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Prodotti della tipologia (ordinati per Data di deposito in Decrescente ordine): 1 a 20 di 333
| Titolo | Data di deposito | Autore(i) |
|---|---|---|
| Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors | 14-dic-2018 | Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G. |
| Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors | 14-dic-2018 | Milite, C.; Feoli, A.; Rescigno, D.; Pisapia, V.; Cosconati, S.; Castellano, S.; Sbardella, G. |
| Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins | 14-dic-2018 | Cipriano, Alessandra; Milite, Ciro; Filippakopoulos, Panagis; Castellano, Sabrina; Sbardella, Gianluca |
| Identification of new KDM4 inhibitors through a HTS and hit refinement strategy | 14-dic-2018 | Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach | 14-dic-2018 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach | 14-dic-2018 | Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH | 14-dic-2018 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca |
| IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY | 14-dic-2018 | Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors | 11-dic-2018 | Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca |
| Discovery of new chemical probes for the MRG15 chromo domain. | 11-dic-2018 | Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 | 11-dic-2018 | Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors | 11-dic-2018 | Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, Maria Giovanna; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. | 11-dic-2018 | Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. | 11-dic-2018 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. | 11-dic-2018 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. | 11-dic-2018 | Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. | 11-dic-2018 | Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina |
| Sunset. Belong to nature | 7-dic-2018 | Cucco, Pasquale |
| Zero, bellezza senza sprechi | 7-dic-2018 | Cucco, Pasquale; Giuditta, Serena |
| A potential estimates approach to a priori estimates for elliptic equations | 18-nov-2018 | Mamedov, Farman; Monsurro', Sara; Transirico, Maria |
Prodotti della tipologia (ordinati per Data di deposito in Decrescente ordine): 1 a 20 di 333
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Per tipologia
Data di pubblicazione
- 232 2010 - 2018
- 76 2000 - 2009
- 17 1990 - 1999
- 8 1983 - 1989
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- 3 eng
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