Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach
2017 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach
2017 Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
2016 Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY
2016 Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors
2015 Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca
Discovery of new chemical probes for the MRG15 chromo domain.
2015 Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20
2015 Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors
2015 Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.
2015 Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.
2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.
2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.
2015 Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
2015 Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina
Sunset. Belong to nature
2017 Cucco, Pasquale
Zero, bellezza senza sprechi
2017 Cucco, Pasquale; Giuditta, Serena
A potential estimates approach to a priori estimates for elliptic equations
2015 Mamedov, Farman; Monsurro', Sara; Transirico, Maria
LA INGENIERÍA BIM PARA EL DISEÑO DE LA ARQUITECTURA
2018 Barba, Salvatore; Barbato, Davide; Ferreyra, Carla
Synthesis of bifunctional calixarene hosts
2018 Iuliano, Veronica; Talotta, Carmen; Gaeta, Carmine; DE ROSA, Margherita; Soriente, Annunziata; Neri, Placido
Characterization of the seismic dynamical state of Ischia Volcanic Island (Italy) through the ICA and the polarization analysis applied to background seismic noise
2018 Cusano, P.; Petrosino, S.; Falanga, M.; De Lauro, E.; De Martino, S.
Seismic polarization of LP and VT earthquakes at Campi Flegrei by ICAP
2018 De Lauro, E.; Falanga, M.; De Martino, S.; Petrosino, S.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach | 1-gen-2017 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach | 1-gen-2017 | Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH | 1-gen-2016 | Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
| IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY | 1-gen-2016 | Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
| Discovery of new chemical probes for the MRG15 chromo domain. | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 | 1-gen-2015 | Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors | 1-gen-2015 | Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. | 1-gen-2015 | Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. | 1-gen-2015 | Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. | 1-gen-2015 | Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. | 1-gen-2015 | Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
| Sunset. Belong to nature | 1-gen-2017 | Cucco, Pasquale | |
| Zero, bellezza senza sprechi | 1-gen-2017 | Cucco, Pasquale; Giuditta, Serena | |
| A potential estimates approach to a priori estimates for elliptic equations | 1-gen-2015 | Mamedov, Farman; Monsurro', Sara; Transirico, Maria | |
| LA INGENIERÍA BIM PARA EL DISEÑO DE LA ARQUITECTURA | 1-gen-2018 | Barba, Salvatore; Barbato, Davide; Ferreyra, Carla | |
| Synthesis of bifunctional calixarene hosts | 1-gen-2018 | Iuliano, Veronica; Talotta, Carmen; Gaeta, Carmine; DE ROSA, Margherita; Soriente, Annunziata; Neri, Placido | |
| Characterization of the seismic dynamical state of Ischia Volcanic Island (Italy) through the ICA and the polarization analysis applied to background seismic noise | 1-gen-2018 | Cusano, P.; Petrosino, S.; Falanga, M.; De Lauro, E.; De Martino, S. | |
| Seismic polarization of LP and VT earthquakes at Campi Flegrei by ICAP | 1-gen-2018 | De Lauro, E.; Falanga, M.; De Martino, S.; Petrosino, S. |
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Scopri
Tipologia
- 4 Contributo in Atti convegno(ex ...568
Data di pubblicazione
- In corso di stampa2
- 2020 - 2026125
- 2010 - 2019326
- 2000 - 200994
- 1990 - 199913
- 1983 - 19898
Editore
- Antonella Rossi4
- Association for computing machinery2
- ASSOCIAZIONE ITALIANA D'INGEGNERI...2
- edita.me2
- Edizioni Scientifiche Italiane2
- Giunti OS psychometrics2
- Il Mulino2
- MV Congressi2
- National Meeting on Medicinal Che...2
- Pandemos s.r.l.2
Rivista
- GIORNALE ITALIANO DI NEFROLOGIA4
- NEUROLOGICAL SCIENCES4
- EUROPEAN RESPIRATORY JOURNAL2
- URBANISTICA INFORMAZIONI2
- ALZHEIMER'S & DEMENTIA1
- FARADAY DISCUSSIONS1
- GIORNALE ITALIANO DI NEFROLOGIA1
- JOURNAL OF HUMAN SPORT AND EXERCISE1
- MEDITERRANEAN JOURNAL OF CLINICAL...1
- MISCELLANEA INGV1
Serie
- MISCELLANEA INGV3
Keyword
- boron cluster3
- Fluorescence3
- Urban planning3
- Clustering2
- CPTED2
- efficienza energetica2
- ESI2
- Extraction2
- H2S sensors2
- Inulin2
Lingua
- eng3
Accesso al fulltext
- no fulltext568