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) | 1-gen-2024 | Gazzillo, E.; Colarusso, E.; Giordano, A.; Chini, M. G.; Potenza, M.; Hofstetter, R. K.; Iorizzi, M.; Werz, O.; Lauro, G.; Bifulco, G. | |
Structure-based screening for the discovery of 1,2,4-oxadiazoles as promising hits for the development of new anti-inflammatory agents interfering with eicosanoid biosynthesis pathways | 1-gen-2021 | Potenza, M.; Sciarretta, M.; Chini, M. G.; Saviano, A.; Maione, F.; D'Auria, M. V.; De Marino, S.; Giordano, A.; Hofstetter, R. K.; Festa, C.; Werz, O.; Bifulco, G. |