UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 8.091
NA - Nord America 7.538
EU - Europa 2.708
SA - Sud America 644
Continente sconosciuto - Info sul continente non disponibili 306
AF - Africa 98
OC - Oceania 3
Totale 19.388
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Nazione #
US - Stati Uniti d'America 7.384
HK - Hong Kong 4.878
SG - Singapore 1.389
IT - Italia 1.098
CN - Cina 684
BR - Brasile 485
VN - Vietnam 462
UA - Ucraina 321
RU - Federazione Russa 309
DE - Germania 225
TR - Turchia 189
FR - Francia 143
IE - Irlanda 137
IN - India 107
FI - Finlandia 105
KR - Corea 104
SE - Svezia 103
GB - Regno Unito 89
BD - Bangladesh 65
CA - Canada 59
AR - Argentina 57
MX - Messico 49
JP - Giappone 36
PL - Polonia 36
IQ - Iraq 32
PK - Pakistan 27
ID - Indonesia 26
ZA - Sudafrica 26
ES - Italia 24
NL - Olanda 23
CO - Colombia 21
EC - Ecuador 21
AT - Austria 18
CZ - Repubblica Ceca 18
VE - Venezuela 16
UZ - Uzbekistan 15
MA - Marocco 14
CL - Cile 13
PE - Perù 13
DZ - Algeria 11
PH - Filippine 11
IL - Israele 10
PY - Paraguay 10
GR - Grecia 9
JM - Giamaica 9
MY - Malesia 8
TN - Tunisia 8
AE - Emirati Arabi Uniti 7
SA - Arabia Saudita 7
TT - Trinidad e Tobago 7
AL - Albania 6
BO - Bolivia 6
EG - Egitto 6
ET - Etiopia 6
EU - Europa 6
JO - Giordania 6
KE - Kenya 6
RO - Romania 6
AZ - Azerbaigian 5
HN - Honduras 5
HU - Ungheria 5
PA - Panama 5
BG - Bulgaria 4
CH - Svizzera 4
CR - Costa Rica 4
LY - Libia 4
BE - Belgio 3
DO - Repubblica Dominicana 3
GT - Guatemala 3
HR - Croazia 3
IR - Iran 3
LB - Libano 3
LT - Lituania 3
NO - Norvegia 3
BB - Barbados 2
CG - Congo 2
KZ - Kazakistan 2
LU - Lussemburgo 2
NG - Nigeria 2
NI - Nicaragua 2
NP - Nepal 2
NZ - Nuova Zelanda 2
OM - Oman 2
PR - Porto Rico 2
PS - Palestinian Territory 2
PT - Portogallo 2
RS - Serbia 2
SV - El Salvador 2
UY - Uruguay 2
AM - Armenia 1
AO - Angola 1
AU - Australia 1
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CI - Costa d'Avorio 1
CM - Camerun 1
CW - ???statistics.table.value.countryCode.CW??? 1
CY - Cipro 1
DK - Danimarca 1
Totale 19.067
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Città #
Hong Kong 4.864
Ann Arbor 1.456
Singapore 716
San Jose 581
Chandler 527
Woodbridge 503
Houston 427
Jacksonville 421
Princeton 384
Ashburn 379
Milan 365
Dallas 333
Wilmington 311
Beijing 206
Salerno 181
Dong Ket 177
Izmir 160
Council Bluffs 132
Dublin 130
The Dalles 119
Ho Chi Minh City 105
Rome 96
Lauterbourg 95
Munich 87
Nanjing 82
Boardman 79
Andover 78
Santa Clara 75
Los Angeles 70
Hanoi 62
New York 56
Moscow 53
Pellezzano 51
São Paulo 44
Dearborn 41
Fairfield 40
Columbus 36
Hebei 34
Tokyo 33
Warsaw 33
Figino 32
Shenyang 26
Turku 26
Brooklyn 25
Naples 23
Chicago 22
Montreal 22
Orem 22
Pune 22
Fisciano 21
Mestre 21
Atlanta 20
Denver 20
Nanchang 20
Philadelphia 20
Basingstoke 19
Frankfurt am Main 19
Memphis 17
Mexico City 17
Rio de Janeiro 17
Boston 16
Changsha 16
Jiaxing 16
Norwalk 16
Seattle 16
Seoul 16
Helsinki 15
Johannesburg 15
Nuremberg 15
Redwood City 15
Tashkent 15
Turin 15
Chennai 14
Guangzhou 14
Jakarta 14
San Francisco 14
Washington 14
Amsterdam 13
Düsseldorf 13
Falls Church 13
Phoenix 13
Shanghai 13
Baghdad 12
Belo Horizonte 12
Haiphong 12
London 12
Stockholm 12
Tianjin 12
Brno 11
Da Nang 11
Hải Dương 11
Poplar 11
Ankara 10
Baronissi 9
Buffalo 9
Cambridge 9
Campinas 9
Florence 9
Lahore 9
Scafati 9
Totale 14.563
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.248
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 688
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 532
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 466
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 443
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 383
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 379
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 302
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 270
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 260
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 258
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 250
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 249
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 242
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 238
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 228
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 218
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 203
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 199
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 197
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 193
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 187
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 183
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 178
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 173
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 171
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 171
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 168
Microbiologia Molecolare e Cellulare 167
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 167
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 166
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 163
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 161
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 158
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 157
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 156
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 155
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 154
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 154
Chemical biology of Histone acetyltransferase natural compounds modulators. 152
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 149
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 149
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 149
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 148
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 146
Azole antifungal agents related to naftifine and butenafine 145
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 143
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 143
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 137
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 137
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 136
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 135
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 133
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 132
Antimycobacterial activity of ionic fullerene derivatives. 132
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 132
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 130
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 128
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 127
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 127
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 126
The emerging role of lysine methyltransferase SETD8 in human diseases 126
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 126
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 126
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 125
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 125
N-Pyrrylarylsulfones with High Therapeutic Potential 125
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 125
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 124
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 124
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 123
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 123
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 122
Exploiting acylaminopyrazole scaffold for polypharmacology approach in Alzheimer's disease 121
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 121
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 120
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 120
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 118
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 118
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 117
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 115
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 114
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 113
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 112
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 110
Lysine methyltransferase inhibitors: where we are now. 110
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 109
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 108
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 106
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 106
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 104
Discovery of new chemical probes for the MRG15 chromo domain. 102
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 102
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 101
Enhancement of lysine acetylation accelerates wound repair 100
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 99
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 99
Synthesis and pharmacological characterization of new analogs of broxaterol. 98
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 97
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 97
Totale 17.902
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Categoria #
all - tutte 56.269
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 56.269
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/202610.024 1.139 2.239 2.228 439 719 324 895 234 406 562 159 680
2026/2027242 242 0 0 0 0 0 0 0 0 0 0 0
Totale 19.388