CASTELLANO, Sabrina

CASTELLANO, Sabrina  

Dipartimento di Farmacia/DIFARMA  

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11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 1-gen-2017 Ikawa, Masamichi; Lohith, Talakad G; Shrestha, Stal; Telu, Sanjay; Zoghbi, Sami S; Castellano, Sabrina; Taliani, Sabrina; Da Settimo, Federico; Fujita, Masahiro; Pike, Victor W; Innis, Robert B.
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 1-gen-2006 Rizzetto, E; Castellano, Sabrina; Florio, C; Vadori, M; Stefancich, G.
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 1-gen-2006 Sbardella, Gianluca; Bartolini, S; Castellano, Sabrina; Artico, M; Paesano, N; Rotili, D; Spadafora, C; Mai, A.
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 1-gen-2000 Dallanoce, C.; DE AMICI, M.; Carrea, G.; Secundo, F.; Castellano, Sabrina; DE MICHELI, C.
A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors 1-gen-2023 Donati, Greta; Viviano, Monica; D'Amore, Vincenzo Maria; Cipriano, Alessandra; Diakogiannaki, Isidora; Amato, Jussara; Tomassi, Stefano; Brancaccio, Diego; Russomanno, Pasquale; Di Leva, Francesco Saverio; Arosio, Daniela; Seneci, Pierfausto; Taliani, Sabrina; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Skalniak, Lukasz; Holak, Tad A; Castellano, Sabrina; La Pietra, Valeria; Marinelli, Luciana
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 1-gen-2015 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 1-gen-2015 Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 1-gen-2000 Castellano, Sabrina; Stefancich, G.; Musiu, C.; LA COLLA, P.
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 1-gen-2015 Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 1-gen-2008 Castellano, Sabrina; Bertamino, Alessia; Gomez Monterrey, Isabel; Santoriello, Marisabella; Grieco, Paolo; Campiglia, Pietro; Sbardella, Gianluca; Novellino, Ettore
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 1-gen-2009 Castellano, Sabrina; Santoriello, Marisabella; Campiglia, Pietro; Cardillo, Giovanna; Bertamino, Alessia; Gomez Monterrey, Isabel; Novellino, Ettore; Sbardella, Gianluca
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 1-gen-2011 M., Vecellio; G., Pompilio; F., Spallotta; C., Colussi; Sbardella, Gianluca; Castellano, Sabrina; A., Mai; M. C., Capogrossi; A., Rossini; C., Gaetano
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 1-gen-2022 Creighton, Samantha D.; Jardine, Kristen H.; Desimone, Alexa; Zmetana, Megan; Castellano, Sabrina; Milite, Ciro; Sbardella, Gianluca; Winters, Boyer D.
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 1-gen-2013 Calabrese, ELENA CONCETTA; Castellano, Sabrina; M., Santoriello; C., Sgherri; M. F., Quartacci; L., Calucci; A. G. S., Warrilow; D. C., Lamb; S. L., Kelly; Milite, Ciro; Granata, Ilaria; Sbardella, Gianluca; G., Stefancich; Maresca, Bruno; Porta, Amalia
Antimycobacterial activity of ionic fullerene derivatives. 1-gen-2000 Bosi, S.; DA ROS, T.; Castellano, Sabrina; Banfi, E.; Prato, M.
Azole antifungal agents related to naftifine and butenafine 1-gen-2000 Castellano, Sabrina; LA COLLA, P.; Musiu, C.; Stefancich, G.
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 1-gen-2015 Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 1-gen-2015 Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E.
Chemical biology of Histone acetyltransferase natural compounds modulators. 1-gen-2011 DAL PIAZ, Fabrizio; Vassallo, Antonio; Osmany Cuesta, Rubio; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 1-gen-2015 Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca