BIFULCO, Giuseppe
BIFULCO, Giuseppe
Dipartimento di Farmacia/DIFARMA
(±)-Gelliusines A and B, Two Diastereomeric Brominated Tris-indole Alkaloids from a Deep Water New Caledonian Marine Sponge (Gellius or Orina sp.)
1994-01-01 Bifulco, Giuseppe; Bruno, Ines; Luigi, Minale; Riccio, Raffaele; Antonio, Calignano; Cécile, Debitus
1H-1H scalar coupling across two stacked aromatic rings: DFT calculations and experimental proof
2008-01-01 Bifulco, Giuseppe; A., Mangoni
2'-Methyl taxanes: synthesis and NMR configurational assignment.
2005-01-01 Dambruoso, Paolo; Bassarello, Carla; Bifulco, Giuseppe; Appendino, Giovanni; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; GOMEZ PALOMA, Luigi
2,3-Dihydrobenzofuran privileged structures as new bioinspired lead compounds for the design of mPGES-1 inhibitors
2016-01-01 DI MICCO, Simone; Spatafora, Carmela; Cardullo, Nunzio; Riccio, Raffaele; Fischer, Katrin; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Chalal, Malik; Vervandier Fasseur, Dominique; Tringali, Corrado; Bifulco, Giuseppe
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines
2023-01-01 De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity
2012-01-01 Simona De, Marino; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Claudio, D’Amore; Barbara, Renga; Andrea, Mencarelli; Sylvain, Petek; Stefano, Fiorucci; Angela, Zampella
40 th "A. Corbella" International Summer School on Organic Synthesis - ISOS 2015
2015-01-01 Foglia, Antonio; Di Micco, Simone; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Oppermann, Udo; Bifulco, Giuseppe; Bruno, Ines
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates
2025-01-01 Colarusso, E.; Lauro, G.; Potenza, M.; Galatello, P.; Garigliota, M. L. D.; Ferraro, M. G.; Piccolo, M.; Chini, M. G.; Irace, C.; Campiglia, P.; Hoffstetter, R. K.; Werz, O.; Ramunno, A.; Bifulco, G.
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
2022-01-01 Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain
2015-01-01 Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis
A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors
2013-01-01 DAL PIAZ, Fabrizio; Vassallo, A.; Temraz, A.; Cotugno, Roberta; Belisario, MARIA ANTONIETTA; Bifulco, Giuseppe; Chini, MARIA GIOVANNA; Pisano, C.; DE TOMMASI, Nunziatina; Braca, A.
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids
2023-01-01 Rogati, F.; Maioli, C.; Lauro, G.; Caprioglio, D.; Imperio, D.; Del Grosso, E.; Botta, B.; Mannina, L.; Bifulco, G.; Ingallina, C.; Minassi, A.
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors
2020-01-01 Lauro, G.; Terracciano, S.; Cantone, V.; Ruggiero, D.; Fischer, K.; Pace, S.; Werz, O.; Bruno, I.; Bifulco, G.
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors
2024-01-01 Vestuto, Vincenzo; Ciaglia, Tania; Musella, Simona; Di Sarno, Veronica; Smaldone, Gerardina; Di Matteo, Francesca; Scala, Maria Carmina; Napolitano, Valeria; Miranda, Maria Rosaria; Amodio, Giuseppina; Novi, Sara; Pepe, Giacomo; Basilicata, Manuela Giovanna; Gazzillo, Erica; Pace, Simona; Gomez-Monterrey, Isabel M.; Sala, Marina; Bifulco, Giuseppe; Tecce, Mario Felice; Campiglia, Pietro; Ostacolo, Carmine; Lauro, Gianluigi; Manfra, Michele; Bertamino, Alessia
A NOVEL PHENOLIC SPIRO DERIVATIVE, YUCCAONE A, FROM YUCCA SCHIDIGERA BARK.
2002-01-01 Piacente, Sonia; Bifulco, Giuseppe; Pizza, Cosimo; Stochmal, A.; Oleszek, W.
A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry
2010-01-01 G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19)
2020-01-01 De Vita, S.; Chini, M. G.; Lauro, G.; Bifulco, G.
Accurate prediction of 1H chemical shifts in interstrand cross-linked DNA
2013-01-01 Ewald, Pauwels; Diederica, Claeys; José C., Martins; Michel, Waroquier; Bifulco, Giuseppe; Veronique Van, Speybroeck; Annemieke, Madder
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches
2021-01-01 Chini, M. G.; Lauro, G.; Bifulco, G.
Advances in the Universal NMR Database Approach. 2'-Substituted Taxanes as Probes for an Improved Protocol of Diastereomeric Differentiation.
