MILITE, Ciro

MILITE, Ciro  

Dipartimento di Farmacia/DIFARMA  

Mostra records
Risultati 1 - 20 di 66 (tempo di esecuzione: 0.061 secondi).
Titolo Data di pubblicazione Autore(i) File
2‐Phenylquinolines Exhibit Anti‐Severe Acute Respiratory Syndrome Coronavirus‐2 Activity Through the Nonstructural Protein 13 Helicase Inhibition 1-gen-2026 Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 1-gen-2018 Salerno, Silvia; Barresi, Elisabetta; Amendola, Giorgio; Berrino, Emanuela; Milite, Ciro; Marini, Anna Maria; DA SETTIMO PASSETTI, Federico; Novellino, Ettore; Supuran, Claudiu T.; Cosconati, Sandro; Taliani, Sabrina
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 1-gen-2015 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 1-gen-2015 Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 1-gen-2015 Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 1-gen-2022 Creighton, Samantha D.; Jardine, Kristen H.; Desimone, Alexa; Zmetana, Megan; Castellano, Sabrina; Milite, Ciro; Sbardella, Gianluca; Winters, Boyer D.
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 1-gen-2013 Calabrese, ELENA CONCETTA; Castellano, Sabrina; M., Santoriello; C., Sgherri; M. F., Quartacci; L., Calucci; A. G. S., Warrilow; D. C., Lamb; S. L., Kelly; Milite, Ciro; Granata, Ilaria; Sbardella, Gianluca; G., Stefancich; Maresca, Bruno; Porta, Amalia
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 1-gen-2019 Salerno, S.; La Pietra, V.; Hyeraci, M.; Taliani, S.; Robello, M.; Barresi, E.; Milite, C.; Simorini, F.; García-Argáez, A. N.; Marinelli, L.; Novellino, E.; Da Settimo, F.; Marini, A. M.; Dalla Via, L.
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 1-gen-2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 1-gen-2015 Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E.
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 1-gen-2015 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 1-gen-2016 Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca
Coactivator-associated arginine methyltransferase 1 (CARM1) inhibitors: a patenting perspective (2018-present) 1-gen-2025 Viviano, Monica; Cipriano, Alessandra; Feoli, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 1-gen-2010 Castellano, Sabrina; Milite, Ciro; Ragno, R; Simeoni, S; Mai, A; Limongelli, V; Novellino, E; Bauer, I; Brosch, G; Spannhoff, A; Cheng, Dh; Bedford, Mt; Sbardella, Gianluca
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1-gen-2018 Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G.
Design, synthesis and biological evaluation of new small molecule modulators of Arginine methyltransferases 21-feb-2011 Milite, Ciro
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 1-gen-2016 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 1-gen-2017 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 1-gen-2015 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 1-gen-2017 Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca