UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 11.410
NA - Nord America 4.940
EU - Europa 2.264
SA - Sud America 579
Continente sconosciuto - Info sul continente non disponibili 261
AF - Africa 105
OC - Oceania 2
Totale 19.561
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Nazione #
HK - Hong Kong 8.970
US - Stati Uniti d'America 4.777
IT - Italia 1.139
SG - Singapore 1.068
CN - Cina 448
BR - Brasile 440
VN - Vietnam 368
RU - Federazione Russa 251
DE - Germania 217
UA - Ucraina 115
FR - Francia 99
IN - India 99
IE - Irlanda 85
TR - Turchia 80
BD - Bangladesh 77
CA - Canada 76
GB - Regno Unito 71
KR - Corea 63
AR - Argentina 56
SE - Svezia 56
JP - Giappone 49
FI - Finlandia 47
MX - Messico 46
NL - Olanda 38
IQ - Iraq 35
ZA - Sudafrica 32
ID - Indonesia 30
AT - Austria 28
DZ - Algeria 26
PL - Polonia 25
ES - Italia 24
CO - Colombia 21
CZ - Repubblica Ceca 21
EC - Ecuador 21
PK - Pakistan 21
SA - Arabia Saudita 16
MA - Marocco 14
PH - Filippine 12
UZ - Uzbekistan 12
CL - Cile 11
VE - Venezuela 10
CH - Svizzera 9
HU - Ungheria 9
JM - Giamaica 8
AZ - Azerbaigian 7
CR - Costa Rica 7
PY - Paraguay 7
TT - Trinidad e Tobago 7
MY - Malesia 6
EG - Egitto 5
JO - Giordania 5
KE - Kenya 5
NP - Nepal 5
PE - Perù 5
UY - Uruguay 5
BE - Belgio 4
BH - Bahrain 4
GT - Guatemala 4
IL - Israele 4
KZ - Kazakistan 4
NI - Nicaragua 4
PT - Portogallo 4
RO - Romania 4
AL - Albania 3
DK - Danimarca 3
DO - Repubblica Dominicana 3
EU - Europa 3
LT - Lituania 3
OM - Oman 3
TH - Thailandia 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
BO - Bolivia 2
ET - Etiopia 2
GA - Gabon 2
GE - Georgia 2
IR - Iran 2
LB - Libano 2
LU - Lussemburgo 2
NG - Nigeria 2
PR - Porto Rico 2
PS - Palestinian Territory 2
QA - Qatar 2
SN - Senegal 2
SY - Repubblica araba siriana 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
BJ - Benin 1
BN - Brunei Darussalam 1
BY - Bielorussia 1
CI - Costa d'Avorio 1
CU - Cuba 1
CY - Cipro 1
GD - Grenada 1
GN - Guinea 1
GP - Guadalupe 1
GY - Guiana 1
HR - Croazia 1
Totale 19.283
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Città #
Hong Kong 8.949
Dallas 696
Singapore 575
Ann Arbor 558
San Jose 468
Milan 340
Chandler 326
Ashburn 314
Princeton 198
Woodbridge 151
Wilmington 146
Jacksonville 143
Beijing 121
Ho Chi Minh City 118
Council Bluffs 114
Salerno 100
The Dalles 91
Naples 86
Los Angeles 85
Dublin 84
Munich 84
Rome 84
Lauterbourg 76
Hanoi 74
Santa Clara 73
Houston 71
New York 63
Izmir 53
Fisciano 46
Tokyo 46
São Paulo 45
Moscow 44
Memphis 42
Dong Ket 38
Montreal 37
Andover 33
Frankfurt am Main 28
Turku 28
Figino 27
Dearborn 26
Nanjing 26
Pellezzano 26
Brooklyn 23
Columbus 23
Nuremberg 23
Orem 23
Denver 22
Boardman 21
Johannesburg 21
Warsaw 21
Chennai 19
Da Nang 19
Mexico City 19
Seattle 18
Stockholm 18
Chicago 17
Phoenix 17
Washington 17
London 16
Redwood City 16
Brno 15
Chengdu 15
Turin 15
Amsterdam 14
Haiphong 14
Atlanta 13
Baghdad 13
Belo Horizonte 13
Hải Dương 13
Afragola 12
Boston 12
Vienna 12
Fairfield 11
Jiaxing 11
Lucca 11
Montoro 11
Nanchang 11
Poplar 11
Seoul 11
Toronto 11
Buffalo 10
Campinas 10
Curitiba 10
Istanbul 10
Jakarta 10
Mestre 10
New Delhi 10
Pune 10
San Francisco 10
Düsseldorf 9
Manchester 9
Ninh Bình 9
Pagani 9
Shanghai 9
Tashkent 9
Bogotá 8
El Hadjira 8
Guayaquil 8
Sarno 8
Shenyang 8
Totale 15.519
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.279
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.133
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 946
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 624
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 593
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 562
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 523
Target identification by structure-based computational approaches: Recent advances and perspectives 458
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 453
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 421
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 404
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 373
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 328
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 315
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 308
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 265
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 262
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 235
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 228
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 205
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 197
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 196
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 190
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 178
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 176
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 171
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 167
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 164
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 163
Anti-inflammatory trends of new benzimidazole derivatives 160
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 153
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 151
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 148
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 145
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 144
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 142
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 137
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 136
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 136
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 135
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 134
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 133
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 132
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 132
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 131
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 127
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 126
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 123
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 120
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 119
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 118
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 118
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 118
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 117
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 114
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 112
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 112
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 111
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 111
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 110
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 108
Discovery of noscapine derivatives as potential β-tubulin inhibitors 107
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 107
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 107
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 103
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 100
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 99
Reranking docking poses using molecular simulations and approximate free energy methods 99
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 98
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 97
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 97
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 96
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 95
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 94
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 93
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 92
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 90
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 87
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 84
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 84
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 83
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 82
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 81
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 78
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 76
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 73
Identification and Development of BRD9 Chemical Probes 63
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 62
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 61
Discovery of RUVBL1 as a Target of the Marine Alkaloid Caulerpin via MS-Based Functional Proteomics 58
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 54
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 46
The Role of LC-MS in Profiling Bioactive Compounds from Plant Waste for Cosmetic Applications: A General Overview 37
A 5-Br-1-Propylisatin Derivative as a Promising BRD9 Ligand: Insights from Computational and STD NMR Investigation 26
Identification of a New Interesting BAG3 Modulator Able to Disrupt Cancer-Related Pathways 26
Unveiling New Triazoloquinoxaline‐Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9 24
Disruption of c-Myc/Max heterodimerization induced by a novel anticancer agent endowed with 1,3-diphenylurea moiety: an in silico, chemoproteomics-based, and in vitro combined approach 20
The future of BRD9 inhibitors: a patent perspective (2019-present) 19
Potential Nutraceutical Properties of Vicia faba L: LC-ESI-HR-MS/MS-Based Profiling of Ancient Faba Bean Varieties and Their Biological Activity 19
Carnosol modulates mPGES-1/PPAR-γ biological axis: from in silico to in vivo clinical imaging and investigations 17
Totale 19.464
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Categoria #
all - tutte 47.834
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 47.834
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022390 0 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/202613.710 3.004 3.426 3.077 610 700 276 708 157 269 647 237 599
2026/2027389 329 60 0 0 0 0 0 0 0 0 0 0
Totale 19.561