UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 11.440
NA - Nord America 5.946
EU - Europa 2.355
SA - Sud America 594
Continente sconosciuto - Info sul continente non disponibili 266
AF - Africa 108
OC - Oceania 3
Totale 20.712
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Nazione #
HK - Hong Kong 8.971
US - Stati Uniti d'America 5.704
IT - Italia 1.208
SG - Singapore 1.071
CN - Cina 458
BR - Brasile 452
VN - Vietnam 369
RU - Federazione Russa 254
DE - Germania 220
CA - Canada 128
UA - Ucraina 115
FR - Francia 99
IN - India 99
IE - Irlanda 85
TR - Turchia 83
GB - Regno Unito 79
BD - Bangladesh 77
KR - Corea 63
AR - Argentina 56
SE - Svezia 56
JP - Giappone 51
FI - Finlandia 48
MX - Messico 47
NL - Olanda 39
IQ - Iraq 35
ZA - Sudafrica 32
ID - Indonesia 30
AT - Austria 28
PL - Polonia 27
DZ - Algeria 26
ES - Italia 24
CO - Colombia 22
CZ - Repubblica Ceca 21
EC - Ecuador 21
PK - Pakistan 21
SA - Arabia Saudita 16
MA - Marocco 14
CL - Cile 13
CR - Costa Rica 13
IL - Israele 13
JM - Giamaica 12
PH - Filippine 12
UZ - Uzbekistan 12
CH - Svizzera 11
TT - Trinidad e Tobago 10
VE - Venezuela 10
HU - Ungheria 9
NI - Nicaragua 8
AZ - Azerbaigian 7
PY - Paraguay 7
GT - Guatemala 6
MY - Malesia 6
EG - Egitto 5
JO - Giordania 5
KE - Kenya 5
NP - Nepal 5
PE - Perù 5
UY - Uruguay 5
BE - Belgio 4
BH - Bahrain 4
KZ - Kazakistan 4
PT - Portogallo 4
RO - Romania 4
AL - Albania 3
DK - Danimarca 3
DO - Repubblica Dominicana 3
EU - Europa 3
LT - Lituania 3
OM - Oman 3
PR - Porto Rico 3
SC - Seychelles 3
SK - Slovacchia (Repubblica Slovacca) 3
TH - Thailandia 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
AU - Australia 2
BO - Bolivia 2
BS - Bahamas 2
ET - Etiopia 2
GA - Gabon 2
GE - Georgia 2
IR - Iran 2
LB - Libano 2
LU - Lussemburgo 2
NG - Nigeria 2
PS - Palestinian Territory 2
QA - Qatar 2
SN - Senegal 2
SY - Repubblica araba siriana 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AM - Armenia 1
BB - Barbados 1
BG - Bulgaria 1
BJ - Benin 1
BN - Brunei Darussalam 1
BQ - ???statistics.table.value.countryCode.BQ??? 1
BY - Bielorussia 1
BZ - Belize 1
CI - Costa d'Avorio 1
CU - Cuba 1
Totale 20.422
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Città #
Hong Kong 8.950
Dallas 700
San Jose 661
Singapore 578
Ann Arbor 558
Ashburn 416
Milan 347
Chandler 327
Council Bluffs 210
Princeton 199
Woodbridge 151
Wilmington 147
Jacksonville 145
Beijing 128
Ho Chi Minh City 119
Salerno 100
Los Angeles 98
Naples 95
Santa Clara 95
New York 91
The Dalles 91
Rome 89
Dublin 84
Munich 84
Lauterbourg 76
Houston 75
Hanoi 74
São Paulo 55
Izmir 53
Phoenix 50
Tokyo 48
Fisciano 46
Moscow 44
Memphis 43
Montreal 41
Dong Ket 38
Andover 33
Brooklyn 29
Frankfurt am Main 29
Chicago 28
Turku 28
Figino 27
Columbus 26
Dearborn 26
Denver 26
Nanjing 26
Pellezzano 26
Orem 25
Nuremberg 23
Boardman 22
Warsaw 22
Johannesburg 21
Seattle 21
Toronto 21
Washington 21
Atlanta 19
Chennai 19
Da Nang 19
Mexico City 19
Stockholm 18
London 16
Redwood City 16
Turin 16
Brno 15
Chengdu 15
Amsterdam 14
Boston 14
Haiphong 14
Baghdad 13
Belo Horizonte 13
Hải Dương 13
Afragola 12
Buffalo 12
Fairfield 12
Vienna 12
Jiaxing 11
Lucca 11
Montoro 11
Nanchang 11
Poplar 11
San Francisco 11
Seoul 11
Campinas 10
Curitiba 10
Istanbul 10
Jakarta 10
Mestre 10
New Delhi 10
Newark 10
Philadelphia 10
Pune 10
San Diego 10
Bologna 9
Charlotte 9
Düsseldorf 9
Kingston 9
Manchester 9
Ninh Bình 9
Nocera Superiore 9
Pagani 9
Totale 16.136
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.302
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.142
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 987
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 632
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 601
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 568
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 540
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 468
Target identification by structure-based computational approaches: Recent advances and perspectives 465
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 430
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 410
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 388
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 338
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 322
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 321
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 274
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 274
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 249
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 235
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 210
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 202
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 202
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 201
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 189
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 185
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 183
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 176
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 176
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 172
