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NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
2015-01-01 Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.
2015-01-01 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors
2018-01-01 Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G.
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
2016-01-01 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach
2017-01-01 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors
2015-01-01 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins
2017-01-01 Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.
2015-01-01 Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Discovery of new chemical probes for the MRG15 chromo domain.
2015-01-01 Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors
2018-01-01 Milite, C.; Feoli, A.; Rescigno, Donatella; Pisapia, Vincenzo; Cosconati, S.; Castellano, S.; Sbardella, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. | 1-gen-2015 | Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors | 1-gen-2018 | Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G. | |
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH | 1-gen-2016 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach | 1-gen-2017 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors | 1-gen-2015 | Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins | 1-gen-2017 | Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca | |
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. | 1-gen-2015 | Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
Discovery of new chemical probes for the MRG15 chromo domain. | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors | 1-gen-2018 | Milite, C.; Feoli, A.; Rescigno, Donatella; Pisapia, Vincenzo; Cosconati, S.; Castellano, S.; Sbardella, G. |
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- 2017 4
- 2016 2
- 2015 9
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