Sfoglia per Autore
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction.
2008-01-01 Castellano, Sabrina; Bertamino, Alessia; Gomez Monterrey, Isabel; Santoriello, Marisabella; Grieco, Paolo; Campiglia, Pietro; Sbardella, Gianluca; Novellino, Ettore
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases
2009-01-01 Mai, A; Rotili, D; Tarantino, D; Nebbioso, A; Castellano, Sabrina; Sbardella, Gianluca; Tini, M; Altucci, L.
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems
2009-01-01 Castellano, Sabrina; Santoriello, Marisabella; Campiglia, Pietro; Cardillo, Giovanna; Bertamino, Alessia; Gomez Monterrey, Isabel; Novellino, Ettore; Sbardella, Gianluca
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters
2010-01-01 Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Nicoletta De, Simone; Sala, Marina; Castellano, Sabrina; Marisabella, Santoriello; Paolo, Grieco; Ettore, Novellino; Isabel Maria Gomez, Monterrey
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1)
2010-01-01 Castellano, Sabrina; Milite, Ciro; Ragno, R; Simeoni, S; Mai, A; Limongelli, V; Novellino, E; Bauer, I; Brosch, G; Spannhoff, A; Cheng, Dh; Bedford, Mt; Sbardella, Gianluca
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies.
2010-01-01 Castellano, Sabrina; Lucia, Tamborini; Viviano, Monica; Andrea, Pinto; Sbardella, Gianluca; Paola, Conti
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators
2011-01-01 DAL PIAZ, Fabrizio; Vassallo, Antonio; Cuesta Rubio, Osmany; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina
Chemical biology of Histone acetyltransferase natural compounds modulators.
2011-01-01 DAL PIAZ, Fabrizio; Vassallo, Antonio; Osmany Cuesta, Rubio; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors
2011-01-01 Castellano, Sabrina; Dirk, Kuck; Viviano, Monica; Jakyung, Yoo; Fabian López, Vallejo; Paola, Conti; Lucia, Tamborini; Andrea, Pinto; José L., Medina Franco; Sbardella, Gianluca
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents
2011-01-01 Wang, Zhiming; Castellano, Sabrina; Kinderman, Sape S.; Argueta, Christian E.; Beshir, Anwar B.; Fenteany, Gabriel; Kwon, Ohyun
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity.
2011-01-01 Donghang, Cheng; Sergio, Valente; Castellano, Sabrina; Sbardella, Gianluca; Roberto Di, Santo; Roberta, Costi; Mark T., Bedford; Antonello, Mai
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs)
2011-01-01 Milite, Ciro; Castellano, Sabrina; Benedetti, Rosaria; Tosco, Alessandra; Ciliberti, Carmen; Vicidomini, Caterina; Boully, Ludovic; Franci, Gianluigi; Altucci, Lucia; Mai, Antonello; Sbardella, Gianluca
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart
2011-01-01 Claudia, Colussi; Jessica, Rosati; Stefania, Straino; Francesco, Spallotta; Roberta, Berni; Donatella, Stilli; Stefano, Rossi; Ezio, Musso; Emilio, Macchi; Antonello, Mai; Sbardella, Gianluca; Castellano, Sabrina; Cristina, Chimenti; Andrea, Frustaci; Angela, Nebbioso; Lucia, Altucci; Maurizio C., Capogrossi; Carlo, Gaetano
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees.
2011-01-01 Astrid, Spannhoff; Yong Kee, Kim; Noel J. M., Raynal; Vazganush, Gharibyan; Ming Bo, Su; Yue Yang, Zhou; Jia, Li; Castellano, Sabrina; Sbardella, Gianluca; Jean Pierre J., Issa; Mark T., Bedford
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors.
2011-01-01 Sbardella, Gianluca; Mai, Antonello; Bartolini, Sara; Castellano, Sabrina; Cirilli, Roberto; Rotili, Dante; Milite, Ciro; Santoriello, Marisabella; Orlando, Serena; Sciamanna, Ilaria; Serafino, Annalucia; Lavia, Patrizia; Spadafora, Corrado
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients
2011-01-01 M., Vecellio; G., Pompilio; F., Spallotta; C., Colussi; Sbardella, Gianluca; Castellano, Sabrina; A., Mai; M. C., Capogrossi; A., Rossini; C., Gaetano
Microbiologia Molecolare e Cellulare
2012-01-01 Maresca, Bruno; Castellano, Sabrina; Fortino, Vittorio; Morello, Silvana; Porta, Amalia
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins
2012-01-01 Colussi, Claudia); Scopece, Alessandro; Vitale, Serena; Spallotta, Francesco; Mattiussi, Stefania; Rosati, Jessica; Illi, Barbara; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca; Farsetti, Antonella; Capogrossi, Maurizio C.; Gaetano, Carlo
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear
2012-01-01 Wei, Wei; Coelho, Carlos M.; Li, Xiang; Marek, Roger; Yan, Shanzhi; Anderson, Shawn; Meyers, David; Mukherjee, Chandrani; Sbardella, Gianluca; Castellano, Sabrina; Milite, Ciro; Rotili, Dante; Mai, Antonello; Cole, Philip A.; Sah, Pankaj; Kobor, Michael S.; Bredy, Timothy W.
