Sfoglia per Autore
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds
2011 Lauro, Gianluigi; A., Romano; Riccio, Raffaele; Bifulco, Giuseppe
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist
2012 Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, Dauria; Lauro, Gianluigi; Bifulco, Giuseppe; Claudio, D'Amore; Barbara, Renga; Stefano, Fiorucci; Angela, Zampella
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor
2012 Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A.
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ
2012 Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds
2012 Lauro, Gianluigi; Masullo, Milena; Piacente, Sonia; Riccio, Raffaele; Bifulco, Giuseppe
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells
2013 DAL PIAZ, Fabrizio; Cotugno, Roberta; Lepore, Laura; Vassallo, Antonio; Malafronte, Nicola; Lauro, Gianluigi; Bifulco, Giuseppe; Belisario, MARIA ANTONIETTA; DE TOMMASI, Nunziatina
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists
2013 Festa, Carmen; D'Amore, Claudio; Renga, Barbara; Lauro, Gianluigi; De Marino, Simona; D'Auria, Maria Valeria; Bifulco, Giuseppe; Zampella, Angela; Fiorucci, Stefano
New techniques of molecular modelling and structural chemistry for the development of bioactive compounds
2013 Lauro, Gianluigi
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum
2014 Suvd, Nadmid; Alberto, Plaza; Lauro, Gianluigi; Ronald, Garcia; Bifulco, Giuseppe; Rolf, Müller
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1)
2014 Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines
2014 Syed Nasir Abbas, Bukhari; Lauro, Gianluigi; Ibrahim, Jantan; Bifulco, Giuseppe; Muhammad Wahab, Amjad
Reranking docking poses using molecular simulations and approximate free energy methods
2014 Lauro, G.; Ferruz, N.; Fulle, S.; Harvey, M. J.; Finn, P. W.; De Fabritiis, G.
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase
2014 Scrima, Mario; Lauro, Gianluigi; Grimaldi, Manuela; Sara Di, Marino; Tosco, Alessandra; Picardi, Paola; Gazzerro, Patrizia; Riccio, Raffaele; Ettore, Novellino; Bifulco, Maurizio; Bifulco, Giuseppe; D'Ursi, Anna Maria
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei
2014 Jun, Gong; Peng, Sun; Nan, Jiang; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Tie Jun, Li; William H., Gerwick; Wen, Zhang
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs
2015 Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors
2015 Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs
2015 Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni"
2015 Masullo, Milena; Cantone, Vincenza; Cerulli, Antonietta; Lauro, Gianluigi; Messano, Francesco; Russo, Gian Luigi; Pizza, Cosimo; Bifulco, Giuseppe; Piacente, Sonia
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain
2015 Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride
2016 Sun, Peng; Yu, Qing; Li, Jiao; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Kurtán, Tibor; Mándi, Attila; Tang, Hua; Li, Tie Jun; Zhuang, Chun Lin; Gerwick, William H.; Zhang, Wen
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds | 1-gen-2011 | Lauro, Gianluigi; A., Romano; Riccio, Raffaele; Bifulco, Giuseppe | |
| Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist | 1-gen-2012 | Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, Dauria; Lauro, Gianluigi; Bifulco, Giuseppe; Claudio, D'Amore; Barbara, Renga; Stefano, Fiorucci; Angela, Zampella | |
| Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor | 1-gen-2012 | Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A. | |
| Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ | 1-gen-2012 | Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela | |
| Inverse Virtual Screening allows the discovery of the biological activity of natural compounds | 1-gen-2012 | Lauro, Gianluigi; Masullo, Milena; Piacente, Sonia; Riccio, Raffaele; Bifulco, Giuseppe | |
| Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells | 1-gen-2013 | DAL PIAZ, Fabrizio; Cotugno, Roberta; Lepore, Laura; Vassallo, Antonio; Malafronte, Nicola; Lauro, Gianluigi; Bifulco, Giuseppe; Belisario, MARIA ANTONIETTA; DE TOMMASI, Nunziatina | |
| Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists | 1-gen-2013 | Festa, Carmen; D'Amore, Claudio; Renga, Barbara; Lauro, Gianluigi; De Marino, Simona; D'Auria, Maria Valeria; Bifulco, Giuseppe; Zampella, Angela; Fiorucci, Stefano | |
| New techniques of molecular modelling and structural chemistry for the development of bioactive compounds | 14-mag-2013 | Lauro, Gianluigi | |
| Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum | 1-gen-2014 | Suvd, Nadmid; Alberto, Plaza; Lauro, Gianluigi; Ronald, Garcia; Bifulco, Giuseppe; Rolf, Müller | |
| Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) | 1-gen-2014 | Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
| Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines | 1-gen-2014 | Syed Nasir Abbas, Bukhari; Lauro, Gianluigi; Ibrahim, Jantan; Bifulco, Giuseppe; Muhammad Wahab, Amjad | |
| Reranking docking poses using molecular simulations and approximate free energy methods | 1-gen-2014 | Lauro, G.; Ferruz, N.; Fulle, S.; Harvey, M. J.; Finn, P. W.; De Fabritiis, G. | |
| Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase | 1-gen-2014 | Scrima, Mario; Lauro, Gianluigi; Grimaldi, Manuela; Sara Di, Marino; Tosco, Alessandra; Picardi, Paola; Gazzerro, Patrizia; Riccio, Raffaele; Ettore, Novellino; Bifulco, Maurizio; Bifulco, Giuseppe; D'Ursi, Anna Maria | |
| New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei | 1-gen-2014 | Jun, Gong; Peng, Sun; Nan, Jiang; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Tie Jun, Li; William H., Gerwick; Wen, Zhang | |
| Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs | 1-gen-2015 | Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors | 1-gen-2015 | Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs | 1-gen-2015 | Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" | 1-gen-2015 | Masullo, Milena; Cantone, Vincenza; Cerulli, Antonietta; Lauro, Gianluigi; Messano, Francesco; Russo, Gian Luigi; Pizza, Cosimo; Bifulco, Giuseppe; Piacente, Sonia | |
| 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain | 1-gen-2015 | Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
| Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride | 1-gen-2016 | Sun, Peng; Yu, Qing; Li, Jiao; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Kurtán, Tibor; Mándi, Attila; Tang, Hua; Li, Tie Jun; Zhuang, Chun Lin; Gerwick, William H.; Zhang, Wen |
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