UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 11.331
NA - Nord America 4.676
EU - Europa 1.745
SA - Sud America 571
AF - Africa 105
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 2
Totale 18.434
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Nazione #
HK - Hong Kong 8.949
US - Stati Uniti d'America 4.539
SG - Singapore 1.046
IT - Italia 633
BR - Brasile 436
CN - Cina 421
VN - Vietnam 368
RU - Federazione Russa 251
DE - Germania 217
UA - Ucraina 114
FR - Francia 98
IN - India 98
IE - Irlanda 85
TR - Turchia 80
BD - Bangladesh 70
GB - Regno Unito 70
CA - Canada 65
KR - Corea 63
AR - Argentina 55
SE - Svezia 55
JP - Giappone 49
FI - Finlandia 47
MX - Messico 44
IQ - Iraq 35
NL - Olanda 34
ZA - Sudafrica 32
ID - Indonesia 29
AT - Austria 28
DZ - Algeria 26
PL - Polonia 25
ES - Italia 23
EC - Ecuador 21
PK - Pakistan 21
CO - Colombia 20
CZ - Repubblica Ceca 19
SA - Arabia Saudita 16
MA - Marocco 14
PH - Filippine 12
UZ - Uzbekistan 12
CL - Cile 10
VE - Venezuela 10
CH - Svizzera 9
HU - Ungheria 9
AZ - Azerbaigian 7
JM - Giamaica 7
PY - Paraguay 7
MY - Malesia 6
EG - Egitto 5
JO - Giordania 5
KE - Kenya 5
NP - Nepal 5
PE - Perù 5
BE - Belgio 4
BH - Bahrain 4
IL - Israele 4
KZ - Kazakistan 4
NI - Nicaragua 4
RO - Romania 4
TT - Trinidad e Tobago 4
UY - Uruguay 4
AL - Albania 3
DK - Danimarca 3
DO - Repubblica Dominicana 3
EU - Europa 3
GT - Guatemala 3
LT - Lituania 3
OM - Oman 3
PT - Portogallo 3
TH - Thailandia 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
BO - Bolivia 2
CR - Costa Rica 2
ET - Etiopia 2
GA - Gabon 2
GE - Georgia 2
IR - Iran 2
LB - Libano 2
LU - Lussemburgo 2
NG - Nigeria 2
PS - Palestinian Territory 2
QA - Qatar 2
SN - Senegal 2
SY - Repubblica araba siriana 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
BJ - Benin 1
BN - Brunei Darussalam 1
CI - Costa d'Avorio 1
CU - Cuba 1
CY - Cipro 1
GN - Guinea 1
GY - Guiana 1
HR - Croazia 1
KG - Kirghizistan 1
KI - Kiribati 1
LC - Santa Lucia 1
LK - Sri Lanka 1
Totale 18.416
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Città #
Hong Kong 8.930
Dallas 694
Ann Arbor 558
Singapore 556
San Jose 466
Chandler 326
Ashburn 305
Princeton 198
Woodbridge 151
Wilmington 146
Jacksonville 143
Ho Chi Minh City 118
Council Bluffs 109
Beijing 96
Salerno 96
The Dalles 91
Dublin 84
Munich 84
Naples 82
Los Angeles 81
Lauterbourg 76
Hanoi 74
Houston 70
New York 59
Izmir 53
Santa Clara 50
Fisciano 46
Tokyo 46
Moscow 44
São Paulo 43
Memphis 40
Dong Ket 38
Montreal 35
Andover 33
Frankfurt am Main 28
Turku 28
Dearborn 26
Nanjing 26
Pellezzano 26
Brooklyn 23
Columbus 23
Nuremberg 23
Orem 23
Denver 22
Boardman 21
Johannesburg 21
Warsaw 21
Chennai 19
Da Nang 19
Milan 18
Mexico City 17
Phoenix 17
Seattle 17
Stockholm 17
Chicago 16
London 16
Redwood City 16
Brno 15
Chengdu 15
Haiphong 14
Washington 14
Amsterdam 13
Baghdad 13
Belo Horizonte 13
Hải Dương 13
Rome 13
Afragola 12
Boston 12
Vienna 12
Fairfield 11
Jiaxing 11
Montoro 11
Nanchang 11
Poplar 11
Seoul 11
Toronto 11
Campinas 10
Curitiba 10
Istanbul 10
Lucca 10
Mestre 10
New Delhi 10
Pune 10
San Francisco 10
Atlanta 9
Düsseldorf 9
Jakarta 9
Manchester 9
Ninh Bình 9
Shanghai 9
Tashkent 9
El Hadjira 8
Guayaquil 8
Sarno 8
Shenyang 8
West Jordan 8
Bogotá 7
Buffalo 7
Chandigarh 7
Fes 7
Totale 14.951
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.269
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.128
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 942
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 615
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 579
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 560
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 522
Target identification by structure-based computational approaches: Recent advances and perspectives 457
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 442
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 413
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 401
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 325
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 306
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 304
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 284
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 260
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 252
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 230
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 217
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 194
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 191
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 185
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 184
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 173
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 171
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 166
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 165
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 155
Anti-inflammatory trends of new benzimidazole derivatives 154
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 153
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 149
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 144
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 144
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 143
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 135
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 135
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 133
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 132
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 128
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 127
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 127
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 126
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 124
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 122
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 121
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 121
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 120
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 119
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 119
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 115
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 112
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 111
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 110
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 110
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 110
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 109
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 107
Discovery of noscapine derivatives as potential β-tubulin inhibitors 104
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 104
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 103
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 102
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 102
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 102
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 95
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 94
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 94
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 93
Reranking docking poses using molecular simulations and approximate free energy methods 90
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 90
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 89
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 89
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 87
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 86
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 85
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 84
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 82
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 82
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 82
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 81
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 79
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 78
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 76
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 75
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 70
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 69
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 66
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 58
Identification and Development of BRD9 Chemical Probes 52
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 46
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 45
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 44
The Role of LC-MS in Profiling Bioactive Compounds from Plant Waste for Cosmetic Applications: A General Overview 24
Identification of a New Interesting BAG3 Modulator Able to Disrupt Cancer-Related Pathways 16
New techniques of molecular modelling and structural chemistry for the development of bioactive compounds 14
Carnosol modulates mPGES-1/PPAR-γ biological axis: from in silico to in vivo clinical imaging and investigations 13
A 5-Br-1-Propylisatin Derivative as a Promising BRD9 Ligand: Insights from Computational and STD NMR Investigation 13
Unveiling New Triazoloquinoxaline‐Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9 11
Disruption of c-Myc/Max heterodimerization induced by a novel anticancer agent endowed with 1,3-diphenylurea moiety: an in silico, chemoproteomics-based, and in vitro combined approach 11
Potential Nutraceutical Properties of Vicia faba L: LC-ESI-HR-MS/MS-Based Profiling of Ancient Faba Bean Varieties and Their Biological Activity 11
Marine Natural Products in Preclinical Cancer Studies: Ten Years of Advanced Total Synthesis 10
Totale 18.651
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Categoria #
all - tutte 44.853
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 44.853
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/202152 0 0 0 0 0 0 0 0 0 0 0 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/202613.225 3.004 3.426 3.077 610 700 276 708 157 269 647 237 114
Totale 18.687