Sfoglia per Autore
Synthesis, Pharmacokinetics and anticonvulsant activity of 7 – chlorokynurenic acid prodrugs
2000-01-01 F. P., Bonina; L., Arenare; R., Ippolito; G., Boatto; G., Battaglia; V., Bruno; DE CAPRARIIS, Paolo
Separation of optical antipodes of calcium antagonist drugs and in vitro and in vivo evaluation of the enantiomer stability and pharmacological activities by biochemical methods.
2000-01-01 DE CAPRARIIS, Paolo
In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of chetoprofen, naproxen and diclofenac
2001-01-01 Bonina, F; Puglia, C; Barbuzzi, T; DE CAPRARIIS, Paolo; Palagiano, F; RIMOLI M., G; Saia, A.
Separation and analysis of the pharmacologic properties of chiral dihydropyridines: comparative evaluation of optical isomers of amlodipine and lercanidipine.
2002-01-01 DE CAPRARIIS, Paolo; Giampiero, Boatto; Maria, Nieddu; Mauro, Cataldi; Daniela, Melisi; Salvatore, Amoroso
New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical prperties and skin permeation studies.
2002-01-01 F. P., Bonina; M. G., Rimoli; L. A., Vallone; M., Amato; C., Puglia; M., Ricci; DE CAPRARIIS, Paolo; F., Barbato
Synthesis and in vitro chemical and enzymatica stability of glycosil 3'-azido-3'-deoxythymidine derivatives as potential anti-HIV agents
2002-01-01 Bonina, F; Puglia, C; RIMOLI M., G; Avallone, L; Abbignente, E; Boatto, G; Neddu, M; Meli, R; Amorena, M; DE CAPRARIIS, Paolo
In vitro antioxidant and in vivo photoprotective effects of a lyophilized extract of Capparis spinosa L. buds
2002-01-01 Bonina, F.; Puglia, C.; Ventura, D.; Aquino, Rita Patrizia; Tortora, S.; Sacchi, A.; Saija, A.; Tomaino, A.; Pellegrino, M. L.; DE CAPRARIIS, Paolo
Glycosyl derivatives of dopamine and l-dopa as Anti-Parkinson prodrugs: Synthesis pharmacological activity and in vitro stability studies
2003-01-01 Bonina, F; Puglia, C; RIMOLI M., G; Melisi, D; Boatto, G; Neddu, M; Calignano, A; LA RANA, G; DE CAPRARIIS, Paolo
Enantiomeric separation by HPLC of 1,4-dihydropyridines with vancomycin as chiral sector
2003-01-01 Boatto, G; Nieddu, M; FAEDDA M., V; DE CAPRARIIS, Paolo
Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent.
2003-01-01 Saturnino, Carmela; M., Buonerba; G., Boatto; Pascale, Maria; Moltedo, Ornella; L., DE NAPOLI; D., Montesarchio; J. C., Lancelot; DE CAPRARIIS, Paolo
Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives.
2004-01-01 Pau, A; Asproni, B; Boatto, G; GRELLA G., E; DE CAPRARIIS, Paolo; Costantino, L; Pinna, G. A.
Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery
2006-01-01 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi
Antiproliferative triterpene saponins from Entada africana
2006-01-01 Cioffi, Giuseppina; DAL PIAZ, Fabrizio; DE CAPRARIIS, Paolo; P, ; Sanogo, R; Marzocco, Stefania; Autore, Giuseppina; DE TOMMASI, Nunziatina
Galactosyl Derivatives of L-Arginine and D-Arginine: Synthesis, Stability, Cell Permeation, and Nitric Oxide Production in Pituitary GH3 Cells
2006-01-01 Melisi, D; Secondo, A; Montoro, Paola; Piacente, Sonia; Rimoli, Mg; Minale, M; DE CAPRARIIS, Paolo; Annunziato, L.
Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives
2007-01-01 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate.
2007-01-01 Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B.
Galactosilated dopamine increases attention without reducing activity in C57BL/6 mice
2008-01-01 RUOCCO L., A; Viggiano, D; Pignatelli, M; Iannaccone, T; RIMOLI M., G; Melisi, D; Curcio, A; DE LUCIA, S; Carboni, E; CARNEVALE U. A., Gironi; DE CAPRARIIS, Paolo; Sadile, A. G.
Antiproliferative Oleanane Saponins from Meryta denhamii.
