GAZZILLO, ERICA
GAZZILLO, ERICA
Dipartimento di Farmacia/DIFARMA
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
2022-01-01 Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9
2023-01-01 Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
2023-01-01 Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders
2022-01-01 Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G.
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation
2022-01-01 Gazzillo, Erica; Terracciano, Stefania; Ruggiero, Dafne; Potenza, Marianna; Chini, Maria Giovanna; Lauro, Gianluigi; Fischer, Katrin; Hofstetter, Robert Klaus; Giordano, Assunta; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis | 1-gen-2022 | Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G | |
| Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 | 1-gen-2023 | Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi | |
| Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders | 1-gen-2023 | Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi | |
| Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders | 1-gen-2022 | Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G. | |
| Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation | 1-gen-2022 | Gazzillo, Erica; Terracciano, Stefania; Ruggiero, Dafne; Potenza, Marianna; Chini, Maria Giovanna; Lauro, Gianluigi; Fischer, Katrin; Hofstetter, Robert Klaus; Giordano, Assunta; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe |