UniSa - IRIS Institutional Research Information System

LAURO, Gianluigi
 Distribuzione geografica
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Continente #
AS - Asia 10.661
NA - Nord America 3.629
EU - Europa 1.467
SA - Sud America 474
AF - Africa 69
Continente sconosciuto - Info sul continente non disponibili 4
OC - Oceania 2
Totale 16.306
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Nazione #
HK - Hong Kong 8.900
US - Stati Uniti d'America 3.527
SG - Singapore 840
IT - Italia 525
BR - Brasile 391
CN - Cina 359
RU - Federazione Russa 244
VN - Vietnam 226
DE - Germania 189
UA - Ucraina 109
IE - Irlanda 81
TR - Turchia 68
IN - India 66
GB - Regno Unito 58
KR - Corea 56
CA - Canada 53
SE - Svezia 52
FI - Finlandia 46
AR - Argentina 38
JP - Giappone 38
MX - Messico 36
NL - Olanda 31
AT - Austria 27
ZA - Sudafrica 25
ID - Indonesia 23
PL - Polonia 22
DZ - Algeria 20
ES - Italia 20
BD - Bangladesh 18
CZ - Repubblica Ceca 17
FR - Francia 16
IQ - Iraq 16
PK - Pakistan 14
CO - Colombia 12
EC - Ecuador 11
MA - Marocco 8
PY - Paraguay 7
CH - Svizzera 6
CL - Cile 5
UZ - Uzbekistan 5
BE - Belgio 4
RO - Romania 4
SA - Arabia Saudita 4
VE - Venezuela 4
AZ - Azerbaigian 3
DK - Danimarca 3
EG - Egitto 3
EU - Europa 3
GT - Guatemala 3
HU - Ungheria 3
IL - Israele 3
PE - Perù 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
AL - Albania 2
BH - Bahrain 2
DO - Repubblica Dominicana 2
GA - Gabon 2
GE - Georgia 2
JM - Giamaica 2
JO - Giordania 2
KE - Kenya 2
KZ - Kazakistan 2
LT - Lituania 2
LU - Lussemburgo 2
NG - Nigeria 2
NI - Nicaragua 2
NP - Nepal 2
UY - Uruguay 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AM - Armenia 1
AU - Australia 1
BG - Bulgaria 1
CU - Cuba 1
CY - Cipro 1
GN - Guinea 1
GY - Guiana 1
KI - Kiribati 1
LB - Libano 1
LC - Santa Lucia 1
LK - Sri Lanka 1
MC - Monaco 1
ML - Mali 1
MN - Mongolia 1
OM - Oman 1
PA - Panama 1
PT - Portogallo 1
QA - Qatar 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
SY - Repubblica araba siriana 1
TH - Thailandia 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
ZM - Zambia 1
Totale 16.306
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Città #
Hong Kong 8.887
Dallas 689
Ann Arbor 558
Singapore 415
Chandler 326
Ashburn 233
Princeton 198
Woodbridge 151
Wilmington 145
Jacksonville 142
Salerno 90
Munich 84
Dublin 80
Beijing 76
Los Angeles 70
Houston 69
Ho Chi Minh City 67
Naples 66
Izmir 52
Hanoi 43
Moscow 43
Fisciano 42
New York 41
São Paulo 39
Dong Ket 38
The Dalles 38
Tokyo 35
Andover 33
Montreal 32
Turku 28
Dearborn 26
Nanjing 26
Pellezzano 26
Columbus 23
Nuremberg 22
Brooklyn 21
Johannesburg 21
Boardman 20
Denver 19
Santa Clara 19
Warsaw 18
Chennai 17
Orem 16
Redwood City 16
Seattle 16
Brno 15
Chengdu 14
Phoenix 14
Stockholm 14
Mexico City 13
Afragola 12
Belo Horizonte 12
Boston 12
London 12
Vienna 12
Washington 12
Amsterdam 11
Fairfield 11
Frankfurt am Main 11
Jiaxing 11
Nanchang 11
Seoul 11
Curitiba 10
Lucca 10
Mestre 10
Milan 10
Poplar 10
Atlanta 9
Campinas 9
Chicago 9
Council Bluffs 9
Düsseldorf 9
Hải Dương 9
Pune 9
Da Nang 8
El Hadjira 8
Jakarta 8
Manchester 8
Rome 8
San Jose 8
Sarno 8
Shanghai 8
Shenyang 8
West Jordan 8
Haiphong 7
Hebei 7
Jinan 7
Napoli 7
New Delhi 7
Ninh Bình 7
Tianjin 7
Chandigarh 6
Fes 6
Mumbai 6
Norwalk 6
Ortona 6
Redondo Beach 6
San Francisco 6
Toronto 6
Uster 6
Totale 13.620
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Nome #
Predicting PROTAC-mediated ternary complex structures through in silico approaches 2.201
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 1.104
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 921
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 584
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 562
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 542
In Silico Design, Chemical Synthesis, Biophysical and in Vitro Evaluation for the Identification of 1-Ethyl-1H-Pyrazolo[3,4-b]Pyridine-Based BRD9 Binders 505
Target identification by structure-based computational approaches: Recent advances and perspectives 447
Phytochemical investigation of Cannabis sativa: Isolation and structure determination of spiroindans 418
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 391
Identification of Novel Bromodomain-Containing Protein 4 (BRD4) Binders through 3D Pharmacophore-Based Repositioning Screening Campaign 375
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 305
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 286
PharmaCore: The Automatic Generation of 3D Structure-Based Pharmacophore Models from Protein/Ligand Complexes 275
Investigation analysis of the phytochemical composition of Laurus nobilis L. leaves essential oil: a study of the antioxidant and anti-inflammatory properties using a combination of in vitro and in silico methods 244
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 230
Essential Oils of Laurus nobilis L.: From Chemical Analysis to In Silico Investigation of Anti-Inflammatory Activity by Soluble Epoxide Hydrolase (sEH) Inhibition 228
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 205
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 190
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 177
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 168
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 166
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 156
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 154
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 151
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 147
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 144
Anti-inflammatory trends of new benzimidazole derivatives 131
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 130
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 128
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 121
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 117
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 114
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 113
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 113
Virtual screening of 3-(1H-1,2,3-triazol-1-yl)piperidine-2,6-dione-based compounds as new potential Cereblon modulators amenable for targeted protein degradation 112
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 112
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 109
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 108
Dihydroaurones and Isoflavan Derivatives from the Roots of Glycyrrhiza asymmetrica 107
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 107
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 105
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 103
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 100
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 99
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 99
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 98
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 97
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 95
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 94
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 94
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 94
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 92
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 90
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 89
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization 86
Discovery of noscapine derivatives as potential β-tubulin inhibitors 86
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 85
Identification of the first-in-class dual inhibitor targeting BAG3 and HSP70 proteins to disrupt multiple chaperone pathways 81
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 81
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 80
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 78
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 77
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 76
Reranking docking poses using molecular simulations and approximate free energy methods 75
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 73
5-methyl-2-carboxamidepyrrole-based novel dual mPGES-1/sEH inhibitors as promising anticancer candidates 72
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 72
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 70
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 70
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 69
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 69
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 68
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 67
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition 65
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 65
Unveiling the Potential Biological and Chemical Mechanism of Pergularia tomentosa Extracts by Liquid Chromatography‐Electrospray Ionisation‐High‐Resolution Tandem Mass Spectrometry, In‐Vitro and In‐Vivo Pharmacological Studies 65
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 63
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 63
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 59
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution 58
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 58
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 55
Chemical Profiling of Polar Lipids and the Polyphenolic Fraction of Commercial Italian Phaseolus Seeds by UHPLC-HRMS and Biological Evaluation 51
Identification of a New Promising BAG3 Modulator Featuring the Imidazopyridine Scaffold 50
Repositioning of Small Molecules through the Inverse Virtual Screening in silico Tool: Case of Benzothiazole-Based Inhibitors of Soluble Epoxide Hydrolase (sEH) 49
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 32
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 32
A Classic Photochemical Approach Inducing an Unexpected Rearrangement: Exploring the Photoreactivity of Pentacyclic Triterpenic Acids 31
Identification and Development of BRD9 Chemical Probes 31
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 28
New techniques of molecular modelling and structural chemistry for the development of bioactive compounds 2
Totale 16.539
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Categoria #
all - tutte 39.892
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 39.892
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021255 0 0 0 0 0 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/20252.207 58 14 11 71 47 115 388 115 248 73 180 887
2025/202611.077 3.004 3.426 3.077 610 700 260 0 0 0 0 0 0
Totale 16.539