Sfoglia per Autore
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds
2011-01-01 Lauro, Gianluigi; A., Romano; Riccio, Raffaele; Bifulco, Giuseppe
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds
2012-01-01 Lauro, Gianluigi; Masullo, Milena; Piacente, Sonia; Riccio, Raffaele; Bifulco, Giuseppe
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor
2012-01-01 Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A.
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist
2012-01-01 Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, Dauria; Lauro, Gianluigi; Bifulco, Giuseppe; Claudio, D'Amore; Barbara, Renga; Stefano, Fiorucci; Angela, Zampella
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ
2012-01-01 Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells
2013-01-01 DAL PIAZ, Fabrizio; Cotugno, Roberta; Lepore, Laura; Vassallo, Antonio; Malafronte, Nicola; Lauro, Gianluigi; Bifulco, Giuseppe; Belisario, MARIA ANTONIETTA; DE TOMMASI, Nunziatina
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists
2013-01-01 Festa, Carmen; D'Amore, Claudio; Renga, Barbara; Lauro, Gianluigi; De Marino, Simona; D'Auria, Maria Valeria; Bifulco, Giuseppe; Zampella, Angela; Fiorucci, Stefano
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum
2014-01-01 Suvd, Nadmid; Alberto, Plaza; Lauro, Gianluigi; Ronald, Garcia; Bifulco, Giuseppe; Rolf, Müller
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei
2014-01-01 Jun, Gong; Peng, Sun; Nan, Jiang; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Tie Jun, Li; William H., Gerwick; Wen, Zhang
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines
2014-01-01 Syed Nasir Abbas, Bukhari; Lauro, Gianluigi; Ibrahim, Jantan; Bifulco, Giuseppe; Muhammad Wahab, Amjad
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase
2014-01-01 Scrima, Mario; Lauro, Gianluigi; Grimaldi, Manuela; Sara Di, Marino; Tosco, Alessandra; Picardi, Paola; Gazzerro, Patrizia; Riccio, Raffaele; Ettore, Novellino; Bifulco, Maurizio; Bifulco, Giuseppe; D'Ursi, Anna Maria
Reranking docking poses using molecular simulations and approximate free energy methods
2014-01-01 Lauro, G.; Ferruz, N.; Fulle, S.; Harvey, M. J.; Finn, P. W.; De Fabritiis, G.
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1)
2014-01-01 Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs
2015-01-01 Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs
2015-01-01 Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni"
2015-01-01 Masullo, Milena; Cantone, Vincenza; Cerulli, Antonietta; Lauro, Gianluigi; Messano, Francesco; Russo, Gian Luigi; Pizza, Cosimo; Bifulco, Giuseppe; Piacente, Sonia
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors
2015-01-01 Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain
2015-01-01 Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis
Anti-inflammatory trends of new benzimidazole derivatives
2016-01-01 Bukhari, Syed Nasir Abbas; Lauro, Gianluigi; Jantan, Ibrahim; Chee, Chin Fei; Amjad, Muhammad Wahab; Bifulco, Giuseppe; Sher, Hassan; Abdullah, Iskandar; Rahman, Noorsaadah Abd
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme
2016-01-01 Lauro, Gianluigi; Tortorella, Paolo; Bertamino, Alessia; Ostacolo, Carmine; Koeberle, Andreas; Fischer, Katrin; Bruno, Ines; Terracciano, Stefania; Gomez Monterrey, Isabel Maria; Tauro, Marilena; Loiodice, Fulvio; Novellino, Ettore; Riccio, Raffaele; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds | 1-gen-2011 | Lauro, Gianluigi; A., Romano; Riccio, Raffaele; Bifulco, Giuseppe | |
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds | 1-gen-2012 | Lauro, Gianluigi; Masullo, Milena; Piacente, Sonia; Riccio, Raffaele; Bifulco, Giuseppe | |
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor | 1-gen-2012 | Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A. | |
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist | 1-gen-2012 | Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, Dauria; Lauro, Gianluigi; Bifulco, Giuseppe; Claudio, D'Amore; Barbara, Renga; Stefano, Fiorucci; Angela, Zampella | |
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ | 1-gen-2012 | Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela | |
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells | 1-gen-2013 | DAL PIAZ, Fabrizio; Cotugno, Roberta; Lepore, Laura; Vassallo, Antonio; Malafronte, Nicola; Lauro, Gianluigi; Bifulco, Giuseppe; Belisario, MARIA ANTONIETTA; DE TOMMASI, Nunziatina | |
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists | 1-gen-2013 | Festa, Carmen; D'Amore, Claudio; Renga, Barbara; Lauro, Gianluigi; De Marino, Simona; D'Auria, Maria Valeria; Bifulco, Giuseppe; Zampella, Angela; Fiorucci, Stefano | |
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum | 1-gen-2014 | Suvd, Nadmid; Alberto, Plaza; Lauro, Gianluigi; Ronald, Garcia; Bifulco, Giuseppe; Rolf, Müller | |
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei | 1-gen-2014 | Jun, Gong; Peng, Sun; Nan, Jiang; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Tie Jun, Li; William H., Gerwick; Wen, Zhang | |
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines | 1-gen-2014 | Syed Nasir Abbas, Bukhari; Lauro, Gianluigi; Ibrahim, Jantan; Bifulco, Giuseppe; Muhammad Wahab, Amjad | |
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase | 1-gen-2014 | Scrima, Mario; Lauro, Gianluigi; Grimaldi, Manuela; Sara Di, Marino; Tosco, Alessandra; Picardi, Paola; Gazzerro, Patrizia; Riccio, Raffaele; Ettore, Novellino; Bifulco, Maurizio; Bifulco, Giuseppe; D'Ursi, Anna Maria | |
Reranking docking poses using molecular simulations and approximate free energy methods | 1-gen-2014 | Lauro, G.; Ferruz, N.; Fulle, S.; Harvey, M. J.; Finn, P. W.; De Fabritiis, G. | |
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) | 1-gen-2014 | Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs | 1-gen-2015 | Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs | 1-gen-2015 | Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" | 1-gen-2015 | Masullo, Milena; Cantone, Vincenza; Cerulli, Antonietta; Lauro, Gianluigi; Messano, Francesco; Russo, Gian Luigi; Pizza, Cosimo; Bifulco, Giuseppe; Piacente, Sonia | |
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors | 1-gen-2015 | Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain | 1-gen-2015 | Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
Anti-inflammatory trends of new benzimidazole derivatives | 1-gen-2016 | Bukhari, Syed Nasir Abbas; Lauro, Gianluigi; Jantan, Ibrahim; Chee, Chin Fei; Amjad, Muhammad Wahab; Bifulco, Giuseppe; Sher, Hassan; Abdullah, Iskandar; Rahman, Noorsaadah Abd | |
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme | 1-gen-2016 | Lauro, Gianluigi; Tortorella, Paolo; Bertamino, Alessia; Ostacolo, Carmine; Koeberle, Andreas; Fischer, Katrin; Bruno, Ines; Terracciano, Stefania; Gomez Monterrey, Isabel Maria; Tauro, Marilena; Loiodice, Fulvio; Novellino, Ettore; Riccio, Raffaele; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile