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Titolo Data di pubblicazione Autore(i) File
Synthesis, Pharmacokinetics and anticonvulsant activity of 7 – chlorokynurenic acid prodrugs 1-gen-2000 F. P., Bonina; L., Arenare; R., Ippolito; G., Boatto; G., Battaglia; V., Bruno; DE CAPRARIIS, Paolo
Separation of optical antipodes of calcium antagonist drugs and in vitro and in vivo evaluation of the enantiomer stability and pharmacological activities by biochemical methods. 1-gen-2000 DE CAPRARIIS, Paolo
In vitro and in vivo evaluation of polyoxyethylene esters as dermal prodrugs of chetoprofen, naproxen and diclofenac 1-gen-2001 Bonina, F; Puglia, C; Barbuzzi, T; DE CAPRARIIS, Paolo; Palagiano, F; RIMOLI M., G; Saia, A.
Separation and analysis of the pharmacologic properties of chiral dihydropyridines: comparative evaluation of optical isomers of amlodipine and lercanidipine. 1-gen-2002 DE CAPRARIIS, Paolo; Giampiero, Boatto; Maria, Nieddu; Mauro, Cataldi; Daniela, Melisi; Salvatore, Amoroso
New oligoethylene ester derivatives of 5-iodo-2'-deoxyuridine as dermal prodrugs: synthesis, physicochemical prperties and skin permeation studies. 1-gen-2002 F. P., Bonina; M. G., Rimoli; L. A., Vallone; M., Amato; C., Puglia; M., Ricci; DE CAPRARIIS, Paolo; F., Barbato
Synthesis and in vitro chemical and enzymatica stability of glycosil 3'-azido-3'-deoxythymidine derivatives as potential anti-HIV agents 1-gen-2002 Bonina, F; Puglia, C; RIMOLI M., G; Avallone, L; Abbignente, E; Boatto, G; Neddu, M; Meli, R; Amorena, M; DE CAPRARIIS, Paolo
In vitro antioxidant and in vivo photoprotective effects of a lyophilized extract of Capparis spinosa L. buds 1-gen-2002 Bonina, F.; Puglia, C.; Ventura, D.; Aquino, Rita Patrizia; Tortora, S.; Sacchi, A.; Saija, A.; Tomaino, A.; Pellegrino, M. L.; DE CAPRARIIS, Paolo
Glycosyl derivatives of dopamine and l-dopa as Anti-Parkinson prodrugs: Synthesis pharmacological activity and in vitro stability studies 1-gen-2003 Bonina, F; Puglia, C; RIMOLI M., G; Melisi, D; Boatto, G; Neddu, M; Calignano, A; LA RANA, G; DE CAPRARIIS, Paolo
Enantiomeric separation by HPLC of 1,4-dihydropyridines with vancomycin as chiral sector 1-gen-2003 Boatto, G; Nieddu, M; FAEDDA M., V; DE CAPRARIIS, Paolo
Synthesis and preliminary biological evaluation of a new pyridocarbazole derivative covalently linked to a thymidine nucleoside as a potential targeted antitumoral agent. 1-gen-2003 Saturnino, Carmela; M., Buonerba; G., Boatto; Pascale, Maria; Moltedo, Ornella; L., DE NAPOLI; D., Montesarchio; J. C., Lancelot; DE CAPRARIIS, Paolo
Synthesis and aldose reductase inhibitory activities of novel thienocinnolinone derivatives. 1-gen-2004 Pau, A; Asproni, B; Boatto, G; GRELLA G., E; DE CAPRARIIS, Paolo; Costantino, L; Pinna, G. A.
Evaluation of Alternative Strategies to Optimize Ketorolac TransdermalDelivery 1-gen-2006 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Luisa, Rizza; Francesco, Bonina; Paolo, Blasi
Antiproliferative triterpene saponins from Entada africana 1-gen-2006 Cioffi, Giuseppina; DAL PIAZ, Fabrizio; DE CAPRARIIS, Paolo; P, ; Sanogo, R; Marzocco, Stefania; Autore, Giuseppina; DE TOMMASI, Nunziatina
Galactosyl Derivatives of L-Arginine and D-Arginine: Synthesis, Stability, Cell Permeation, and Nitric Oxide Production in Pituitary GH3 Cells 1-gen-2006 Melisi, D; Secondo, A; Montoro, Paola; Piacente, Sonia; Rimoli, Mg; Minale, M; DE CAPRARIIS, Paolo; Annunziato, L.
Synthesis, Physicochemical Propertiesand In Vitro Permeation Studies of New Ketorolac Ester Derivatives 1-gen-2007 Carmelo, Puglia; Filosa, Rosanna; Peduto, Antonella; DE CAPRARIIS, Paolo; Gianpiero, Boatto; Maria, Nieddu; Natale Alfredo, Santagati; Francesco, Bonina
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate. 1-gen-2007 Dalpiaz, A; Filosa, Rosanna; DE CAPRARIIS, Paolo; Conte, G; Bortolotti, F; Biondi, C; Scatturin, A; Prasad, Pd; Pavan, B.
Galactosilated dopamine increases attention without reducing activity in C57BL/6 mice 1-gen-2008 RUOCCO L., A; Viggiano, D; Pignatelli, M; Iannaccone, T; RIMOLI M., G; Melisi, D; Curcio, A; DE LUCIA, S; Carboni, E; CARNEVALE U. A., Gironi; DE CAPRARIIS, Paolo; Sadile, A. G.
Antiproliferative Oleanane Saponins from Meryta denhamii. 1-gen-2008 Cioffi, Giuseppina; DAL PIAZ, Fabrizio; Vassallo, A; Venturella, F; DE CAPRARIIS, Paolo; DE SIMONE, F; DE TOMMASI, Nunziatina
A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels–Alder Reaction Promoted by Silicon Tetrachloride 1-gen-2009 Massa, Antonio; DE SIO, Vincenzo; Villano, Rosaria; Acocella, MARIA ROSARIA; Palombi, Laura; Giusi, Sellitto; Peduto, Antonella; Filosa, Rosanna; DE CAPRARIIS, Paolo; Scettri, Arrigo
Molecular modelling studies, synthesis and biological activity of a series of novelbisnaphthalimides and their development as new DNA topoisomeraseII inhibitors 1-gen-2009 Filosa, Rosanna; Peduto, Antonella; DI MICCO, Simone; DE CAPRARIIS, Paolo; Festa, Michela; Petrella, Antonello; Giovanni, Capranico; Bifulco, Giuseppe
Mostrati risultati da 21 a 40 di 62
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