UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
Salva come PNG Salva come JPEG
Continente #
NA - Nord America 5.192
EU - Europa 1.592
AS - Asia 1.344
SA - Sud America 232
AF - Africa 22
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 1
Totale 8.389
Salva come PNG Salva come JPEG
Nazione #
US - Stati Uniti d'America 5.176
SG - Singapore 479
IT - Italia 459
CN - Cina 389
UA - Ucraina 305
RU - Federazione Russa 294
BR - Brasile 208
VN - Vietnam 180
TR - Turchia 167
IE - Irlanda 135
DE - Germania 116
SE - Svezia 94
FI - Finlandia 69
KR - Corea 48
FR - Francia 38
IN - India 28
GB - Regno Unito 19
HK - Hong Kong 19
AT - Austria 15
CZ - Repubblica Ceca 11
AR - Argentina 10
NL - Olanda 7
PK - Pakistan 7
EU - Europa 6
MA - Marocco 6
PE - Perù 6
GR - Grecia 5
HU - Ungheria 5
IQ - Iraq 5
CA - Canada 4
ZA - Sudafrica 4
BG - Bulgaria 3
IL - Israele 3
JO - Giordania 3
MX - Messico 3
PA - Panama 3
PL - Polonia 3
RO - Romania 3
TN - Tunisia 3
UZ - Uzbekistan 3
AZ - Azerbaigian 2
BE - Belgio 2
CL - Cile 2
CO - Colombia 2
DO - Repubblica Dominicana 2
DZ - Algeria 2
EC - Ecuador 2
HR - Croazia 2
IR - Iran 2
JP - Giappone 2
NO - Norvegia 2
SA - Arabia Saudita 2
VE - Venezuela 2
AL - Albania 1
BD - Bangladesh 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
CH - Svizzera 1
CM - Camerun 1
EG - Egitto 1
ES - Italia 1
GH - Ghana 1
GT - Guatemala 1
ID - Indonesia 1
KE - Kenya 1
KH - Cambogia 1
LU - Lussemburgo 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
PH - Filippine 1
PS - Palestinian Territory 1
RS - Serbia 1
SC - Seychelles 1
TT - Trinidad e Tobago 1
Totale 8.389
Salva come PNG Salva come JPEG
Città #
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Jacksonville 420
Houston 417
Princeton 384
Wilmington 310
Dong Ket 177
Salerno 167
Singapore 164
Izmir 160
Ashburn 159
Dublin 128
Beijing 101
Nanjing 82
Andover 78
Boardman 78
Moscow 52
Pellezzano 51
Dearborn 41
Fairfield 40
Hebei 34
Shenyang 25
Mestre 21
Nanchang 20
Pune 20
Hong Kong 17
Philadelphia 17
Rome 17
Changsha 16
Fisciano 16
Norwalk 16
São Paulo 16
Council Bluffs 15
Jiaxing 15
Redwood City 15
Düsseldorf 13
Falls Church 13
Dallas 12
Guangzhou 12
Los Angeles 12
Tianjin 12
Washington 12
Brno 11
New York 10
Seattle 10
Cambridge 9
Nuremberg 9
Shanghai 9
Munich 8
Jinan 7
Napoli 7
San Diego 7
Helsinki 6
Indiana 6
Munro 6
Renton 6
Tappahannock 6
The Dalles 6
Vienna 6
Florence 5
Palermo 5
Sarno 5
Sorrento 5
Spinea 5
Campinas 4
Edinburgh 4
Joinville 4
Menlo Park 4
Naples 4
Stockholm 4
Amman 3
Belo Horizonte 3
Cagliari 3
Casoria 3
Catania 3
Clifton 3
Durham 3
Fortaleza 3
Hefei 3
Lappeenranta 3
London 3
Marcianise 3
Messina 3
Montes Claros 3
Mugnano del Cardinale 3
Newcastle upon Tyne 3
Néa Smýrni 3
Orange 3
Panama City 3
Santa Clara 3
Scafati 3
São Gonçalo 3
Tashkent 3
Warsaw 3
Wuhan 3
Acerra 2
Aparecida de Goiânia 2
Athens 2
Atlanta 2
Totale 6.122
Salva come PNG Salva come JPEG
Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 166
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 166
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 146
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 135
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 126
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 126
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 125
Microbiologia Molecolare e Cellulare 123
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 123
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 120
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 118
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 118
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 117
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 116
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 115
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 115
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 114
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 114
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 108
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 106
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 105
Azole antifungal agents related to naftifine and butenafine 101
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 99
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 99
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 99
Chemical biology of Histone acetyltransferase natural compounds modulators. 96
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 96
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 96
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 95
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 95
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 94
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 94
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 94
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 93
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 90
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 89
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 88
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 87
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 87
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 86
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 85
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 85
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 84
Antimycobacterial activity of ionic fullerene derivatives. 82
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 82
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 82
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 81
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 79
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 79
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 78
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 78
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 77
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 77
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 76
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 76
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 76
N-Pyrrylarylsulfones with High Therapeutic Potential 75
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 75
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 74
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 74
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 74
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 73
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 72
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 72
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 72
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 71
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 71
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 70
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 70
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 69
The emerging role of lysine methyltransferase SETD8 in human diseases 69
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 69
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 68
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 68
Enhancement of lysine acetylation accelerates wound repair 67
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 64
Synthesis of tricyclic triazepinones related to nevirapine. 63
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 63
Synthesis and pharmacological characterization of new analogs of broxaterol. 61
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 60
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 60
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 59
Design and Synthesis of Novel [60]Fullerene Derivatives as Potential HIV Aspartic Protease Inhibitors. 58
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 58
Discovery of new chemical probes for the MRG15 chromo domain. 57
Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives. 56
Lysine methyltransferase inhibitors: where we are now. 56
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 55
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 54
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 54
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 52
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 50
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 49
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 44
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 44
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 43
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 41
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 39
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 38
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 38
Totale 8.326
Salva come PNG Salva come JPEG
Categoria #
all - tutte 30.871
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 30.871
Salva come PNG Salva come JPEG


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020147 0 0 0 0 0 0 0 0 0 0 142 5
2020/2021785 5 71 88 4 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.259 66 25 31 69 121 171 263 148 280 78 7 0
Totale 8.680