LAURO, Gianluigi
 Distribuzione geografica
Continente #
NA - Nord America 2.168
EU - Europa 694
AS - Asia 330
Continente sconosciuto - Info sul continente non disponibili 4
SA - Sud America 4
OC - Oceania 1
Totale 3.201
Nazione #
US - Stati Uniti d'America 2.156
IT - Italia 310
CN - Cina 147
UA - Ucraina 98
DE - Germania 82
IE - Irlanda 79
SG - Singapore 68
TR - Turchia 56
VN - Vietnam 38
SE - Svezia 37
FI - Finlandia 17
CZ - Repubblica Ceca 15
IN - India 14
FR - Francia 10
GB - Regno Unito 9
RU - Federazione Russa 9
CA - Canada 8
CH - Svizzera 6
ES - Italia 6
MX - Messico 4
NL - Olanda 4
BR - Brasile 3
EU - Europa 3
JP - Giappone 2
KR - Corea 2
LU - Lussemburgo 2
PL - Polonia 2
SA - Arabia Saudita 2
A2 - ???statistics.table.value.countryCode.A2??? 1
AE - Emirati Arabi Uniti 1
AR - Argentina 1
AT - Austria 1
AU - Australia 1
BE - Belgio 1
BG - Bulgaria 1
DK - Danimarca 1
HU - Ungheria 1
MC - Monaco 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
Totale 3.201
Città #
Ann Arbor 558
Chandler 326
Princeton 198
Woodbridge 151
Wilmington 145
Jacksonville 142
Ashburn 110
Salerno 84
Dublin 79
Houston 61
Izmir 52
Singapore 40
Dong Ket 38
Andover 33
Beijing 32
Dearborn 26
Nanjing 26
Pellezzano 26
Fisciano 22
Naples 19
Boardman 18
Redwood City 16
Brno 13
Los Angeles 12
Munich 12
Fairfield 11
Jiaxing 11
Nanchang 11
Washington 11
Dallas 10
Mestre 10
Düsseldorf 9
Pune 9
Shenyang 8
Hebei 7
Napoli 7
Seattle 7
Jinan 6
Norwalk 6
Ortona 6
Uster 6
Cava de' Tirreni 5
Chicago 5
Guangzhou 5
Nocera Superiore 5
Pozzuoli 5
San Diego 5
Shanghai 5
Tianjin 5
Dormagen 4
Montreal 4
Pignola 4
Amsterdam 3
Buonabitacolo 3
Cambridge 3
Cardito 3
Changsha 3
Granada 3
New York 3
Nürnberg 3
Ravenna 3
Spinea 3
Torre Annunziata 3
Altavilla Silentina 2
Antalya 2
Assago 2
Bari 2
Cadoneghe 2
Darmstadt 2
Delhi 2
Donostia / San Sebastian 2
Dundee 2
Edinburgh 2
Indiana 2
Lappeenranta 2
Lodz 2
Lucknow 2
Luxembourg 2
Morciano di Leuca 2
Nola 2
Rome 2
Sarno 2
Springfield 2
Stockholm 2
Taizhou 2
Tappahannock 2
Tokyo 2
Toronto 2
Zhengzhou 2
Acerra 1
Afragola 1
Benevento 1
Bratislava 1
Brooklyn 1
Brussels 1
Budapest 1
Buenos Aires 1
Buffalo 1
Cabras 1
Caianello 1
Totale 2.522
Nome #
9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain 137
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ 125
Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase 107
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor 101
Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" 100
Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening 100
Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride 98
Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) 89
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist 88
Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum 87
Anti-inflammatory trends of new benzimidazole derivatives 87
Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors 85
Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs 85
Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells 82
Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines 78
New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei 78
Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme 78
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds 76
Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization 70
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 69
Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge 68
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds 67
Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities 66
Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp 63
Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp 62
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics 59
Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs 58
A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors 52
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies 49
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach 42
Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) 42
Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists 40
Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds 40
DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data 39
Discovery of noscapine derivatives as potential β-tubulin inhibitors 39
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein 39
Reranking docking poses using molecular simulations and approximate free energy methods 37
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities 37
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells 36
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol 34
Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells 34
Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches 33
The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane 33
Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches 30
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway 30
Biological Profile of Two Gentiana lutea L. Metabolites Using Computational Approaches and In Vitro Tests 29
Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins 27
Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods 25
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders 25
Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities 24
Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) 22
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders 21
Target identification by structure-based computational approaches: Recent advances and perspectives 19
Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach 19
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation 18
Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods 18
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches 17
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis 17
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation 16
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition 13
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models 13
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines 12
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization 11
A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors 8
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies 7
Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A 7
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors 5
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor 3
Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches 2
NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity 2
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 2
Totale 3.331
Categoria #
all - tutte 13.239
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 13.239


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020230 0 0 33 7 22 11 26 7 21 33 56 14
2020/2021334 8 22 22 0 27 14 54 10 76 9 40 52
2021/2022393 3 1 8 20 24 6 6 19 58 43 49 156
2022/2023740 58 77 19 115 76 142 12 72 95 5 43 26
2023/2024385 17 40 31 21 43 90 24 24 13 21 11 50
2024/202576 58 14 4 0 0 0 0 0 0 0 0 0
Totale 3.331