2005-01-01 Dambruoso, Paolo; Bassarello, Carla; Bifulco, Giuseppe; Appendino, Giovanni; Battaglia, Arturo; Fontana, Gabriele; GOMEZ PALOMA, Luigi
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (±)-Gelliusines A and B, Two Diastereomeric Brominated Tris-indole Alkaloids from a Deep Water New Caledonian Marine Sponge (Gellius or Orina sp.) | 1-gen-1994 | Bifulco, Giuseppe; Bruno, Ines; Luigi, Minale; Riccio, Raffaele; Antonio, Calignano; Cécile, Debitus | |
| 1H-1H scalar coupling across two stacked aromatic rings: DFT calculations and experimental proof | 1-gen-2008 | Bifulco, Giuseppe; A., Mangoni | |
| 2'-Methyl taxanes: synthesis and NMR configurational assignment. | 1-gen-2005 | Dambruoso, Paolo; Bassarello, Carla; Bifulco, Giuseppe; Appendino, Giovanni; Battaglia, Arturo; Guerrini, Andrea; Fontana, Gabriele; GOMEZ PALOMA, Luigi | |
| 2,3-Dihydrobenzofuran privileged structures as new bioinspired lead compounds for the design of mPGES-1 inhibitors | 1-gen-2016 | DI MICCO, Simone; Spatafora, Carmela; Cardullo, Nunzio; Riccio, Raffaele; Fischer, Katrin; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Chalal, Malik; Vervandier Fasseur, Dominique; Tringali, Corrado; Bifulco, Giuseppe | |
| 2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines | 1-gen-2023 | De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe | |
| 4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity | 1-gen-2012 | Simona De, Marino; Raffaella, Ummarino; Maria Valeria, D’Auria; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Claudio, D’Amore; Barbara, Renga; Andrea, Mencarelli; Sylvain, Petek; Stefano, Fiorucci; Angela, Zampella | |
| 40 th "A. Corbella" International Summer School on Organic Synthesis - ISOS 2015 | 1-gen-2015 | Foglia, Antonio; Di Micco, Simone; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Oppermann, Udo; Bifulco, Giuseppe; Bruno, Ines | |
| 5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates | 1-gen-2025 | Colarusso, E.; Lauro, G.; Potenza, M.; Galatello, P.; Garigliota, M. L. D.; Ferraro, M. G.; Piccolo, M.; Chini, M. G.; Irace, C.; Campiglia, P.; Hoffstetter, R. K.; Werz, O.; Ramunno, A.; Bifulco, G. | |
| 6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis | 1-gen-2022 | Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G | |
| 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain | 1-gen-2015 | Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
| A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors | 1-gen-2013 | DAL PIAZ, Fabrizio; Vassallo, A.; Temraz, A.; Cotugno, Roberta; Belisario, MARIA ANTONIETTA; Bifulco, Giuseppe; Chini, MARIA GIOVANNA; Pisano, C.; DE TOMMASI, Nunziatina; Braca, A. | |
| A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids | 1-gen-2023 | Rogati, F.; Maioli, C.; Lauro, G.; Caprioglio, D.; Imperio, D.; Del Grosso, E.; Botta, B.; Mannina, L.; Bifulco, G.; Ingallina, C.; Minassi, A. | |
| A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors | 1-gen-2020 | Lauro, G.; Terracciano, S.; Cantone, V.; Ruggiero, D.; Fischer, K.; Pace, S.; Werz, O.; Bruno, I.; Bifulco, G. | |
| A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors | 1-gen-2024 | Vestuto, Vincenzo; Ciaglia, Tania; Musella, Simona; Di Sarno, Veronica; Smaldone, Gerardina; Di Matteo, Francesca; Scala, Maria Carmina; Napolitano, Valeria; Miranda, Maria Rosaria; Amodio, Giuseppina; Novi, Sara; Pepe, Giacomo; Basilicata, Manuela Giovanna; Gazzillo, Erica; Pace, Simona; Gomez-Monterrey, Isabel M.; Sala, Marina; Bifulco, Giuseppe; Tecce, Mario Felice; Campiglia, Pietro; Ostacolo, Carmine; Lauro, Gianluigi; Manfra, Michele; Bertamino, Alessia | |
| A NOVEL PHENOLIC SPIRO DERIVATIVE, YUCCAONE A, FROM YUCCA SCHIDIGERA BARK. | 1-gen-2002 | Piacente, Sonia; Bifulco, Giuseppe; Pizza, Cosimo; Stochmal, A.; Oleszek, W. | |
| A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry | 1-gen-2010 | G., Colombano; C., Travelli; U., Galli; A., Caldarelli; Chini, MARIA GIOVANNA; P. L., Canonico; G., Sorba; Bifulco, Giuseppe; G. C., Tron; A. A., Genazzani | |
| Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) | 1-gen-2020 | De Vita, S.; Chini, M. G.; Lauro, G.; Bifulco, G. | |
| Accurate prediction of 1H chemical shifts in interstrand cross-linked DNA | 1-gen-2013 | Ewald, Pauwels; Diederica, Claeys; José C., Martins; Michel, Waroquier; Bifulco, Giuseppe; Veronique Van, Speybroeck; Annemieke, Madder | |
| Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches | 1-gen-2021 | Chini, M. G.; Lauro, G.; Bifulco, G. | |
| Advances in the Universal NMR Database Approach. 2'-Substituted Taxanes as Probes for an Improved Protocol of Diastereomeric Differentiation. | 1-gen-2005 | Dambruoso, Paolo; Bassarello, Carla; Bifulco, Giuseppe; Appendino, Giovanni; Battaglia, Arturo; Fontana, Gabriele; GOMEZ PALOMA, Luigi |