Colarusso, Ester

Colarusso, Ester  

Dipartimento di Farmacia/DIFARMA  

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Risultati 1 - 14 di 14 (tempo di esecuzione: 0.034 secondi).
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2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 1-gen-2023 De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 1-gen-2025 Colarusso, E.; Lauro, G.; Potenza, M.; Galatello, P.; Garigliota, M. L. D.; Ferraro, M. G.; Piccolo, M.; Chini, M. G.; Irace, C.; Campiglia, P.; Hoffstetter, R. K.; Werz, O.; Ramunno, A.; Bifulco, G.
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 1-gen-2022 Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 1-gen-2024 Samukha, V.; Fantasma, F.; D'Urso, G.; Colarusso, E.; Schettino, A.; Marigliano, N.; Chini, M. G.; Saviano, G.; De Felice, V.; Lauro, G.; Maione, F.; Bifulco, G.; Casapullo, A.; Iorizzi, M.
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 1-gen-2024 Fantasma, F.; Samukha, V.; Aliberti, M.; Colarusso, E.; Chini, M. G.; Saviano, G.; De Felice, V.; Lauro, G.; Casapullo, A.; Bifulco, G.; Iorizzi, M.
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 1-gen-2023 Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi
Identification and Development of BRD9 Chemical Probes 1-gen-2024 Colarusso, E.; Chini, M. G.; Bifulco, G.; Lauro, G.; Giordano, A.
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 1-gen-2023 Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 1-gen-2024 Colarusso, E.; Gazzillo, E.; Boccia, E.; Terracciano, S.; Bruno, I.; Bifulco, G.; Chini, M. G.; Lauro, G.
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 1-gen-2024 Colarusso, E.; Gazzillo, E.; Pierri, M.; Ruggiero, D.; Chini, M. G.; Bruno, I.; Bifulco, G.; Terracciano, S.; Lauro, G.
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 1-gen-2024 De Vita, S.; Colarusso, E.; Chini, M. G.; Bifulco, G.; Lauro, G.
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 1-gen-2024 Gazzillo, E.; Colarusso, E.; Giordano, A.; Chini, M. G.; Potenza, M.; Hofstetter, R. K.; Iorizzi, M.; Werz, O.; Lauro, G.; Bifulco, G.
Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE2Levels 1-gen-2020 Chini, M. G.; Giordano, A.; Potenza, M.; Terracciano, S.; Fischer, K.; Vaccaro, M. C.; Colarusso, E.; Bruno, I.; Riccio, R.; Koeberle, A.; Werz, O.; Bifulco, G.
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 1-gen-2022 Colarusso, Ester; Potenza, Marianna; Lauro, Gianluigi; Giovanna Chini, Maria; Sepe, Valentina; Zampella, Angela; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Bifulco, Giuseppe