UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 9.763
NA - Nord America 3.076
EU - Europa 1.310
SA - Sud America 242
AF - Africa 42
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 2
Totale 14.439
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Nazione #
HK - Hong Kong 8.859
US - Stati Uniti d'America 3.019
IT - Italia 460
SG - Singapore 361
CN - Cina 250
RU - Federazione Russa 240
BR - Brasile 215
DE - Germania 183
UA - Ucraina 101
IE - Irlanda 80
VN - Vietnam 77
TR - Turchia 58
IN - India 47
KR - Corea 43
SE - Svezia 43
FI - Finlandia 42
GB - Regno Unito 33
CA - Canada 32
NL - Olanda 26
AT - Austria 24
DZ - Algeria 20
JP - Giappone 18
CZ - Repubblica Ceca 17
MX - Messico 17
FR - Francia 15
ES - Italia 12
BD - Bangladesh 11
PL - Polonia 9
AR - Argentina 8
MA - Marocco 8
ZA - Sudafrica 8
ID - Indonesia 7
CH - Svizzera 6
EC - Ecuador 6
IQ - Iraq 6
BE - Belgio 4
CO - Colombia 4
PK - Pakistan 4
SA - Arabia Saudita 4
UZ - Uzbekistan 4
EU - Europa 3
HU - Ungheria 3
RO - Romania 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
DO - Repubblica Dominicana 2
JO - Giordania 2
LU - Lussemburgo 2
NI - Nicaragua 2
PE - Perù 2
PY - Paraguay 2
UY - Uruguay 2
VE - Venezuela 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AL - Albania 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
BH - Bahrain 1
CL - Cile 1
CU - Cuba 1
DK - Danimarca 1
EG - Egitto 1
GE - Georgia 1
GN - Guinea 1
GT - Guatemala 1
IL - Israele 1
JM - Giamaica 1
KE - Kenya 1
KI - Kiribati 1
KZ - Kazakistan 1
LT - Lituania 1
MC - Monaco 1
NG - Nigeria 1
PT - Portogallo 1
QA - Qatar 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
SY - Repubblica araba siriana 1
TN - Tunisia 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
Totale 14.439
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Città #
Hong Kong 8.847
Ann Arbor 558
Dallas 524
Chandler 326
Princeton 198
Singapore 161
Ashburn 153
Woodbridge 151
Wilmington 145
Jacksonville 142
Munich 84
Salerno 84
Dublin 80
Houston 61
Izmir 52
Beijing 50
Naples 48
Moscow 43
Dong Ket 38
Fisciano 37
Los Angeles 34
Andover 33
Dearborn 26
Nanjing 26
Pellezzano 26
Turku 24
Columbus 23
Nuremberg 22
Boardman 20
Montreal 19
São Paulo 19
The Dalles 19
New York 17
Brooklyn 16
Redwood City 16
Brno 15
Ho Chi Minh City 15
Tokyo 15
Seattle 14
Hanoi 13
Afragola 12
Washington 12
Fairfield 11
Jiaxing 11
Nanchang 11
Vienna 11
Mestre 10
Belo Horizonte 9
Düsseldorf 9
Pune 9
Santa Clara 9
Boston 8
Chicago 8
El Hadjira 8
Sarno 8
Shanghai 8
Shenyang 8
West Jordan 8
Chennai 7
Council Bluffs 7
Hebei 7
Jinan 7
Johannesburg 7
Napoli 7
Rome 7
Tianjin 7
Amsterdam 6
Chandigarh 6
Fes 6
London 6
Mexico City 6
Milan 6
Norwalk 6
Ortona 6
Phoenix 6
Redondo Beach 6
San Francisco 6
Uster 6
Caivano 5
Campinas 5
Cava de' Tirreni 5
Denver 5
Domicella 5
Frankfurt am Main 5
Guangzhou 5
Jakarta 5
New Delhi 5
Nocera Superiore 5
Pozzuoli 5
San Diego 5
Stockholm 5
Toronto 5
Warsaw 5
Arzano 4
Casagiove 4
Caserta 4
Charlotte 4
Curitiba 4
Dormagen 4
Mumbai 4
Totale 12.595
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.129
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.085
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 903
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 561
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 542
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 523
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 490
Target identification by structure-based computational approaches: Recent advances and perspectives 437
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 411
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 363
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 362
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 292
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 264
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 261
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 216
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 204
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 176
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 174
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 171
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 160
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 154
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 153
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 142
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 137
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 125
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 124
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 123
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 118
Anti-inflammatory trends of new benzimidazole derivatives 117
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 107
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 105
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 103
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 100
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 100
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 98
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 96
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 95
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 92
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 91
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 90
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 87
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 86
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 86
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 85
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 84
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 81
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 81
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 77
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 75
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 75
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 72
Discovery of noscapine derivatives as potential β-tubulin inhibitors 72
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 63
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 63
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 63
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 62
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 62
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 60
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 60
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 60
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 59
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 57
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 57
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 56
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 55
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 55
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 54
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 53
Reranking docking poses using molecular simulations and approximate free energy methods 52
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 51
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 48
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 48
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 43
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 41
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 38
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 37
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 35
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 34
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 33
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 33
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 32
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 31
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 30
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 28
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 27
Identification and Development of BRD9 Chemical Probes 25
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 24
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 24
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 22
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 22
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 20
Totale 14.672
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Categoria #
all - tutte 34.445
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 34.445
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021304 0 0 22 0 27 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/20269.210 3.004 3.426 2.780 0 0 0 0 0 0 0 0 0
Totale 14.672