Pierri, Martina
Pierri, Martina
Dipartimento di Farmacia/DIFARMA
Identification of 2,4-Dinitro-Biphenyl-Based Compounds as MAPEG Inhibitors
2022 Di Micco, Simone; Terracciano, Stefania; Pierri, Martina; Cantone, Vincenza; Liening, Stefanie; König, Stefanie; Garscha, Ulrike; Hofstetter, Robert Klaus; Koeberle, Andreas; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders
2024 Colarusso, E.; Gazzillo, E.; Pierri, M.; Ruggiero, D.; Chini, M. G.; Bruno, I.; Bifulco, G.; Terracciano, S.; Lauro, G.
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders
2022 Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G.
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation
2024 Aliberti, Michela; Pierri, Martina; Terracciano, Stefania; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Identification of 2,4-Dinitro-Biphenyl-Based Compounds as MAPEG Inhibitors | 1-gen-2022 | Di Micco, Simone; Terracciano, Stefania; Pierri, Martina; Cantone, Vincenza; Liening, Stefanie; König, Stefanie; Garscha, Ulrike; Hofstetter, Robert Klaus; Koeberle, Andreas; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe | |
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders | 1-gen-2024 | Colarusso, E.; Gazzillo, E.; Pierri, M.; Ruggiero, D.; Chini, M. G.; Bruno, I.; Bifulco, G.; Terracciano, S.; Lauro, G. | |
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders | 1-gen-2022 | Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G. | |
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation | 1-gen-2024 | Aliberti, Michela; Pierri, Martina; Terracciano, Stefania; Giovanna Chini, Maria; Bifulco, Giuseppe; Lauro, Gianluigi |