UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
NA - Nord America 5.065
EU - Europa 1.206
AS - Asia 713
SA - Sud America 13
Continente sconosciuto - Info sul continente non disponibili 6
AF - Africa 4
OC - Oceania 1
Totale 7.008
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Nazione #
US - Stati Uniti d'America 5.056
IT - Italia 419
CN - Cina 337
UA - Ucraina 304
VN - Vietnam 178
TR - Turchia 161
IE - Irlanda 135
DE - Germania 100
SE - Svezia 94
FI - Finlandia 61
FR - Francia 38
IN - India 19
GB - Regno Unito 15
RU - Federazione Russa 9
AR - Argentina 6
EU - Europa 6
HU - Ungheria 5
KR - Corea 5
PE - Perù 5
AT - Austria 3
BG - Bulgaria 3
CA - Canada 3
IL - Israele 3
NL - Olanda 3
PA - Panama 3
RO - Romania 3
BE - Belgio 2
CL - Cile 2
GR - Grecia 2
HR - Croazia 2
JP - Giappone 2
NO - Norvegia 2
PL - Polonia 2
SA - Arabia Saudita 2
BZ - Belize 1
CH - Svizzera 1
CM - Camerun 1
EG - Egitto 1
ES - Italia 1
GH - Ghana 1
ID - Indonesia 1
IR - Iran 1
KH - Cambogia 1
LU - Lussemburgo 1
MX - Messico 1
NZ - Nuova Zelanda 1
PH - Filippine 1
PK - Pakistan 1
RS - Serbia 1
SC - Seychelles 1
SG - Singapore 1
TT - Trinidad e Tobago 1
Totale 7.008
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Città #
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Jacksonville 420
Houston 417
Princeton 384
Wilmington 310
Dong Ket 177
Salerno 167
Izmir 160
Dublin 128
Ashburn 124
Beijing 101
Nanjing 82
Andover 78
Boardman 78
Pellezzano 51
Dearborn 41
Fairfield 40
Hebei 34
Shenyang 25
Mestre 21
Nanchang 20
Philadelphia 17
Norwalk 16
Pune 16
Changsha 15
Jiaxing 15
Redwood City 15
Rome 15
Düsseldorf 13
Falls Church 13
Tianjin 12
Washington 12
Fisciano 10
Seattle 10
Cambridge 9
Jinan 7
Los Angeles 7
Napoli 7
San Diego 7
Guangzhou 6
Indiana 6
Munro 6
Renton 6
Tappahannock 6
Florence 5
New York 5
Palermo 5
Sorrento 5
Spinea 5
Edinburgh 4
Menlo Park 4
Naples 4
Stockholm 4
Cagliari 3
Casoria 3
Catania 3
Hefei 3
Marcianise 3
Messina 3
Mugnano del Cardinale 3
Munich 3
Orange 3
Panama City 3
Scafati 3
Vienna 3
Athens 2
Atlanta 2
Brussels 2
Caivano 2
Calvisano 2
Chicago 2
Contrada 2
Durham 2
Hangzhou 2
Hanover 2
Krimpen Aan Den Ijssel 2
London 2
Maddaloni 2
Mercato San Severino 2
Montreal 2
Mumbai 2
Nocera Superiore 2
Nürnberg 2
Oslo 2
Pescara 2
Seoul 2
Trumbull 2
Warsaw 2
Yekaterinburg 2
Zagreb 2
Alexandria 1
Arcevia 1
Auckland 1
Bari 1
Belgrade 1
Belize City 1
Benevento 1
Birkenhead 1
Totale 5.725
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Nome #
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 149
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 144
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 121
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 117
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 116
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 115
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 114
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 110
Microbiologia Molecolare e Cellulare 109
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 105
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 105
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 102
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 101
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 100
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 96
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 95
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 94
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 93
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 92
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 91
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 91
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 90
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 90
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 89
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 89
Azole antifungal agents related to naftifine and butenafine 88
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 87
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 86
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 85
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 84
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 83
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 82
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 82
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 81
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 81
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 81
Chemical biology of Histone acetyltransferase natural compounds modulators. 80
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 80
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 79
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 77
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 75
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 75
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 74
Antimycobacterial activity of ionic fullerene derivatives. 71
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 71
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 71
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 70
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 69
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 69
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 69
N-Pyrrylarylsulfones with High Therapeutic Potential 69
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 68
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 68
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 67
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 65
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 64
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 63
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 62
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 62
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 61
Enhancement of lysine acetylation accelerates wound repair 60
The emerging role of lysine methyltransferase SETD8 in human diseases 60
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 60
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 60
Synthesis of tricyclic triazepinones related to nevirapine. 59
Synthesis and pharmacological characterization of new analogs of broxaterol. 58
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 57
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 57
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 57
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 57
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 56
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 56
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 55
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 55
Design and Synthesis of Novel [60]Fullerene Derivatives as Potential HIV Aspartic Protease Inhibitors. 54
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 54
Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives. 53
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 53
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 52
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 51
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 50
Lysine methyltransferase inhibitors: where we are now. 50
Discovery of new chemical probes for the MRG15 chromo domain. 47
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 46
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 46
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 45
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 45
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 44
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 41
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 38
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 38
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 37
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 35
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 33
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 33
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 33
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 32
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 30
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 25
Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment 24
Totale 7.113
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Categoria #
all - tutte 19.802
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 19.802
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019283 0 0 0 0 0 0 0 0 0 0 268 15
2019/2020757 215 13 75 10 60 21 72 12 71 61 142 5
2020/2021785 5 71 88 4 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024392 41 67 38 14 39 94 28 40 5 23 3 0
Totale 7.273