UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 7.020
NA - Nord America 6.129
EU - Europa 1.865
SA - Sud America 484
AF - Africa 53
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 2
Totale 15.559
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Nazione #
US - Stati Uniti d'America 6.050
HK - Hong Kong 4.742
SG - Singapore 999
CN - Cina 569
IT - Italia 487
BR - Brasile 407
UA - Ucraina 311
RU - Federazione Russa 302
VN - Vietnam 280
DE - Germania 200
TR - Turchia 176
IE - Irlanda 135
SE - Svezia 102
FI - Finlandia 97
KR - Corea 88
GB - Regno Unito 59
IN - India 51
FR - Francia 42
CA - Canada 34
AR - Argentina 32
MX - Messico 31
PL - Polonia 28
JP - Giappone 23
ES - Italia 19
ID - Indonesia 17
AT - Austria 16
CZ - Repubblica Ceca 16
BD - Bangladesh 14
ZA - Sudafrica 14
NL - Olanda 13
IQ - Iraq 12
PK - Pakistan 12
EC - Ecuador 11
PE - Perù 11
CO - Colombia 9
MA - Marocco 8
UZ - Uzbekistan 8
EU - Europa 6
GR - Grecia 6
DZ - Algeria 5
HU - Ungheria 5
PY - Paraguay 5
RO - Romania 5
CL - Cile 4
EG - Egitto 4
IL - Israele 4
SA - Arabia Saudita 4
TN - Tunisia 4
VE - Venezuela 4
AE - Emirati Arabi Uniti 3
BG - Bulgaria 3
JO - Giordania 3
KE - Kenya 3
PA - Panama 3
TT - Trinidad e Tobago 3
AL - Albania 2
AZ - Azerbaigian 2
BE - Belgio 2
CG - Congo 2
CH - Svizzera 2
DO - Repubblica Dominicana 2
HR - Croazia 2
IR - Iran 2
KZ - Kazakistan 2
LB - Libano 2
LT - Lituania 2
LY - Libia 2
NO - Norvegia 2
NZ - Nuova Zelanda 2
PS - Palestinian Territory 2
RS - Serbia 2
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CM - Camerun 1
CR - Costa Rica 1
DM - Dominica 1
EE - Estonia 1
ET - Etiopia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
IS - Islanda 1
JM - Giamaica 1
KH - Cambogia 1
KW - Kuwait 1
LU - Lussemburgo 1
MW - Malawi 1
MY - Malesia 1
MZ - Mozambico 1
NA - Namibia 1
NG - Nigeria 1
NI - Nicaragua 1
NP - Nepal 1
PH - Filippine 1
PT - Portogallo 1
SC - Seychelles 1
SN - Senegal 1
UY - Uruguay 1
Totale 15.559
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Città #
Hong Kong 4.734
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Houston 425
Jacksonville 421
Singapore 417
Princeton 384
Dallas 325
Wilmington 311
Ashburn 248
Dong Ket 177
Salerno 167
Beijing 165
Izmir 160
Dublin 128
Munich 87
Nanjing 82
Boardman 79
Andover 78
Los Angeles 55
Moscow 52
Pellezzano 51
New York 42
Dearborn 41
Fairfield 40
Ho Chi Minh City 39
São Paulo 39
The Dalles 36
Columbus 34
Hebei 34
Santa Clara 27
Turku 26
Warsaw 26
Shenyang 25
Mestre 21
Tokyo 21
Nanchang 20
Pune 20
Rome 20
Council Bluffs 18
Montreal 18
Philadelphia 17
Changsha 16
Chicago 16
Denver 16
Fisciano 16
Hanoi 16
Norwalk 16
Seoul 16
Brooklyn 15
Jiaxing 15
Redwood City 15
Atlanta 14
Boston 14
Guangzhou 14
Seattle 14
Düsseldorf 13
Falls Church 13
Washington 13
Nuremberg 12
San Francisco 12
Tianjin 12
Brno 11
Chennai 11
Mexico City 11
Poplar 11
Rio de Janeiro 11
Stockholm 11
Belo Horizonte 10
Jakarta 10
Johannesburg 10
London 10
Phoenix 10
Shanghai 10
Ankara 9
Cambridge 9
Scafati 9
Campinas 8
Orem 8
Tashkent 8
Helsinki 7
Jinan 7
Manchester 7
Napoli 7
San Diego 7
Santo André 7
Vienna 7
Amsterdam 6
Baronissi 6
Guarulhos 6
Indiana 6
Joinville 6
Munro 6
Naples 6
Renton 6
Tappahannock 6
Da Nang 5
Florence 5
Oklahoma City 5
Totale 12.179
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.207
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 665
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 493
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 436
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 413
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 367
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 353
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 270
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 242
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 239
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 226
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 218
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 211
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 209
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 195
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 187
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 178
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 168
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 167
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 160
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 151
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 149
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 145
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 144
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 141
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 139
Microbiologia Molecolare e Cellulare 138
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 138
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 138
Chemical biology of Histone acetyltransferase natural compounds modulators. 133
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 133
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 132
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 131
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 130
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 128
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 127
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 126
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 126
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 123
Azole antifungal agents related to naftifine and butenafine 117
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 116
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 116
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 115
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 114
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 114
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 111
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 110
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 110
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 110
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 110
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 109
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 109
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 108
N-Pyrrylarylsulfones with High Therapeutic Potential 108
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 104
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 103
Antimycobacterial activity of ionic fullerene derivatives. 102
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 102
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 102
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 101
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 100
The emerging role of lysine methyltransferase SETD8 in human diseases 100
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 99
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 98
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 97
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 96
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 96
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 96
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 96
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 95
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 95
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 93
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 92
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 92
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 90
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 90
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 90
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 89
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 87
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 87
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 87
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 86
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 85
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 85
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 84
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 84
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 84
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 84
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 80
Lysine methyltransferase inhibitors: where we are now. 80
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 78
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 77
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 77
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 77
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 76
Synthesis of tricyclic triazepinones related to nevirapine. 75
Enhancement of lysine acetylation accelerates wound repair 74
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 73
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 73
Synthesis and pharmacological characterization of new analogs of broxaterol. 72
Totale 14.936
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Categoria #
all - tutte 47.781
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 47.781
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021617 0 0 0 0 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/20266.729 1.139 2.239 2.228 439 684 0 0 0 0 0 0 0
Totale 15.851