SOLVATOCHROMIC PROPERTIES AND SOLID-STATE INCLUSION OF A P-PYRIDINIUM-CALIX[4]ARENE
2018 Iuliano, Veronica; Talotta, C.; Gaeta, C.; Geremia, S.; Hickey, N.; Mennucci, B.; Neri, P.
Solid state self-assembling of resorcin[6]arene macrocycles in a twin molecular capsule
2018 Della Sala, Paolo; Brancatelli, Giovanna; Geremia, Silvano; Talotta, Carmen; De Rosa, Margherita; Neri, Placido; Gaeta, Carmine
On a stochastic model for fluctuating systems under state-dependent dichotomous noise
2018 Di Crescenzo, Antonio; Travaglino, Fabio
PHOTOGRAMMETRY FOR ARCHAEOLOGICAL 3D SURVEYING: THE CASE-STUDY OF PONTE ROTTO ALONG THE ANCIENT APPIA (BENEVENTO, ITALY)
2018 Limongiello, Marco; Barba, Salvatore; Chiara, Germinario; Francesco, Izzo; Gaetano, Memmolo; Musmeci, Daniela; Santoriello, Alfonso
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors
2018 Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G.
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors
2018 Milite, C.; Feoli, A.; Rescigno, Donatella; Pisapia, Vincenzo; Cosconati, S.; Castellano, S.; Sbardella, G.
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins
2017 Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy
2017 Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach
2017 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach
2017 Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
2016 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY
2016 Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors
2015 Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca
Discovery of new chemical probes for the MRG15 chromo domain.
2015 Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20
2015 Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors
2015 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.
2015 Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.
2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.
2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.
2015 Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| SOLVATOCHROMIC PROPERTIES AND SOLID-STATE INCLUSION OF A P-PYRIDINIUM-CALIX[4]ARENE | 1-gen-2018 | Iuliano, Veronica; Talotta, C.; Gaeta, C.; Geremia, S.; Hickey, N.; Mennucci, B.; Neri, P. | |
| Solid state self-assembling of resorcin[6]arene macrocycles in a twin molecular capsule | 1-gen-2018 | Della Sala, Paolo; Brancatelli, Giovanna; Geremia, Silvano; Talotta, Carmen; De Rosa, Margherita; Neri, Placido; Gaeta, Carmine | |
| On a stochastic model for fluctuating systems under state-dependent dichotomous noise | 1-gen-2018 | Di Crescenzo, Antonio; Travaglino, Fabio | |
| PHOTOGRAMMETRY FOR ARCHAEOLOGICAL 3D SURVEYING: THE CASE-STUDY OF PONTE ROTTO ALONG THE ANCIENT APPIA (BENEVENTO, ITALY) | 1-gen-2018 | Limongiello, Marco; Barba, Salvatore; Chiara, Germinario; Francesco, Izzo; Gaetano, Memmolo; Musmeci, Daniela; Santoriello, Alfonso | |
| Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors | 1-gen-2018 | Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G. | |
| Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors | 1-gen-2018 | Milite, C.; Feoli, A.; Rescigno, Donatella; Pisapia, Vincenzo; Cosconati, S.; Castellano, S.; Sbardella, G. | |
| Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins | 1-gen-2017 | Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of new KDM4 inhibitors through a HTS and hit refinement strategy | 1-gen-2017 | Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca | |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach | 1-gen-2017 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach | 1-gen-2017 | Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH | 1-gen-2016 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
| IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY | 1-gen-2016 | Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
| Discovery of new chemical probes for the MRG15 chromo domain. | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors | 1-gen-2015 | Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. | 1-gen-2015 | Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca |
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Scopri
Tipologia
- 4 Contributo in Atti convegno(ex ...556
Data di pubblicazione
- In corso di stampa2
- 2020 - 2026113
- 2010 - 2019326
- 2000 - 200994
- 1990 - 199913
- 1983 - 19898
Editore
- Antonella Rossi4
- Association for computing machinery2
- ASSOCIAZIONE ITALIANA D'INGEGNERI...2
- edita.me2
- Edizioni Scientifiche Italiane2
- Giunti OS psychometrics2
- Il Mulino2
- MV Congressi2
- National Meeting on Medicinal Che...2
- Pandemos s.r.l.2
Rivista
- GIORNALE ITALIANO DI NEFROLOGIA4
- NEUROLOGICAL SCIENCES4
- EUROPEAN RESPIRATORY JOURNAL2
- URBANISTICA INFORMAZIONI2
- ALZHEIMER'S & DEMENTIA1
- FARADAY DISCUSSIONS1
- GIORNALE ITALIANO DI NEFROLOGIA1
- JOURNAL OF HUMAN SPORT AND EXERCISE1
- MEDITERRANEAN JOURNAL OF CLINICAL...1
- MISCELLANEA INGV1
Serie
- MISCELLANEA INGV3
Keyword
- boron cluster3
- Urban planning3
- Clustering2
- CPTED2
- efficienza energetica2
- ESI2
- Extraction2
- Inulin2
- liposome2
- PEF2
Lingua
- eng3
Accesso al fulltext
- no fulltext556