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds
2012-01-01 Granata, Ilaria; Castellano, Sabrina; Armenante, Annunziata; Maresca, Bruno; Porta, Amalia
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. | 1-gen-2008 | Castellano, Sabrina; Bertamino, Alessia; Gomez Monterrey, Isabel; Santoriello, Marisabella; Grieco, Paolo; Campiglia, Pietro; Sbardella, Gianluca; Novellino, Ettore | |
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases | 1-gen-2009 | Mai, A; Rotili, D; Tarantino, D; Nebbioso, A; Castellano, Sabrina; Sbardella, Gianluca; Tini, M; Altucci, L. | |
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems | 1-gen-2009 | Castellano, Sabrina; Santoriello, Marisabella; Campiglia, Pietro; Cardillo, Giovanna; Bertamino, Alessia; Gomez Monterrey, Isabel; Novellino, Ettore; Sbardella, Gianluca | |
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters | 1-gen-2010 | Campiglia, Pietro; Claudio, Aquino; Bertamino, Alessia; Nicoletta De, Simone; Sala, Marina; Castellano, Sabrina; Marisabella, Santoriello; Paolo, Grieco; Ettore, Novellino; Isabel Maria Gomez, Monterrey | |
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) | 1-gen-2010 | Castellano, Sabrina; Milite, Ciro; Ragno, R; Simeoni, S; Mai, A; Limongelli, V; Novellino, E; Bauer, I; Brosch, G; Spannhoff, A; Cheng, Dh; Bedford, Mt; Sbardella, Gianluca | |
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. | 1-gen-2010 | Castellano, Sabrina; Lucia, Tamborini; Viviano, Monica; Andrea, Pinto; Sbardella, Gianluca; Paola, Conti | |
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators | 1-gen-2011 | DAL PIAZ, Fabrizio; Vassallo, Antonio; Cuesta Rubio, Osmany; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina | |
Chemical biology of Histone acetyltransferase natural compounds modulators. | 1-gen-2011 | DAL PIAZ, Fabrizio; Vassallo, Antonio; Osmany Cuesta, Rubio; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina | |
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors | 1-gen-2011 | Castellano, Sabrina; Dirk, Kuck; Viviano, Monica; Jakyung, Yoo; Fabian López, Vallejo; Paola, Conti; Lucia, Tamborini; Andrea, Pinto; José L., Medina Franco; Sbardella, Gianluca | |
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents | 1-gen-2011 | Wang, Zhiming; Castellano, Sabrina; Kinderman, Sape S.; Argueta, Christian E.; Beshir, Anwar B.; Fenteany, Gabriel; Kwon, Ohyun | |
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. | 1-gen-2011 | Donghang, Cheng; Sergio, Valente; Castellano, Sabrina; Sbardella, Gianluca; Roberto Di, Santo; Roberta, Costi; Mark T., Bedford; Antonello, Mai | |
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) | 1-gen-2011 | Milite, Ciro; Castellano, Sabrina; Benedetti, Rosaria; Tosco, Alessandra; Ciliberti, Carmen; Vicidomini, Caterina; Boully, Ludovic; Franci, Gianluigi; Altucci, Lucia; Mai, Antonello; Sbardella, Gianluca | |
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart | 1-gen-2011 | Claudia, Colussi; Jessica, Rosati; Stefania, Straino; Francesco, Spallotta; Roberta, Berni; Donatella, Stilli; Stefano, Rossi; Ezio, Musso; Emilio, Macchi; Antonello, Mai; Sbardella, Gianluca; Castellano, Sabrina; Cristina, Chimenti; Andrea, Frustaci; Angela, Nebbioso; Lucia, Altucci; Maurizio C., Capogrossi; Carlo, Gaetano | |
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. | 1-gen-2011 | Astrid, Spannhoff; Yong Kee, Kim; Noel J. M., Raynal; Vazganush, Gharibyan; Ming Bo, Su; Yue Yang, Zhou; Jia, Li; Castellano, Sabrina; Sbardella, Gianluca; Jean Pierre J., Issa; Mark T., Bedford | |
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. | 1-gen-2011 | Sbardella, Gianluca; Mai, Antonello; Bartolini, Sara; Castellano, Sabrina; Cirilli, Roberto; Rotili, Dante; Milite, Ciro; Santoriello, Marisabella; Orlando, Serena; Sciamanna, Ilaria; Serafino, Annalucia; Lavia, Patrizia; Spadafora, Corrado | |
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients | 1-gen-2011 | M., Vecellio; G., Pompilio; F., Spallotta; C., Colussi; Sbardella, Gianluca; Castellano, Sabrina; A., Mai; M. C., Capogrossi; A., Rossini; C., Gaetano | |
Microbiologia Molecolare e Cellulare | 1-gen-2012 | Maresca, Bruno; Castellano, Sabrina; Fortino, Vittorio; Morello, Silvana; Porta, Amalia | |
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins | 1-gen-2012 | Colussi, Claudia); Scopece, Alessandro; Vitale, Serena; Spallotta, Francesco; Mattiussi, Stefania; Rosati, Jessica; Illi, Barbara; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca; Farsetti, Antonella; Capogrossi, Maurizio C.; Gaetano, Carlo | |
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear | 1-gen-2012 | Wei, Wei; Coelho, Carlos M.; Li, Xiang; Marek, Roger; Yan, Shanzhi; Anderson, Shawn; Meyers, David; Mukherjee, Chandrani; Sbardella, Gianluca; Castellano, Sabrina; Milite, Ciro; Rotili, Dante; Mai, Antonello; Cole, Philip A.; Sah, Pankaj; Kobor, Michael S.; Bredy, Timothy W. | |
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds | 1-gen-2012 | Granata, Ilaria; Castellano, Sabrina; Armenante, Annunziata; Maresca, Bruno; Porta, Amalia |
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