Sarno, Giuliana
Sarno, Giuliana
Dipartimento di Farmacia/DIFARMA
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain
2022 Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca
Discovery of the First-in-Class Dual TSPO/Carbonic Anhydrase Modulators with Promising Neurotrophic Activity
2024 Poggetti, Valeria; Angeloni, Elisa; Germelli, Lorenzo; Natale, Benito; Waqas, Muhammad; Sarno, Giuliana; Angeli, Andrea; Daniele, Simona; Salerno, Silvia; Barresi, Elisabetta; Cosconati, Sandro; Castellano, Sabrina; Da Pozzo, Eleonora; Costa, Barbara; Supuran, Claudiu T.; Da Settimo, Federico; Taliani, Sabrina
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8
2024 Feoli, Alessandra; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor
2023 Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors
2023 Cipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors
2024 Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Chini, Maria Giovanna; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella, Gianluca
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain | 1-gen-2022 | Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca | |
Discovery of the First-in-Class Dual TSPO/Carbonic Anhydrase Modulators with Promising Neurotrophic Activity | 1-gen-2024 | Poggetti, Valeria; Angeloni, Elisa; Germelli, Lorenzo; Natale, Benito; Waqas, Muhammad; Sarno, Giuliana; Angeli, Andrea; Daniele, Simona; Salerno, Silvia; Barresi, Elisabetta; Cosconati, Sandro; Castellano, Sabrina; Da Pozzo, Eleonora; Costa, Barbara; Supuran, Claudiu T.; Da Settimo, Federico; Taliani, Sabrina | |
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 | 1-gen-2024 | Feoli, Alessandra; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor | 1-gen-2023 | Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca | |
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors | 1-gen-2023 | Cipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors | 1-gen-2024 | Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Chini, Maria Giovanna; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella, Gianluca |