Sfoglia per Autore
Effects of FR235222, a novel HDAC inhibitor, in proliferation and apoptosis of human leukaemia cell lines: role of annexin A1
2008-01-01 Petrella, Antonello; D'Acunto, Cw; Rodriquez, Manuela; Festa, M; Tosco, Alessandra; Bruno, Ines; Terracciano, Stefania; Taddei, M; Paloma, Lg; Parente, Luca
Build/couple/pair strategy: From nonchiral molecules to unbiased scaffolds, a methodological approach for the optimization of microwave-assisted intra-molecular Diels-Alder reaction of furans
2008-01-01 Rodriquez, Manuela; Uchida, Takuya; Provost, Alan; Schreiber, Stuart L.
Microwaves enhance cyclisation of tetrapeptides
2009-01-01 Cini, Elena; BOTTA CINZIA, B; Rodriquez, Manuela; Taddei, Maurizio
Skeletally Diverse Small Molecules Using a Build/Couple/Pair Strategy
2009-01-01 Takuya, Uchida; Rodriquez, Manuela; STUART L., Schreiber
Synthesis and application in SPPS of a stable amino acid isoster of palmitoyl cysteine
2009-01-01 Cini, Elena; LAMPARIELLO L., Raffaella; Rodriquez, Manuela; Taddei, Maurizio
Transformation of Glutamic Acid into (S)-Benzyl 2-(dibenzylamino)-6-(dimethoxyphosphoryl)-5-oxohexanoate for a Convenient Access to 5-Substituted Prolines
2009-01-01 Elena, Cini; Gianluca, Giorgi; Rodriquez, Manuela; Maurizio, Taddei
Histone deacetylase inhibitor FR235222 sensitizes human prostate adenocarcinoma cells to apoptosis through up-regulation of annexin A1.
2010-01-01 COSIMO WALTER D’, Acunto; Fontanella, Bianca; Rodriquez, Manuela; Maurizio, Taddei; Parente, Luca; Petrella, Antonello
LGP1, a histone deacetylase inhibitor analogue of FR235222, sensitizes promyelocytic leukemia U937 cells to TRAIL-mediated apoptosis
2010-01-01 Cosimo Walter, D'Acunto; Anna, Carratù; Rodriquez, Manuela; Maurizio, Taddei; Parente, Luca; Petrella, Antonello
Oxime amides as a novel zinc binding group in histone deacetylase inhibitors: synthesis, biological activity, and computational evaluation
2011-01-01 Botta, Cb; Cabri, W; Cini, E; De Cesare, L; Fattorusso, C; Giannini, G; Persico, M; Petrella, Antonello; Rondinelli, F; Rodriquez, Manuela; Russo, A; Taddei, M.
Histone Deacetylase Inhibitors in the Treatment of Hematological Malignancies
2011-01-01 Petrella, Antonello; Fontanella, B; Carratù, A; Bizzarro, Valentina; Rodriquez, Manuela; Parente, Luca
Synthesis of Enantiopure 7-Substituted Azepane-2-Carboxylic Acids as Templates for Conformationally Constrained Peptidomimetics
2012-01-01 Cini, Elena; Bifulco, Giuseppe; Menchi, Gloria; Rodriquez, Manuela; Taddei, Maurizio
Histone deacetylase inhibitors in the treatment of cancer: overview and perspectives
2012-01-01 Giuseppe, Giannini; Walter, Cabri; Caterina, Fattorusso; Rodriquez, Manuela
Downregulation of Hypoxia-related Responses by Novel Antitumor Histone Deacetylase Inhibitors in MDAMB231 Breast Cancer Cells
2012-01-01 Naldini, Antonella; Filippi, Irene; Cini, Elena; Rodriquez, Manuela; Carraro, Fabio; Taddei, Maurizio
Sintesi di derivati SAHA-like utilizzati per indagare sulla selettività verso le diverse isoforme HDAC
2013-01-01 Daniela, Acunzo; Cristina, Aversa; Alessia De, Palma; Randino, Rosario; Rodriquez, Manuela
Gentamicina: derivatizzazione molecolare per migliorare la maneggevolezza sintetica e la farmacocinetica
2013-01-01 Daniel Salvatore, Cretoso; Federica, Agliata; Ruggiero, Ricci; Randino, Rosario; Crescenzi, Carlo; Rodriquez, Manuela
STEROIDAL HYDROXAMIC ACID DERIVATIVES: A STRUCTURALLY NOVEL CLASS OF HDAC INHIBITORS
2014-01-01 Randino, Rosario; Elena, Cini; Maurizio, Taddei; Rodriquez, Manuela
STRUCTURAL FEATURES OF PEPTIDES DERIVED FROM FELINE IMMUNODEFICIENCY VIRUS TM-GLYCOPROTEIN
2014-01-01 Rodriquez, Manuela; Randino, Rosario; Grimaldi, Manuela; Palisi, Angelica; D'Ursi, Anna Maria
TRYPTOPHAN-BASED LINEAR DIPEPTIDES AND 1,4-DIKETOPIPERAZINES AS SIMPLIFIED SCAFFOLDS OF THE NATURAL CYCLOTETRAPEPTIDE FR235222
2014-01-01 Rodriquez, Manuela; Elena, Cini; Elena, Petricci; D'Ursi, Anna Maria; Saturnino, Carmela; Randino, Rosario
SYNTHESIS AND BIOLOGICAL EVALUATION OF SMALL MOLECULES DERIVATIVES OF THE NATURAL HISTONE DEACETYLASE INHIBITOR FR235222
2014-01-01 Randino, Rosario; Elena, Cini; D'Ursi, Anna Maria; Elena, Petricci; Rodriquez, Manuela
Facile Baeyer–Villiger oxidation of cyclic ketones: conventional versus microwave-assisted approach
2015-01-01 Randino, Rosario; Cini, Elena; D'Ursi, Anna Maria; Novellino, Ettore; Rodriquez, Manuela
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