Sfoglia per Autore
Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90
2012-01-01 DAL PIAZ, Fabrizio; Vassallo, Antonio; Chini, MARIA GIOVANNA; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; Brandi, Alberto
Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors
2013-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Structural basis for the design and synthesis of selective HDAC inhibitors
2013-01-01 DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors
2013-01-01 DAL PIAZ, Fabrizio; Vassallo, A.; Temraz, A.; Cotugno, Roberta; Belisario, MARIA ANTONIETTA; Bifulco, Giuseppe; Chini, MARIA GIOVANNA; Pisano, C.; DE TOMMASI, Nunziatina; Braca, A.
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors
2015-01-01 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Molecular mechanism of tanshinone IIA and cryptotanshinone in platelet anti-aggregating effects: an integrated study of pharmacology and computational analysis
2015-01-01 Maione, Francesco; Cantone, Vincenza; Chini, MARIA GIOVANNA; DE FEO, Vincenzo; Mascolo, Nicola; Bifulco, Giuseppe
Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A
2015-01-01 DAL PIAZ, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Tosco, Alessandra; DE TOMMASI, Nunziatina
Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold
2015-01-01 Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe
Computational NMR Methods in the Stereochemical Analysis of Organic Compounds: Are Proton or Carbon NMR Chemical Shift Data More Discriminating?
2015-01-01 Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe
Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors
2015-01-01 Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe
Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors
2015-01-01 Chini, MARIA GIOVANNA; Ferroni, Claudia; Cantone, Vincenza; Dambruoso, Paolo; Varchi, Greta; Pepe, Antonella; Fischer, Katrin; Pergola, Carlo; Werz, Oliver; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe
New dihydropyrimidin-2(1H)-one based Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Foglia, Antonio; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Russo, Alessandra; DAL PIAZ, Fabrizio; Saturnino, C.; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach
2016-01-01 Chini, MARIA GIOVANNA; Malafronte, Nicola; Vaccaro, Maria C.; Gualtieri, Maria J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; DAL PIAZ, Fabrizio
Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors
2016-01-01 Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Anti-inflammatory and analgesic activity of carnosol and carnosic acid in vivo and in vitro and in silico analysis of their target interactions
2017-01-01 Maione, Francesco; Cantone, Vincenza; Pace, Simona; Chini, MARIA GIOVANNA; Bisio, Angela; Romussi, Giovanni; Pieretti, Stefano; Werz, Oliver; Koeberle, Andreas; Mascolo, Nicola; Bifulco, Giuseppe
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells
2018-01-01 Ayoub, Khalfaoui; Chini, MARIA GIOVANNA; Mohamed, Bouheroum; Soumia, Belaabed; Lauro, Gianluigi; Terracciano, Stefania; Vaccaro, Mariacarmela; Bruno, Ines; Samir, Benayache; Ines, Mancini; Bifulco, Giuseppe
Down regulation of pro-inflammatory pathways by tanshinone IIA and cryptotanshinone in a non-genetic mouse model of Alzheimer's disease
2018-01-01 Maione, Francesco; Piccolo, Marialuisa; DE VITA, Simona; Chini, Maria Giovanna; Cristiano, Claudia; De Caro, Carmen; Lippiello, Pellegrino; Miniaci, Maria Concetta; Santamaria, Rita; Irace, Carlo; De Feo, Vincenzo; Calignano, Antonio; Mascolo, Nicola; Bifulco, Giuseppe
Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain
2018-01-01 Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Guaianolides from Ormenis mixta: Structural Insights and Evaluation of Their Anti-inflammatory Profile
2019-01-01 Benteldjoune, Mounira; Chini, Maria Giovanna; Iannuzzi, Anna Maria; Kabouche, Ahmed; Kabouche, Zahia; Dʼambola, Massimiliano; Marzocco, Stefania; Autore, Giuseppina; Bifulco, Giuseppe; De Tommasi, Nunziatina
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90 | 1-gen-2012 | DAL PIAZ, Fabrizio; Vassallo, Antonio; Chini, MARIA GIOVANNA; Cordero Franca, M.; Cardona, Francesca; Pisano, Claudio; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; Brandi, Alberto | |
| Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors | 1-gen-2013 | Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Structural basis for the design and synthesis of selective HDAC inhibitors | 1-gen-2013 | DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| A Chemical-Biological Study Reveals C-9-type Iridoids as Novel Heat Shock Protein 90 (Hsp90) Inhibitors | 1-gen-2013 | DAL PIAZ, Fabrizio; Vassallo, A.; Temraz, A.; Cotugno, Roberta; Belisario, MARIA ANTONIETTA; Bifulco, Giuseppe; Chini, MARIA GIOVANNA; Pisano, C.; DE TOMMASI, Nunziatina; Braca, A. | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors | 1-gen-2015 | Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Molecular mechanism of tanshinone IIA and cryptotanshinone in platelet anti-aggregating effects: an integrated study of pharmacology and computational analysis | 1-gen-2015 | Maione, Francesco; Cantone, Vincenza; Chini, MARIA GIOVANNA; DE FEO, Vincenzo; Mascolo, Nicola; Bifulco, Giuseppe | |
| Identification and mechanism of action analysis of the new PARP-1 inhibitor 2″-hydroxygenkwanol A | 1-gen-2015 | DAL PIAZ, Fabrizio; Ferro, Piera; Vassallo, Antonio; Vasaturo, Michele; Forte, Giovanni; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Tosco, Alessandra; DE TOMMASI, Nunziatina | |
| Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold | 1-gen-2015 | Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Computational NMR Methods in the Stereochemical Analysis of Organic Compounds: Are Proton or Carbon NMR Chemical Shift Data More Discriminating? | 1-gen-2015 | Chini, MARIA GIOVANNA; Riccio, Raffaele; Bifulco, Giuseppe | |
| Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors | 1-gen-2015 | Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe | |
| Elucidating new structural features of the triazole scaffold for the development of mPGES-1 inhibitors | 1-gen-2015 | Chini, MARIA GIOVANNA; Ferroni, Claudia; Cantone, Vincenza; Dambruoso, Paolo; Varchi, Greta; Pepe, Antonella; Fischer, Katrin; Pergola, Carlo; Werz, Oliver; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| New dihydropyrimidin-2(1H)-one based Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Foglia, Antonio; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Russo, Alessandra; DAL PIAZ, Fabrizio; Saturnino, C.; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach | 1-gen-2016 | Chini, MARIA GIOVANNA; Malafronte, Nicola; Vaccaro, Maria C.; Gualtieri, Maria J.; Vassallo, Antonio; Vasaturo, Michele; Castellano, Sabrina; Milite, Ciro; Leone, Antonietta; Bifulco, Giuseppe; DE TOMMASI, Nunziatina; DAL PIAZ, Fabrizio | |
| Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors | 1-gen-2016 | Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Anti-inflammatory and analgesic activity of carnosol and carnosic acid in vivo and in vitro and in silico analysis of their target interactions | 1-gen-2017 | Maione, Francesco; Cantone, Vincenza; Pace, Simona; Chini, MARIA GIOVANNA; Bisio, Angela; Romussi, Giovanni; Pieretti, Stefano; Werz, Oliver; Koeberle, Andreas; Mascolo, Nicola; Bifulco, Giuseppe | |
| Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells | 1-gen-2018 | Ayoub, Khalfaoui; Chini, MARIA GIOVANNA; Mohamed, Bouheroum; Soumia, Belaabed; Lauro, Gianluigi; Terracciano, Stefania; Vaccaro, Mariacarmela; Bruno, Ines; Samir, Benayache; Ines, Mancini; Bifulco, Giuseppe | |
| Down regulation of pro-inflammatory pathways by tanshinone IIA and cryptotanshinone in a non-genetic mouse model of Alzheimer's disease | 1-gen-2018 | Maione, Francesco; Piccolo, Marialuisa; DE VITA, Simona; Chini, Maria Giovanna; Cristiano, Claudia; De Caro, Carmen; Lippiello, Pellegrino; Miniaci, Maria Concetta; Santamaria, Rita; Irace, Carlo; De Feo, Vincenzo; Calignano, Antonio; Mascolo, Nicola; Bifulco, Giuseppe | |
| Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain | 1-gen-2018 | Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Guaianolides from Ormenis mixta: Structural Insights and Evaluation of Their Anti-inflammatory Profile | 1-gen-2019 | Benteldjoune, Mounira; Chini, Maria Giovanna; Iannuzzi, Anna Maria; Kabouche, Ahmed; Kabouche, Zahia; Dʼambola, Massimiliano; Marzocco, Stefania; Autore, Giuseppina; Bifulco, Giuseppe; De Tommasi, Nunziatina |
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