UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 6.482
NA - Nord America 5.929
EU - Europa 1.803
SA - Sud America 446
AF - Africa 51
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 2
Totale 14.719
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Nazione #
US - Stati Uniti d'America 5.869
HK - Hong Kong 4.742
SG - Singapore 606
CN - Cina 499
IT - Italia 478
BR - Brasile 383
UA - Ucraina 310
RU - Federazione Russa 300
VN - Vietnam 229
DE - Germania 189
TR - Turchia 173
IE - Irlanda 135
SE - Svezia 98
FI - Finlandia 97
KR - Corea 88
IN - India 48
GB - Regno Unito 47
FR - Francia 41
CA - Canada 26
AR - Argentina 23
MX - Messico 20
PL - Polonia 19
JP - Giappone 17
AT - Austria 16
CZ - Repubblica Ceca 16
ID - Indonesia 15
BD - Bangladesh 14
ES - Italia 12
ZA - Sudafrica 12
IQ - Iraq 11
PE - Perù 11
PK - Pakistan 11
NL - Olanda 9
CO - Colombia 8
MA - Marocco 8
EC - Ecuador 7
UZ - Uzbekistan 7
EU - Europa 6
GR - Grecia 6
DZ - Algeria 5
HU - Ungheria 5
PY - Paraguay 5
RO - Romania 5
CL - Cile 4
EG - Egitto 4
IL - Israele 4
TN - Tunisia 4
VE - Venezuela 4
BG - Bulgaria 3
JO - Giordania 3
KE - Kenya 3
PA - Panama 3
TT - Trinidad e Tobago 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
BE - Belgio 2
CG - Congo 2
CH - Svizzera 2
DO - Repubblica Dominicana 2
HR - Croazia 2
IR - Iran 2
KZ - Kazakistan 2
LT - Lituania 2
LY - Libia 2
NO - Norvegia 2
NZ - Nuova Zelanda 2
PS - Palestinian Territory 2
RS - Serbia 2
SA - Arabia Saudita 2
AL - Albania 1
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CM - Camerun 1
CR - Costa Rica 1
DM - Dominica 1
ET - Etiopia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
IS - Islanda 1
JM - Giamaica 1
KH - Cambogia 1
LU - Lussemburgo 1
MW - Malawi 1
MY - Malesia 1
MZ - Mozambico 1
NA - Namibia 1
NG - Nigeria 1
NI - Nicaragua 1
PH - Filippine 1
PT - Portogallo 1
SC - Seychelles 1
SN - Senegal 1
UY - Uruguay 1
Totale 14.719
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Città #
Hong Kong 4.734
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Jacksonville 421
Houston 418
Princeton 384
Dallas 324
Wilmington 311
Singapore 222
Ashburn 209
Dong Ket 177
Salerno 167
Izmir 160
Beijing 144
Dublin 128
Nanjing 82
Boardman 79
Andover 78
Munich 78
Moscow 52
Pellezzano 51
Dearborn 41
Fairfield 40
Los Angeles 40
The Dalles 36
Columbus 34
Hebei 34
São Paulo 34
New York 28
Santa Clara 27
Turku 26
Shenyang 25
Mestre 21
Nanchang 20
Pune 20
Rome 19
Council Bluffs 18
Philadelphia 17
Warsaw 17
Changsha 16
Fisciano 16
Norwalk 16
Seoul 16
Ho Chi Minh City 15
Jiaxing 15
Redwood City 15
Tokyo 15
Boston 14
Brooklyn 14
Düsseldorf 13
Falls Church 13
Seattle 13
Washington 13
Guangzhou 12
Nuremberg 12
San Francisco 12
Tianjin 12
Brno 11
Chicago 11
Montreal 11
Chennai 10
Jakarta 10
Rio de Janeiro 10
Belo Horizonte 9
Cambridge 9
Hanoi 9
London 9
Mexico City 9
Scafati 9
Shanghai 9
Johannesburg 8
Atlanta 7
Denver 7
Helsinki 7
Jinan 7
Manchester 7
Napoli 7
San Diego 7
Santo André 7
Stockholm 7
Tashkent 7
Vienna 7
Ankara 6
Campinas 6
Indiana 6
Joinville 6
Munro 6
Naples 6
Renton 6
Tappahannock 6
Florence 5
Guarulhos 5
Palermo 5
Sarno 5
Sorrento 5
Spinea 5
Brasília 4
Charlotte 4
Da Nang 4
Totale 11.755
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.200
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 654
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 482
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 429
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 404
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 365
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 344
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 253
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 230
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 227
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 220
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 209
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 204
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 192
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 180
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 177
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 172
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 162
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 157
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 148
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 140
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 139
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 137
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 134
Microbiologia Molecolare e Cellulare 133
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 133
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 132
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 131
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 130
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 129
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 126
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 124
Chemical biology of Histone acetyltransferase natural compounds modulators. 123
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 123
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 122
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 121
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 119
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 116
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 116
Azole antifungal agents related to naftifine and butenafine 110
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 110
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 107
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 107
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 106
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 105
N-Pyrrylarylsulfones with High Therapeutic Potential 105
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 105
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 104
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 103
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 103
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 103
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 102
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 101
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 100
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 100
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 99
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 98
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 95
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 95
Antimycobacterial activity of ionic fullerene derivatives. 94
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 94
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 94
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 94
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 93
The emerging role of lysine methyltransferase SETD8 in human diseases 93
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 92
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 91
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 90
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 89
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 88
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 85
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 85
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 85
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 84
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 83
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 83
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 82
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 82
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 82
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 81
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 80
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 79
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 78
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 77
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 77
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 76
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 75
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 75
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 74
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 74
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 73
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 73
Lysine methyltransferase inhibitors: where we are now. 73
Enhancement of lysine acetylation accelerates wound repair 72
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 72
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 71
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 70
Synthesis of tricyclic triazepinones related to nevirapine. 69
Synthesis and pharmacological characterization of new analogs of broxaterol. 67
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 67
Totale 14.211
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Categoria #
all - tutte 45.966
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 45.966
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021621 0 0 0 4 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/20265.889 1.139 2.239 2.228 283 0 0 0 0 0 0 0 0
Totale 15.011