2008-01-01 Cioffi, Giuseppina; DAL PIAZ, Fabrizio; Vassallo, A; Venturella, F; DE CAPRARIIS, Paolo; DE SIMONE, F; DE TOMMASI, Nunziatina
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride
2009-01-01 Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo
Molecular modelling studies, synthesis and biological activity of a series of novelbisnaphthalimides and their development as new DNA topoisomeraseII inhibitors
2009-01-01 Filosa, Rosanna; Peduto, Antonella; DI MICCO, Simone; DE CAPRARIIS, Paolo; Festa, Michela; Petrella, Antonello; Giovanni, Capranico; Bifulco, Giuseppe
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis, Pharmacokinetics and anticonvulsant activity of 7 – chlorokynurenic acid prodrugs | 1-gen-2000 | F. P., Bonina; L., Arenare; R., Ippolito; G., Boatto; G., Battaglia; V., Bruno; DE CAPRARIIS, Paolo | |
Separation of optical antipodes of calcium antagonist drugs and in vitro and in vivo evaluation of the enantiomer stability and pharmacological activities by biochemical methods. | 1-gen-2000 | DE CAPRARIIS, Paolo | |
In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of chetoprofen, naproxen and diclofenac | 1-gen-2001 | Bonina, F; Puglia, C; Barbuzzi, T; DE CAPRARIIS, Paolo; Palagiano, F; RIMOLI M., G; Saia, A. | |
Separation and analysis of the pharmacologic properties of chiral dihydropyridines: comparative evaluation of optical isomers of amlodipine and lercanidipine. | 1-gen-2002 | DE CAPRARIIS, Paolo; Giampiero, Boatto; Maria, Nieddu; Mauro, Cataldi; Daniela, Melisi; Salvatore, Amoroso | |
New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical prperties and skin permeation studies. | 1-gen-2002 | F. P., Bonina; M. G., Rimoli; L. A., Vallone; M., Amato; C., Puglia; M., Ricci; DE CAPRARIIS, Paolo; F., Barbato | |
Synthesis and in vitro chemical and enzymatica stability of glycosil 3'-azido-3'-deoxythymidine derivatives as potential anti-HIV agents | 1-gen-2002 | Bonina, F; Puglia, C; RIMOLI M., G; Avallone, L; Abbignente, E; Boatto, G; Neddu, M; Meli, R; Amorena, M; DE CAPRARIIS, Paolo | |
In vitro antioxidant and in vivo photoprotective effects of a lyophilized extract of Capparis spinosa L. buds | 1-gen-2002 | Bonina, F.; Puglia, C.; Ventura, D.; Aquino, Rita Patrizia; Tortora, S.; Sacchi, A.; Saija, A.; Tomaino, A.; Pellegrino, M. L.; DE CAPRARIIS, Paolo | |
Glycosyl derivatives of dopamine and l-dopa as Anti-Parkinson prodrugs: Synthesis pharmacological activity and in vitro stability studies | 1-gen-2003 | Bonina, F; Puglia, C; RIMOLI M., G; Melisi, D; Boatto, G; Neddu, M; Calignano, A; LA RANA, G; DE CAPRARIIS, Paolo | |
Enantiomeric separation by HPLC of 1,4-dihydropyridines with vancomycin as chiral sector | 1-gen-2003 | Boatto, G; Nieddu, M; FAEDDA M., V; DE CAPRARIIS, Paolo | |
Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent. | 1-gen-2003 | Saturnino, Carmela; M., Buonerba; G., Boatto; Pascale, Maria; Moltedo, Ornella; L., DE NAPOLI; D., Montesarchio; J. C., Lancelot; DE CAPRARIIS, Paolo | |
Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives. | 1-gen-2004 | Pau, A; Asproni, B; Boatto, G; GRELLA G., E; DE CAPRARIIS, Paolo; Costantino, L; Pinna, G. A. | |
Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery | 1-gen-2006 | Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi | |
Antiproliferative triterpene saponins from Entada africana | 1-gen-2006 | Cioffi, Giuseppina; DAL PIAZ, Fabrizio; DE CAPRARIIS, Paolo; P, ; Sanogo, R; Marzocco, Stefania; Autore, Giuseppina; DE TOMMASI, Nunziatina | |
Galactosyl Derivatives of L-Arginine and D-Arginine: Synthesis, Stability, Cell Permeation, and Nitric Oxide Production in Pituitary GH3 Cells | 1-gen-2006 | Melisi, D; Secondo, A; Montoro, Paola; Piacente, Sonia; Rimoli, Mg; Minale, M; DE CAPRARIIS, Paolo; Annunziato, L. | |
Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives | 1-gen-2007 | Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina | |
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate. | 1-gen-2007 | Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B. | |
Galactosilated dopamine increases attention without reducing activity in C57BL/6 mice | 1-gen-2008 | RUOCCO L., A; Viggiano, D; Pignatelli, M; Iannaccone, T; RIMOLI M., G; Melisi, D; Curcio, A; DE LUCIA, S; Carboni, E; CARNEVALE U. A., Gironi; DE CAPRARIIS, Paolo; Sadile, A. G. | |
Antiproliferative Oleanane Saponins from Meryta denhamii. | 1-gen-2008 | Cioffi, Giuseppina; DAL PIAZ, Fabrizio; Vassallo, A; Venturella, F; DE CAPRARIIS, Paolo; DE SIMONE, F; DE TOMMASI, Nunziatina | |
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride | 1-gen-2009 | Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo | |
Molecular modelling studies, synthesis and biological activity of a series of novelbisnaphthalimides and their development as new DNA topoisomeraseII inhibitors | 1-gen-2009 | Filosa, Rosanna; Peduto, Antonella; DI MICCO, Simone; DE CAPRARIIS, Paolo; Festa, Michela; Petrella, Antonello; Giovanni, Capranico; Bifulco, Giuseppe |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile