UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 10.545
NA - Nord America 3.554
EU - Europa 1.444
SA - Sud America 455
AF - Africa 64
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 2
Totale 16.068
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Nazione #
HK - Hong Kong 8.892
US - Stati Uniti d'America 3.458
SG - Singapore 790
IT - Italia 520
BR - Brasile 378
CN - Cina 342
RU - Federazione Russa 244
VN - Vietnam 208
DE - Germania 188
UA - Ucraina 107
IE - Irlanda 81
TR - Turchia 67
IN - India 61
KR - Corea 56
CA - Canada 52
GB - Regno Unito 52
SE - Svezia 50
FI - Finlandia 46
JP - Giappone 37
AR - Argentina 36
MX - Messico 32
NL - Olanda 31
AT - Austria 27
ID - Indonesia 23
ZA - Sudafrica 23
DZ - Algeria 20
PL - Polonia 20
ES - Italia 18
BD - Bangladesh 17
CZ - Repubblica Ceca 17
FR - Francia 15
CO - Colombia 11
EC - Ecuador 11
IQ - Iraq 11
PK - Pakistan 11
MA - Marocco 8
CH - Svizzera 6
PY - Paraguay 6
CL - Cile 5
UZ - Uzbekistan 5
BE - Belgio 4
RO - Romania 4
SA - Arabia Saudita 4
AZ - Azerbaigian 3
DK - Danimarca 3
EU - Europa 3
HU - Ungheria 3
IL - Israele 3
PE - Perù 3
AE - Emirati Arabi Uniti 2
BH - Bahrain 2
DO - Repubblica Dominicana 2
EG - Egitto 2
GA - Gabon 2
GT - Guatemala 2
JM - Giamaica 2
JO - Giordania 2
KE - Kenya 2
LU - Lussemburgo 2
NG - Nigeria 2
NI - Nicaragua 2
TN - Tunisia 2
UY - Uruguay 2
VE - Venezuela 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AL - Albania 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
CU - Cuba 1
CY - Cipro 1
GE - Georgia 1
GN - Guinea 1
GY - Guiana 1
KI - Kiribati 1
KZ - Kazakistan 1
LB - Libano 1
LC - Santa Lucia 1
LT - Lituania 1
MC - Monaco 1
MN - Mongolia 1
PA - Panama 1
PT - Portogallo 1
QA - Qatar 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
SY - Repubblica araba siriana 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
ZM - Zambia 1
Totale 16.068
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Città #
Hong Kong 8.879
Dallas 689
Ann Arbor 558
Singapore 370
Chandler 326
Ashburn 213
Princeton 198
Woodbridge 151
Wilmington 145
Jacksonville 142
Salerno 90
Munich 84
Dublin 80
Beijing 76
Houston 69
Los Angeles 65
Naples 64
Ho Chi Minh City 63
Izmir 52
Moscow 43
Fisciano 42
Hanoi 39
Dong Ket 38
New York 38
São Paulo 38
Tokyo 34
Andover 33
Montreal 31
Turku 28
Dearborn 26
Nanjing 26
Pellezzano 26
Columbus 23
Nuremberg 22
The Dalles 21
Boardman 20
Brooklyn 20
Johannesburg 19
Denver 18
Santa Clara 18
Redwood City 16
Seattle 16
Warsaw 16
Brno 15
Chennai 14
Phoenix 14
Afragola 12
Belo Horizonte 12
Boston 12
Mexico City 12
Stockholm 12
Vienna 12
Washington 12
Amsterdam 11
Fairfield 11
Jiaxing 11
Nanchang 11
Orem 11
Seoul 11
Curitiba 10
Frankfurt am Main 10
Lucca 10
Mestre 10
Milan 10
Atlanta 9
Chicago 9
Düsseldorf 9
London 9
Pune 9
El Hadjira 8
Jakarta 8
Manchester 8
Poplar 8
Rome 8
Sarno 8
Shanghai 8
Shenyang 8
West Jordan 8
Campinas 7
Council Bluffs 7
Da Nang 7
Hebei 7
Hải Dương 7
Jinan 7
Napoli 7
New Delhi 7
Tianjin 7
Chandigarh 6
Chengdu 6
Fes 6
Haiphong 6
Mumbai 6
Norwalk 6
Ortona 6
Redondo Beach 6
San Francisco 6
Toronto 6
Uster 6
Ankara 5
Bogotá 5
Totale 13.464
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.193
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.103
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 921
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 579
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 558
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 539
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 501
Target identification by structure-based computational approaches: Recent advances and perspectives 446
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 417
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 385
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 375
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 304
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 284
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 273
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 235
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 227
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 225
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 198
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 187
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 175
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 167
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 162
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 153
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 151
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 149
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 144
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 141
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 129
Anti-inflammatory trends of new benzimidazole derivatives 129
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 126
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 120
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 113
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 112
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 110
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 110
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 108
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 108
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 106
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 105
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 104
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 102
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 101
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 97
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 97
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 97
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 96
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 96
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 94
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 92
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 92
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 91
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 90
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 89
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 88
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 86
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 84
Discovery of noscapine derivatives as potential β-tubulin inhibitors 84
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 83
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 80
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 80
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 78
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 77
Reranking docking poses using molecular simulations and approximate free energy methods 75
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 74
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 73
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 72
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 70
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 69
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 68
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 67
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 67
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 66
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 65
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 65
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 64
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 63
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 62
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 62
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 62
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 57
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 56
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 55
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 50
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 49
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 48
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 45
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 32
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 31
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 30
Identification and Development of BRD9 Chemical Probes 30
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 27
New techniques of molecular modelling and structural chemistry for the development of bioactive compounds 1
Totale 16.301
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Categoria #
all - tutte 39.216
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 39.216
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021255 0 0 0 0 0 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/202610.839 3.004 3.426 3.077 610 700 22 0 0 0 0 0 0
Totale 16.301