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 171
Anti-inflammatory trends of new benzimidazole derivatives 166
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 162
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 160
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 158
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 152
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 151
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 148
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 147
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 147
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 144
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 143
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 142
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 142
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 141
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 139
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 138
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 134
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 134
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 132
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 131
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 130
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 127
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 127
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 125
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 125
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 124
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 124
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 122
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 120
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 120
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 119
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 119
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 117
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 114
Discovery of noscapine derivatives as potential β-tubulin inhibitors 113
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 112
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 110
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 107
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 106
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 105
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 105
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 104
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 104
Reranking docking poses using molecular simulations and approximate free energy methods 103
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 102
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 100
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 99
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 97
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 94
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 93
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 93
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 90
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 87
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 87
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 85
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 81
Discovery of RUVBL1 as a Target of the Marine Alkaloid Caulerpin via MS-Based Functional Proteomics 76
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 71
Identification and Development of BRD9 Chemical Probes 69
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 67
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 62
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 54
The Role of LC-MS in Profiling Bioactive Compounds from Plant Waste for Cosmetic Applications: A General Overview 46
Disruption of c-Myc/Max heterodimerization induced by a novel anticancer agent endowed with 1,3-diphenylurea moiety: an in silico, chemoproteomics-based, and in vitro combined approach 42
A 5-Br-1-Propylisatin Derivative as a Promising BRD9 Ligand: Insights from Computational and STD NMR Investigation 36
Unveiling New Triazoloquinoxaline‐Based PROTACs Designed for the Selective Degradation of the ncBAF Chromatin Remodeling Subunit BRD9 35
Potential Nutraceutical Properties of Vicia faba L: LC-ESI-HR-MS/MS-Based Profiling of Ancient Faba Bean Varieties and Their Biological Activity 35
Identification of a New Interesting BAG3 Modulator Able to Disrupt Cancer-Related Pathways 34
Chemical Profiling of Polyphenolic Fraction of Cannabis sativa L. vr. Kompolti Industrial Inflorescences: Insights into Cannabidiol Neuroprotective Effects in a Cellular Model of Parkinson’s Disease 32
The future of BRD9 inhibitors: a patent perspective (2019-present) 30
Totale 20.503
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Categoria #
all - tutte 51.639
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 51.639
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022381 0 0 0 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/202613.710 3.004 3.426 3.077 610 700 276 708 157 269 647 237 599
2026/20271.540 329 181 437 593 0 0 0 0 0 0 0 0
Totale 20.712