Sfoglia per Autore
In cell scalaradial interactome profiling using a bio-orthogonal clickable probe
2014-01-01 Cassiano, Chiara; Margarucci, Luigi; Esposito, Roberta; Riccio, Raffaele; Tosco, Alessandra; Casapullo, Agostino; Monti, Maria Chiara
N-Formyl-7-amino-11-cycloamphilectene, a marine sponge metabolite, binds to tubulin and modulates microtubule depolymerization
2014-01-01 Margarucci, Luigi; Monti, Maria Chiara; Esposito, Roberta; Tosco, Alessandra; Ernest, Hamel; Riccio, Raffaele; Casapullo, Agostino
Heteronemin, a marine sponge terpenoid, targets TDP-43, a key factor in several neurodegenerative disorders
2014-01-01 Cassiano, Chiara; Esposito, Roberta; Tosco, Alessandra; Angela, Zampella; Maria Valeria, D'Auria; Riccio, Raffaele; Casapullo, Agostino; Monti, Maria Chiara
Role of arabidopsis UV RESISTANCE LOCUS 8 in plant growth reduction under osmotic stress and low levels of UV-B
2014-01-01 Fasano, Rossella; Gonzalez, Nathalie; Tosco, Alessandra; DAL PIAZ, Fabrizio; Docimo, Teresa; Serrano, Ramon; Grillo, Stefania; Leone, Antonietta; Inzé, Dirk
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach
2015-01-01 Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Trefoil Factor 1 is involved in gastric cell copper homeostasis
2015-01-01 Esposito, Roberta; Sandro, Montefusco; Ferro, Piera; Monti, Maria Chiara; Baldantoni, Daniela; Tosco, Alessandra; Marzullo, Liberato
In Cell Interactome of Oleocanthal, an Extra Virgin Olive Oil Bioactive Component
2015-01-01 Cassiano, Chiara; Casapullo, Agostino; Tosco, Alessandra; Monti, Maria Chiara; Riccio, Raffaele
Theonellasterone, a steroidal metabolite isolated from a Theonella sponge, protects peroxiredoxin-1 from oxidative stress reactions
2015-01-01 Margarucci, Luigi; Monti, Maria Chiara; Tosco, Alessandra; Esposito, Roberta; Zampella, A.; Sepe, V.; Mozzicafreddo, M.; Riccio, Raffaele; Casapullo, Agostino
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.
2015-01-01 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.
2015-01-01 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.
2015-01-01 Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF
2015-01-01 Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca
Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A
2015-01-01 DAL PIAZ, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Tosco, Alessandra; DE TOMMASI, Nunziatina
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015)
2015-01-01 Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20
2015-01-01 Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.
2015-01-01 Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
β-Boswellic acid, a bioactive substance used in food supplements, inhibits protein synthesis by targeting the ribosomal machinery
2016-01-01 Casapullo, Agostino; Cassiano, Chiara; Capolupo, Angela; DEL GAUDIO, Federica; Esposito, Roberta; Tosco, Alessandra; Riccio, Raffaele; Monti, Maria Chiara
Gastric TFF1 Expression from Acute to Chronic Helicobacter Infection
2017-01-01 Esposito, Roberta; Morello, Silvana; Vllahu, Megi; Eletto, Daniela; Porta, Amalia; Tosco, Alessandra
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer
2017-01-01 Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia
Proteasome as a new target for bio-inspired benzo[k,l]xanthene lignans
2017-01-01 Capolupo, Angela; Tosco, Alessandra; Mozzicafreddo, Matteo; Tringali, Corrado; Cardullo, Nunzio; Monti, Maria Chiara; Casapullo, Agostino
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
In cell scalaradial interactome profiling using a bio-orthogonal clickable probe | 1-gen-2014 | Cassiano, Chiara; Margarucci, Luigi; Esposito, Roberta; Riccio, Raffaele; Tosco, Alessandra; Casapullo, Agostino; Monti, Maria Chiara | |
N-Formyl-7-amino-11-cycloamphilectene, a marine sponge metabolite, binds to tubulin and modulates microtubule depolymerization | 1-gen-2014 | Margarucci, Luigi; Monti, Maria Chiara; Esposito, Roberta; Tosco, Alessandra; Ernest, Hamel; Riccio, Raffaele; Casapullo, Agostino | |
Heteronemin, a marine sponge terpenoid, targets TDP-43, a key factor in several neurodegenerative disorders | 1-gen-2014 | Cassiano, Chiara; Esposito, Roberta; Tosco, Alessandra; Angela, Zampella; Maria Valeria, D'Auria; Riccio, Raffaele; Casapullo, Agostino; Monti, Maria Chiara | |
Role of arabidopsis UV RESISTANCE LOCUS 8 in plant growth reduction under osmotic stress and low levels of UV-B | 1-gen-2014 | Fasano, Rossella; Gonzalez, Nathalie; Tosco, Alessandra; DAL PIAZ, Fabrizio; Docimo, Teresa; Serrano, Ramon; Grillo, Stefania; Leone, Antonietta; Inzé, Dirk | |
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
Trefoil Factor 1 is involved in gastric cell copper homeostasis | 1-gen-2015 | Esposito, Roberta; Sandro, Montefusco; Ferro, Piera; Monti, Maria Chiara; Baldantoni, Daniela; Tosco, Alessandra; Marzullo, Liberato | |
In Cell Interactome of Oleocanthal, an Extra Virgin Olive Oil Bioactive Component | 1-gen-2015 | Cassiano, Chiara; Casapullo, Agostino; Tosco, Alessandra; Monti, Maria Chiara; Riccio, Raffaele | |
Theonellasterone, a steroidal metabolite isolated from a Theonella sponge, protects peroxiredoxin-1 from oxidative stress reactions | 1-gen-2015 | Margarucci, Luigi; Monti, Maria Chiara; Tosco, Alessandra; Esposito, Roberta; Zampella, A.; Sepe, V.; Mozzicafreddo, M.; Riccio, Raffaele; Casapullo, Agostino | |
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF | 1-gen-2015 | Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A | 1-gen-2015 | DAL PIAZ, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Tosco, Alessandra; DE TOMMASI, Nunziatina | |
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) | 1-gen-2015 | Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. | 1-gen-2015 | Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
β-Boswellic acid, a bioactive substance used in food supplements, inhibits protein synthesis by targeting the ribosomal machinery | 1-gen-2016 | Casapullo, Agostino; Cassiano, Chiara; Capolupo, Angela; DEL GAUDIO, Federica; Esposito, Roberta; Tosco, Alessandra; Riccio, Raffaele; Monti, Maria Chiara | |
Gastric TFF1 Expression from Acute to Chronic Helicobacter Infection | 1-gen-2017 | Esposito, Roberta; Morello, Silvana; Vllahu, Megi; Eletto, Daniela; Porta, Amalia; Tosco, Alessandra | |
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer | 1-gen-2017 | Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia | |
Proteasome as a new target for bio-inspired benzo[k,l]xanthene lignans | 1-gen-2017 | Capolupo, Angela; Tosco, Alessandra; Mozzicafreddo, Matteo; Tringali, Corrado; Cardullo, Nunzio; Monti, Maria Chiara; Casapullo, Agostino |
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