UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
NA - Nord America 5.115
EU - Europa 1.245
AS - Asia 878
SA - Sud America 13
Continente sconosciuto - Info sul continente non disponibili 6
AF - Africa 4
OC - Oceania 1
Totale 7.262
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Nazione #
US - Stati Uniti d'America 5.106
IT - Italia 435
CN - Cina 364
UA - Ucraina 304
VN - Vietnam 178
TR - Turchia 161
IE - Irlanda 135
SG - Singapore 134
DE - Germania 101
SE - Svezia 94
FI - Finlandia 63
FR - Francia 38
IN - India 21
GB - Regno Unito 19
CZ - Repubblica Ceca 11
RU - Federazione Russa 9
AR - Argentina 6
EU - Europa 6
AT - Austria 5
GR - Grecia 5
HU - Ungheria 5
KR - Corea 5
PE - Perù 5
BG - Bulgaria 3
CA - Canada 3
IL - Israele 3
NL - Olanda 3
PA - Panama 3
RO - Romania 3
BE - Belgio 2
CL - Cile 2
HK - Hong Kong 2
HR - Croazia 2
IR - Iran 2
JP - Giappone 2
NO - Norvegia 2
PL - Polonia 2
SA - Arabia Saudita 2
BZ - Belize 1
CH - Svizzera 1
CM - Camerun 1
EG - Egitto 1
ES - Italia 1
GH - Ghana 1
ID - Indonesia 1
KH - Cambogia 1
LU - Lussemburgo 1
MX - Messico 1
NZ - Nuova Zelanda 1
PH - Filippine 1
PK - Pakistan 1
RS - Serbia 1
SC - Seychelles 1
TT - Trinidad e Tobago 1
Totale 7.262
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Città #
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Jacksonville 420
Houston 417
Princeton 384
Wilmington 310
Dong Ket 177
Salerno 167
Izmir 160
Ashburn 155
Dublin 128
Beijing 101
Nanjing 82
Andover 78
Boardman 78
Singapore 78
Pellezzano 51
Dearborn 41
Fairfield 40
Hebei 34
Shenyang 25
Mestre 21
Nanchang 20
Philadelphia 17
Norwalk 16
Pune 16
Changsha 15
Fisciano 15
Jiaxing 15
Redwood City 15
Rome 15
Düsseldorf 13
Falls Church 13
Dallas 12
Tianjin 12
Washington 12
Brno 11
Guangzhou 11
Seattle 10
Cambridge 9
Jinan 7
Los Angeles 7
Napoli 7
San Diego 7
Indiana 6
Munro 6
Renton 6
Tappahannock 6
Florence 5
New York 5
Palermo 5
Sorrento 5
Spinea 5
Edinburgh 4
Menlo Park 4
Naples 4
Stockholm 4
Cagliari 3
Casoria 3
Catania 3
Clifton 3
Hefei 3
Lappeenranta 3
London 3
Marcianise 3
Messina 3
Mugnano del Cardinale 3
Munich 3
Newcastle upon Tyne 3
Néa Smýrni 3
Orange 3
Panama City 3
Scafati 3
Shanghai 3
Vienna 3
Wuhan 3
Acerra 2
Athens 2
Atlanta 2
Bisamberg 2
Brussels 2
Caivano 2
Calvisano 2
Chicago 2
Contrada 2
Durham 2
Hangzhou 2
Hanover 2
Kolkata 2
Krimpen Aan Den Ijssel 2
Maddaloni 2
Mercato San Severino 2
Montreal 2
Mumbai 2
Nocera Superiore 2
Nürnberg 2
Oslo 2
Pescara 2
Seoul 2
Totale 5.876
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Nome #
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 155
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 147
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 122
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 119
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 118
Microbiologia Molecolare e Cellulare 117
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 117
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 115
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 112
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 108
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 107
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 106
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 103
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 103
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 99
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 98
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 98
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 96
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 94
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 94
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 93
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 92
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 91
Azole antifungal agents related to naftifine and butenafine 90
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 90
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 89
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 89
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 88
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 88
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 85
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 85
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 84
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 83
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 83
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 83
Chemical biology of Histone acetyltransferase natural compounds modulators. 82
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 82
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 82
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 80
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 79
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 76
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 75
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 75
Antimycobacterial activity of ionic fullerene derivatives. 74
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 74
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 74
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 73
N-Pyrrylarylsulfones with High Therapeutic Potential 72
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 71
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 70
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 70
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 70
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 69
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 68
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 67
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 67
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 65
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 63
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 63
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 63
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 63
Enhancement of lysine acetylation accelerates wound repair 62
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 62
Synthesis of tricyclic triazepinones related to nevirapine. 61
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 61
The emerging role of lysine methyltransferase SETD8 in human diseases 61
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 61
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 60
Synthesis and pharmacological characterization of new analogs of broxaterol. 59
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 59
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 58
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 58
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 57
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 57
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 57
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 57
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 57
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 56
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 56
Design and Synthesis of Novel [60]Fullerene Derivatives as Potential HIV Aspartic Protease Inhibitors. 55
Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives. 54
Lysine methyltransferase inhibitors: where we are now. 52
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 51
Discovery of new chemical probes for the MRG15 chromo domain. 48
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 47
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 46
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 45
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 45
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 43
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 41
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 39
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 37
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 36
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 36
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 35
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 34
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 34
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 33
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 26
Polycyclic maleimide-based derivatives as first dual modulators of neuronal calcium channels and GSK-3β for Alzheimer's disease treatment 25
Totale 7.329
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Categoria #
all - tutte 23.343
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 23.343
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020529 0 0 75 10 60 21 72 12 71 61 142 5
2020/2021785 5 71 88 4 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/2025113 66 25 22 0 0 0 0 0 0 0 0 0
Totale 7.534