Sfoglia per Autore
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.
2015-01-01 Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.
2015-01-01 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015)
2015-01-01 Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach
2015-01-01 Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli
2015-01-01 Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E.
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
2015-01-01 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF
2015-01-01 Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach
2016-01-01 Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Nunziata, Antonietta; Castellano, Sabrina; Sbardella, Gianluca
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
2016-01-01 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY
2016-01-01 Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors
2016-01-01 Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors
2016-01-01 Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca
The emerging role of lysine methyltransferase SETD8 in human diseases
2016-01-01 Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach
2016-01-01 Chini, MARIA GIOVANNA; Malafronte, Nicola; Vaccaro, Maria C.; Gualtieri, Maria J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; DAL PIAZ, Fabrizio
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach
2017-01-01 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins
2017-01-01 Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach
2017-01-01 Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy
2017-01-01 Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells
2017-01-01 Miele, Evelina; Valente, Sergio; Alfano, Vincenzo; Silvano, Marianna; Mellini, Paolo; Borovika, Diana; Marrocco, Biagina; Po, Agnese; Mersini Besharat, Zein; Catanzaro, Giuseppina; Battaglia, Giuseppe; Abballe, Luana; Zwergel, Clemens; Stazi, Giulia; Milite, Ciro; Castellano, Sabrina; Tafani, Marco; Trapencieris, Peteris; Mai, Antonello; Ferretti, Elisabetta
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO)
2017-01-01 Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) | 1-gen-2015 | Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli | 1-gen-2015 | Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E. | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery | 1-gen-2015 | Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF | 1-gen-2015 | Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach | 1-gen-2016 | Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Nunziata, Antonietta; Castellano, Sabrina; Sbardella, Gianluca | |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH | 1-gen-2016 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
| IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY | 1-gen-2016 | Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca | |
| ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors | 1-gen-2016 | Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors | 1-gen-2016 | Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| The emerging role of lysine methyltransferase SETD8 in human diseases | 1-gen-2016 | Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach | 1-gen-2016 | Chini, MARIA GIOVANNA; Malafronte, Nicola; Vaccaro, Maria C.; Gualtieri, Maria J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; DAL PIAZ, Fabrizio | |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach | 1-gen-2017 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins | 1-gen-2017 | Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach | 1-gen-2017 | Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of new KDM4 inhibitors through a HTS and hit refinement strategy | 1-gen-2017 | Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca | |
| The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells | 1-gen-2017 | Miele, Evelina; Valente, Sergio; Alfano, Vincenzo; Silvano, Marianna; Mellini, Paolo; Borovika, Diana; Marrocco, Biagina; Po, Agnese; Mersini Besharat, Zein; Catanzaro, Giuseppina; Battaglia, Giuseppe; Abballe, Luana; Zwergel, Clemens; Stazi, Giulia; Milite, Ciro; Castellano, Sabrina; Tafani, Marco; Trapencieris, Peteris; Mai, Antonello; Ferretti, Elisabetta | |
| Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) | 1-gen-2017 | Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia |
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