UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
NA - Nord America 9.189
AS - Asia 8.148
EU - Europa 2.841
SA - Sud America 698
Continente sconosciuto - Info sul continente non disponibili 309
AF - Africa 107
OC - Oceania 3
Totale 21.295
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Nazione #
US - Stati Uniti d'America 8.941
HK - Hong Kong 4.881
SG - Singapore 1.392
IT - Italia 1.161
CN - Cina 696
BR - Brasile 537
VN - Vietnam 462
RU - Federazione Russa 345
UA - Ucraina 321
DE - Germania 228
TR - Turchia 190
FR - Francia 144
IE - Irlanda 138
CA - Canada 120
IN - India 109
FI - Finlandia 105
KR - Corea 104
SE - Svezia 104
GB - Regno Unito 101
BD - Bangladesh 69
AR - Argentina 57
MX - Messico 49
JP - Giappone 42
PL - Polonia 39
IL - Israele 32
IQ - Iraq 32
ES - Italia 29
NL - Olanda 27
PK - Pakistan 27
ZA - Sudafrica 27
ID - Indonesia 26
CO - Colombia 21
EC - Ecuador 21
AT - Austria 18
CZ - Repubblica Ceca 18
VE - Venezuela 18
JM - Giamaica 17
UZ - Uzbekistan 15
MA - Marocco 14
CL - Cile 13
PE - Perù 13
HN - Honduras 12
PH - Filippine 12
DZ - Algeria 11
PY - Paraguay 10
TT - Trinidad e Tobago 10
GR - Grecia 9
SA - Arabia Saudita 9
SC - Seychelles 9
GT - Guatemala 8
MY - Malesia 8
TN - Tunisia 8
AE - Emirati Arabi Uniti 7
AL - Albania 6
BO - Bolivia 6
CR - Costa Rica 6
EG - Egitto 6
ET - Etiopia 6
EU - Europa 6
JO - Giordania 6
KE - Kenya 6
RO - Romania 6
AZ - Azerbaigian 5
HU - Ungheria 5
NI - Nicaragua 5
PA - Panama 5
BE - Belgio 4
BG - Bulgaria 4
CH - Svizzera 4
EE - Estonia 4
LB - Libano 4
LY - Libia 4
BB - Barbados 3
DO - Repubblica Dominicana 3
HR - Croazia 3
IR - Iran 3
LT - Lituania 3
NO - Norvegia 3
PR - Porto Rico 3
SV - El Salvador 3
CG - Congo 2
CW - ???statistics.table.value.countryCode.CW??? 2
KZ - Kazakistan 2
LU - Lussemburgo 2
NG - Nigeria 2
NP - Nepal 2
NZ - Nuova Zelanda 2
OM - Oman 2
PS - Palestinian Territory 2
PT - Portogallo 2
RS - Serbia 2
UY - Uruguay 2
AM - Armenia 1
AO - Angola 1
AU - Australia 1
AW - Aruba 1
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CI - Costa d'Avorio 1
Totale 20.970
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Città #
Hong Kong 4.866
Ann Arbor 1.456
Ashburn 833
San Jose 800
Singapore 718
Chandler 528
Woodbridge 505
Houston 431
Jacksonville 422
Princeton 384
Milan 375
Dallas 346
Wilmington 313
Council Bluffs 244
Beijing 213
Salerno 181
Dong Ket 177
Izmir 160
Dublin 130
The Dalles 121
New York 108
Ho Chi Minh City 105
Rome 102
Lauterbourg 95
Santa Clara 95
São Paulo 94
Munich 87
Nanjing 82
Boardman 79
Andover 78
Los Angeles 76
Hanoi 62
Moscow 53
Pellezzano 51
Dearborn 41
Fairfield 40
Columbus 39
Tokyo 37
Brooklyn 36
Chicago 36
Figino 36
Phoenix 36
Hebei 34
Toronto 34
Warsaw 34
Denver 29
Montreal 29
Shenyang 26
Turku 26
Naples 25
Orem 25
Philadelphia 23
Atlanta 22
Pune 22
Fisciano 21
Memphis 21
Mestre 21
Nanchang 20
Seattle 20
Basingstoke 19
Frankfurt am Main 19
San Francisco 18
Turin 18
Mexico City 17
Rio de Janeiro 17
Boston 16
Changsha 16
Jiaxing 16
Johannesburg 16
Norwalk 16
Seoul 16
Helsinki 15
Nuremberg 15
Redwood City 15
Tashkent 15
Washington 15
Amsterdam 14
Chennai 14
Guangzhou 14
Jakarta 14
Buffalo 13
Düsseldorf 13
Falls Church 13
North Bergen 13
Shanghai 13
Stockholm 13
Baghdad 12
Belo Horizonte 12
Haiphong 12
London 12
Tianjin 12
Brno 11
Charlotte 11
Da Nang 11
Hải Dương 11
Poplar 11
Ankara 10
Miami 10
San Diego 10
Baronissi 9
Totale 15.670
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.289
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 699
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 545
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 513
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 451
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 392
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 384
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 341
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 283
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 282
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 281
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 277
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 269
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 257
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 244
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 238
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 228
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 226
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 215
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 213
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 207
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 204
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 203
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 202
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 197
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 197
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 193
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 188
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 185
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 184
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 184
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 183
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 180
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 175
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 175
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 172
Microbiologia Molecolare e Cellulare 172
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 172
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 171
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 170
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 169
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 167
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 165
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 165
Chemical biology of Histone acetyltransferase natural compounds modulators. 159
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 159
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 158
Azole antifungal agents related to naftifine and butenafine 156
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 154
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 154
Discovery of new chemical probes for the MRG15 chromo domain. 153
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 152
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 148
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 146
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 144
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 144
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 144
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 143
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 143
Antimycobacterial activity of ionic fullerene derivatives. 141
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 141
Exploiting acylaminopyrazole scaffold for polypharmacology approach in Alzheimer's disease 140
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 140
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 140
The emerging role of lysine methyltransferase SETD8 in human diseases 138
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 137
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 137
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 137
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 136
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 136
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 135
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 135
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 135
N-Pyrrylarylsulfones with High Therapeutic Potential 134
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 134
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 134
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 132
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 131
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 131
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 131
Synthesis and pharmacological characterization of new analogs of broxaterol. 130
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 129
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 129
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 126
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 125
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 124
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 124
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 122
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 122
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 120
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 118
Lysine methyltransferase inhibitors: where we are now. 118
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 116
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 114
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 114
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 113
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 112
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 110
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 110
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 109
Totale 19.504
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Categoria #
all - tutte 62.084
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 62.084
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022715 0 0 0 0 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/202610.024 1.139 2.239 2.228 439 719 324 895 234 406 562 159 680
2026/20272.149 242 208 615 1.003 81 0 0 0 0 0 0 0
Totale 21.295