UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
NA - Nord America 2.390
AS - Asia 1.678
EU - Europa 1.226
SA - Sud America 185
AF - Africa 33
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 2
Totale 5.518
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Nazione #
US - Stati Uniti d'America 2.355
HK - Hong Kong 939
IT - Italia 433
SG - Singapore 311
RU - Federazione Russa 239
CN - Cina 211
BR - Brasile 168
DE - Germania 164
UA - Ucraina 101
IE - Irlanda 79
TR - Turchia 58
VN - Vietnam 49
SE - Svezia 41
KR - Corea 39
FI - Finlandia 33
IN - India 32
GB - Regno Unito 25
NL - Olanda 24
AT - Austria 21
DZ - Algeria 20
CA - Canada 18
CZ - Repubblica Ceca 17
FR - Francia 13
MX - Messico 12
ES - Italia 10
JP - Giappone 8
MA - Marocco 8
BD - Bangladesh 7
CH - Svizzera 6
AR - Argentina 5
IQ - Iraq 5
BE - Belgio 4
EC - Ecuador 4
PK - Pakistan 4
PL - Polonia 4
SA - Arabia Saudita 4
EU - Europa 3
ZA - Sudafrica 3
AE - Emirati Arabi Uniti 2
HU - Ungheria 2
JO - Giordania 2
LU - Lussemburgo 2
RO - Romania 2
UY - Uruguay 2
UZ - Uzbekistan 2
VE - Venezuela 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AU - Australia 1
AZ - Azerbaigian 1
BG - Bulgaria 1
CL - Cile 1
CO - Colombia 1
DK - Danimarca 1
DO - Repubblica Dominicana 1
GE - Georgia 1
GT - Guatemala 1
ID - Indonesia 1
JM - Giamaica 1
KE - Kenya 1
KI - Kiribati 1
KZ - Kazakistan 1
LT - Lituania 1
MC - Monaco 1
NI - Nicaragua 1
PE - Perù 1
PT - Portogallo 1
PY - Paraguay 1
QA - Qatar 1
SK - Slovacchia (Repubblica Slovacca) 1
TN - Tunisia 1
TT - Trinidad e Tobago 1
Totale 5.518
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Città #
Hong Kong 938
Ann Arbor 558
Chandler 326
Princeton 198
Woodbridge 151
Wilmington 145
Jacksonville 142
Ashburn 121
Singapore 114
Salerno 84
Dublin 79
Munich 69
Houston 61
Izmir 52
Beijing 49
Moscow 43
Dong Ket 38
Naples 38
Fisciano 35
Andover 33
Dearborn 26
Nanjing 26
Pellezzano 26
Los Angeles 25
Columbus 23
Boardman 20
Nuremberg 19
The Dalles 19
Dallas 17
Redwood City 16
Brno 15
São Paulo 15
Turku 15
Seattle 14
Afragola 12
Washington 12
Fairfield 11
Jiaxing 11
Nanchang 11
Mestre 10
Montreal 10
Vienna 10
Düsseldorf 9
Pune 9
El Hadjira 8
New York 8
Sarno 8
Shanghai 8
Shenyang 8
West Jordan 8
Belo Horizonte 7
Chicago 7
Council Bluffs 7
Hebei 7
Jinan 7
Napoli 7
Tianjin 7
Amsterdam 6
Brooklyn 6
Fes 6
Ho Chi Minh City 6
London 6
Milan 6
Norwalk 6
Ortona 6
Uster 6
Caivano 5
Cava de' Tirreni 5
Domicella 5
Guangzhou 5
Hanoi 5
Nocera Superiore 5
Pozzuoli 5
San Diego 5
Tokyo 5
Arzano 4
Boston 4
Campinas 4
Casagiove 4
Dormagen 4
Frankfurt am Main 4
Mumbai 4
New Delhi 4
Phoenix 4
Pignola 4
Pomigliano d'Arco 4
Rome 4
San Francisco 4
Santander 4
Toronto 4
Buonabitacolo 3
Cambridge 3
Cardito 3
Changsha 3
Chennai 3
Curitiba 3
Enfield 3
Granada 3
Guarulhos 3
Hortolândia 3
Totale 3.941
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 907
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 170
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 143
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 133
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 121
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 120
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 115
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 115
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 113
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 109
Anti-inflammatory trends of new benzimidazole derivatives 105
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 102
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 98
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 98
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 94
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 93
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 92
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 87
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 87
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 87
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 86
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 86
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 84
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 82
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 80
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 76
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 75
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 74
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 74
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 73
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 72
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 70
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 67
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 63
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 61
Discovery of noscapine derivatives as potential β-tubulin inhibitors 61
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 58
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 53
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 51
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 51
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 51
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 48
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 47
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 46
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 46
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 45
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 45
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 44
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 43
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 43
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 43
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 42
Reranking docking poses using molecular simulations and approximate free energy methods 42
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 42
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 40
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 39
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 38
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 37
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 32
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 30
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 29
Target identification by structure-based computational approaches: Recent advances and perspectives 27
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 27
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 27
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 26
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 25
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 24
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 24
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 23
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 22
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 21
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 18
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 18
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 18
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 17
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 15
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 15
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 14
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 14
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 13
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 13
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 12
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 11
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 11
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 11
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 11
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 11
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 8
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 8
Identification and Development of BRD9 Chemical Probes 8
Totale 5.750
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Categoria #
all - tutte 21.974
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 21.974
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021334 8 22 22 0 27 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/2026288 288 0 0 0 0 0 0 0 0 0 0 0
Totale 5.750