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Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1)
2014-01-01 Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe
Garcinol and Related Polyisoprenylated Benzophenones as Topoisomerase II Inhibitors: Biochemical and Molecular Modeling Studies
2019-01-01 Di Micco, S.; Masullo, M.; Bandak, A. F.; Berger, J. M.; Riccio, R.; Piacente, S.; Bifulco, G.
Heat shock proteins as key biological targets of the marine natural cyclopeptide perthamide C
2012-01-01 Margarucci, Luigi; Monti, Maria Chiara; Andrea, Mencarelli; Cassiano, Chiara; Stefano, Fiorucci; Riccio, Raffaele; Angela, Zampella; Casapullo, Agostino
Heteronemin, a marine sponge terpenoid, targets TDP-43, a key factor in several neurodegenerative disorders
2014-01-01 Cassiano, Chiara; Esposito, Roberta; Tosco, Alessandra; Angela, Zampella; Maria Valeria, D'Auria; Riccio, Raffaele; Casapullo, Agostino; Monti, Maria Chiara
HIV-Inhibitory Natural Products. 11. Comparative Studies of Sulfated Sterols from Marine Invertebrates
1994-01-01 Tawnya C., Mckee; John H., Cardellina; Riccio, Raffaele; Maria Valeria, D'Auria; Maria, Iorizzi; Luigi, Minale; Robert A., Moran; Robert J., Gulakowski; James B., Mcmahon
Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors
2018-01-01 DI MICCO, Simone; Luana, Pulvirenti; Bruno, Ines; Terracciano, Stefania; Russo, Alessandra; Vaccaro, Mariacarmela; Ruggiero, Dafne; Vera, Muccilli; Nunzio, Cardullo; Corrado, Tringali; Riccio, Raffaele; Bifulco, Giuseppe
Identification of new γ-hydroxybutenolides that preferentially inhibit the activity of mPGES-1
2012-01-01 Rosa De, Simone; Bruno, Ines; Riccio, Raffaele; Katharina, Stadler; Julia, Bauer; Anja M., Schaible; Stefan, Laufer; Oliver, Werz
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening
2017-01-01 Lauro, Gianluigi; Manfra, Michele; Pedatella, Silvana; Fischer, Katrin; Cantone, Vincenza; Terracciano, Stefania; Bertamino, Alessia; Ostacolo, Carmine; Gomez Monterrey, Isabel; De Nisco, Mauro; Riccio, Raffaele; Novellino, Ettore; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe
Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition
2019-01-01 Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C.; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) | 1-gen-2014 | Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
Garcinol and Related Polyisoprenylated Benzophenones as Topoisomerase II Inhibitors: Biochemical and Molecular Modeling Studies | 1-gen-2019 | Di Micco, S.; Masullo, M.; Bandak, A. F.; Berger, J. M.; Riccio, R.; Piacente, S.; Bifulco, G. | |
Heat shock proteins as key biological targets of the marine natural cyclopeptide perthamide C | 1-gen-2012 | Margarucci, Luigi; Monti, Maria Chiara; Andrea, Mencarelli; Cassiano, Chiara; Stefano, Fiorucci; Riccio, Raffaele; Angela, Zampella; Casapullo, Agostino | |
Heteronemin, a marine sponge terpenoid, targets TDP-43, a key factor in several neurodegenerative disorders | 1-gen-2014 | Cassiano, Chiara; Esposito, Roberta; Tosco, Alessandra; Angela, Zampella; Maria Valeria, D'Auria; Riccio, Raffaele; Casapullo, Agostino; Monti, Maria Chiara | |
HIV-Inhibitory Natural Products. 11. Comparative Studies of Sulfated Sterols from Marine Invertebrates | 1-gen-1994 | Tawnya C., Mckee; John H., Cardellina; Riccio, Raffaele; Maria Valeria, D'Auria; Maria, Iorizzi; Luigi, Minale; Robert A., Moran; Robert J., Gulakowski; James B., Mcmahon | |
Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors | 1-gen-2018 | DI MICCO, Simone; Luana, Pulvirenti; Bruno, Ines; Terracciano, Stefania; Russo, Alessandra; Vaccaro, Mariacarmela; Ruggiero, Dafne; Vera, Muccilli; Nunzio, Cardullo; Corrado, Tringali; Riccio, Raffaele; Bifulco, Giuseppe | |
Identification of new γ-hydroxybutenolides that preferentially inhibit the activity of mPGES-1 | 1-gen-2012 | Rosa De, Simone; Bruno, Ines; Riccio, Raffaele; Katharina, Stadler; Julia, Bauer; Anja M., Schaible; Stefan, Laufer; Oliver, Werz | |
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening | 1-gen-2017 | Lauro, Gianluigi; Manfra, Michele; Pedatella, Silvana; Fischer, Katrin; Cantone, Vincenza; Terracciano, Stefania; Bertamino, Alessia; Ostacolo, Carmine; Gomez Monterrey, Isabel; De Nisco, Mauro; Riccio, Raffaele; Novellino, Ettore; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe | |
Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition | 1-gen-2019 | Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C.; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone | |
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines |
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Opzioni
Scopri
Tipologia
- 1 Contributo su Rivista 136
- 1 Contributo su Rivista::1.1.1 Ar... 136
Data di pubblicazione
- 2010 - 2020 60
- 2000 - 2009 1
- 1990 - 1999 29
- 1980 - 1989 37
- 1971 - 1979 9
Rivista
- JOURNAL OF NATURAL PRODUCTS 36
- TETRAHEDRON LETTERS 15
- JOURNAL OF ORGANIC CHEMISTRY 8
- CHEMICAL COMMUNICATIONS 7
- COMPARATIVE BIOCHEMISTRY AND PHYS... 7
- EUROPEAN JOURNAL OF MEDICINAL CHE... 7
- TETRAHEDRON 7
- BIOORGANIC & MEDICINAL CHEMISTRY 5
- MOLECULAR BIOSYSTEMS 4
- ACS MEDICINAL CHEMISTRY LETTERS 3
Keyword
- Drug Discovery3003 Pharmaceutical... 7
- Organic Chemistry 7
- 3003 4
- Humans 4
- Molecular Medicine 4
- mPGES-1 inhibitors 4
- Pharmacology 4
- Biochemistry 3
- chemical proteomics 3
- Chemistry (all) 3
Lingua
- eng 135
Accesso al fulltext
- no fulltext 124
- reserved 11
- open 1