UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
NA - Nord America 2.225
EU - Europa 1.103
AS - Asia 677
SA - Sud America 143
AF - Africa 28
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 1
Totale 4.181
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Nazione #
US - Stati Uniti d'America 2.203
IT - Italia 406
SG - Singapore 292
RU - Federazione Russa 237
CN - Cina 193
BR - Brasile 131
DE - Germania 107
UA - Ucraina 100
IE - Irlanda 79
TR - Turchia 57
SE - Svezia 40
VN - Vietnam 38
KR - Corea 29
IN - India 25
FI - Finlandia 18
GB - Regno Unito 18
HK - Hong Kong 18
NL - Olanda 18
AT - Austria 17
CZ - Repubblica Ceca 17
DZ - Algeria 16
FR - Francia 13
ES - Italia 10
MX - Messico 10
CA - Canada 8
MA - Marocco 8
CH - Svizzera 6
JP - Giappone 5
AR - Argentina 4
BE - Belgio 4
PL - Polonia 4
SA - Arabia Saudita 4
EC - Ecuador 3
EU - Europa 3
IQ - Iraq 3
PK - Pakistan 3
HU - Ungheria 2
JO - Giordania 2
LU - Lussemburgo 2
ZA - Sudafrica 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AE - Emirati Arabi Uniti 1
AU - Australia 1
AZ - Azerbaigian 1
BD - Bangladesh 1
BG - Bulgaria 1
CL - Cile 1
CO - Colombia 1
DK - Danimarca 1
GE - Georgia 1
GT - Guatemala 1
ID - Indonesia 1
JM - Giamaica 1
KE - Kenya 1
KZ - Kazakistan 1
MC - Monaco 1
NI - Nicaragua 1
PE - Perù 1
PT - Portogallo 1
PY - Paraguay 1
QA - Qatar 1
SK - Slovacchia (Repubblica Slovacca) 1
TN - Tunisia 1
TT - Trinidad e Tobago 1
UZ - Uzbekistan 1
VE - Venezuela 1
Totale 4.181
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Città #
Ann Arbor 558
Chandler 326
Princeton 198
Woodbridge 151
Wilmington 145
Jacksonville 142
Ashburn 111
Singapore 103
Salerno 84
Dublin 79
Houston 61
Izmir 52
Moscow 43
Dong Ket 38
Fisciano 34
Andover 33
Beijing 32
Dearborn 26
Nanjing 26
Naples 26
Pellezzano 26
Boardman 20
Hong Kong 17
Munich 17
Redwood City 16
Brno 15
Nuremberg 14
Los Angeles 13
Seattle 13
Afragola 12
Washington 12
Fairfield 11
Jiaxing 11
Nanchang 11
São Paulo 11
Dallas 10
Mestre 10
Düsseldorf 9
Pune 9
Sarno 8
Shanghai 8
Shenyang 8
Vienna 8
Council Bluffs 7
Hebei 7
Jinan 7
Napoli 7
Tianjin 7
Fes 6
Norwalk 6
Ortona 6
Uster 6
Amsterdam 5
Caivano 5
Cava de' Tirreni 5
Chicago 5
Domicella 5
Guangzhou 5
Milan 5
Nocera Superiore 5
Pozzuoli 5
San Diego 5
West Jordan 5
Arzano 4
Belo Horizonte 4
Campinas 4
Casagiove 4
Dormagen 4
El Hadjira 4
Frankfurt am Main 4
Montreal 4
New York 4
Pignola 4
Pomigliano d'Arco 4
Rome 4
Santander 4
The Dalles 4
Buonabitacolo 3
Cambridge 3
Cardito 3
Changsha 3
Granada 3
Guarulhos 3
Hortolândia 3
London 3
Mexico City 3
Mumbai 3
New Delhi 3
Nürnberg 3
Purley 3
Ravenna 3
Spinea 3
São Bernardo do Campo 3
Taranto 3
Tokyo 3
Torre Annunziata 3
Altavilla Silentina 2
Amman 2
Antalya 2
Araraquara 2
Totale 2.792
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Nome #
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 158
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 132
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 131
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 117
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 115
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 111
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 109
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 109
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 101
Anti-inflammatory trends of new benzimidazole derivatives 100
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 94
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 94
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 93
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 92
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 91
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 85
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 85
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 84
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 84
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 83
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 81
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 79
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 76
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 74
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 73
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 72
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 69
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 66
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 65
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 64
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 62
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 57
Discovery of noscapine derivatives as potential β-tubulin inhibitors 56
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 54
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 53
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 50
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 48
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 47
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 46
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 45
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 43
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 43
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 43
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 42
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 42
Reranking docking poses using molecular simulations and approximate free energy methods 41
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 41
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 39
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 39
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 39
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 39
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 38
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 33
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 33
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 31
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 31
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 30
Predicting PROTAC-mediated ternary complex structures through in silico approaches 29
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 28
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 28
Target identification by structure-based computational approaches: Recent advances and perspectives 26
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 25
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 24
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 24
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 21
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 21
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 21
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 18
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 16
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 14
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 13
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 13
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 13
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 12
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 10
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 10
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 10
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 10
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 8
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 8
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 8
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 7
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 7
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 6
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 6
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 6
Identification and Development of BRD9 Chemical Probes 6
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 6
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 5
Totale 4.411
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Categoria #
all - tutte 19.400
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 19.400
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/202070 0 0 0 0 0 0 0 0 0 0 56 14
2020/2021334 8 22 22 0 27 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20251.156 58 14 11 71 47 115 388 115 248 73 16 0
Totale 4.411