UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 8.113
NA - Nord America 7.981
EU - Europa 2.742
SA - Sud America 647
Continente sconosciuto - Info sul continente non disponibili 308
AF - Africa 99
OC - Oceania 3
Totale 19.893
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Nazione #
US - Stati Uniti d'America 7.801
HK - Hong Kong 4.880
SG - Singapore 1.391
IT - Italia 1.128
CN - Cina 692
BR - Brasile 488
VN - Vietnam 462
UA - Ucraina 321
RU - Federazione Russa 309
DE - Germania 225
TR - Turchia 189
FR - Francia 143
IE - Irlanda 137
IN - India 109
FI - Finlandia 105
KR - Corea 104
SE - Svezia 104
GB - Regno Unito 91
CA - Canada 74
BD - Bangladesh 67
AR - Argentina 57
MX - Messico 49
JP - Giappone 38
PL - Polonia 36
IQ - Iraq 32
PK - Pakistan 27
ZA - Sudafrica 27
ID - Indonesia 26
ES - Italia 24
NL - Olanda 24
CO - Colombia 21
EC - Ecuador 21
AT - Austria 18
CZ - Repubblica Ceca 18
VE - Venezuela 16
UZ - Uzbekistan 15
JM - Giamaica 14
MA - Marocco 14
CL - Cile 13
PE - Perù 13
IL - Israele 12
PH - Filippine 12
DZ - Algeria 11
PY - Paraguay 10
GR - Grecia 9
MY - Malesia 8
SA - Arabia Saudita 8
TN - Tunisia 8
AE - Emirati Arabi Uniti 7
HN - Honduras 7
TT - Trinidad e Tobago 7
AL - Albania 6
BO - Bolivia 6
EG - Egitto 6
ET - Etiopia 6
EU - Europa 6
JO - Giordania 6
KE - Kenya 6
RO - Romania 6
AZ - Azerbaigian 5
CR - Costa Rica 5
HU - Ungheria 5
PA - Panama 5
BG - Bulgaria 4
CH - Svizzera 4
GT - Guatemala 4
LY - Libia 4
BE - Belgio 3
DO - Repubblica Dominicana 3
HR - Croazia 3
IR - Iran 3
LB - Libano 3
LT - Lituania 3
NI - Nicaragua 3
NO - Norvegia 3
PR - Porto Rico 3
BB - Barbados 2
CG - Congo 2
KZ - Kazakistan 2
LU - Lussemburgo 2
NG - Nigeria 2
NP - Nepal 2
NZ - Nuova Zelanda 2
OM - Oman 2
PS - Palestinian Territory 2
PT - Portogallo 2
RS - Serbia 2
SV - El Salvador 2
UY - Uruguay 2
AM - Armenia 1
AO - Angola 1
AU - Australia 1
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CI - Costa d'Avorio 1
CM - Camerun 1
CW - ???statistics.table.value.countryCode.CW??? 1
CY - Cipro 1
DK - Danimarca 1
Totale 19.570
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Città #
Hong Kong 4.865
Ann Arbor 1.456
Singapore 717
San Jose 635
Chandler 527
Woodbridge 503
Houston 428
Jacksonville 422
Ashburn 395
Princeton 384
Milan 372
Dallas 339
Wilmington 311
Council Bluffs 244
Beijing 212
Salerno 181
Dong Ket 177
Izmir 160
Dublin 130
The Dalles 121
Ho Chi Minh City 105
Rome 96
Lauterbourg 95
Munich 87
Nanjing 82
Santa Clara 82
Boardman 79
Andover 78
Los Angeles 72
Hanoi 62
New York 58
Moscow 53
Pellezzano 51
São Paulo 46
Dearborn 41
Fairfield 40
Columbus 36
Figino 36
Hebei 34
Tokyo 33
Warsaw 33
Brooklyn 27
Chicago 27
Shenyang 26
Turku 26
Montreal 25
Naples 24
Orem 24
Phoenix 22
Pune 22
Fisciano 21
Mestre 21
Philadelphia 21
Atlanta 20
Denver 20
Nanchang 20
Basingstoke 19
Frankfurt am Main 19
Memphis 18
Seattle 18
Mexico City 17
Rio de Janeiro 17
Boston 16
Changsha 16
Jiaxing 16
Johannesburg 16
Norwalk 16
San Francisco 16
Seoul 16
Turin 16
Helsinki 15
Nuremberg 15
Redwood City 15
Tashkent 15
Chennai 14
Guangzhou 14
Jakarta 14
Washington 14
Amsterdam 13
Düsseldorf 13
Falls Church 13
Shanghai 13
Stockholm 13
Baghdad 12
Belo Horizonte 12
Buffalo 12
Haiphong 12
London 12
Tianjin 12
Toronto 12
Brno 11
Da Nang 11
Hải Dương 11
Poplar 11
Ankara 10
Baronissi 9
Cambridge 9
Campinas 9
Florence 9
Lahore 9
Totale 14.824
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.251
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 692
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 535
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 470
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 445
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 387
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 380
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 306
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 273
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 272
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 260
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 259
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 252
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 249
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 240
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 232
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 219
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 214
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 208
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 202
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 200
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 191
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 185
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 179
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 176
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 174
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 174
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 171
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 170
Microbiologia Molecolare e Cellulare 169
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 169
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 166
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 166
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 165
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 165
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 164
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 162
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 161
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 160
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 159
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 158
Chemical biology of Histone acetyltransferase natural compounds modulators. 154
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 152
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 152
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 149
Azole antifungal agents related to naftifine and butenafine 148
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 148
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 146
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 144
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 139
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 139
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 138
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 136
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 135
Antimycobacterial activity of ionic fullerene derivatives. 135
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 135
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 133
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 131
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 130
The emerging role of lysine methyltransferase SETD8 in human diseases 130
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 130
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 129
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 129
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 128
N-Pyrrylarylsulfones with High Therapeutic Potential 128
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 128
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 128
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 127
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 127
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 126
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 126
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 126
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 125
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 125
Exploiting acylaminopyrazole scaffold for polypharmacology approach in Alzheimer's disease 124
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 123
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 122
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 121
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 120
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 120
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 117
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 117
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 116
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 116
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 113
Lysine methyltransferase inhibitors: where we are now. 112
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 111
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 111
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 111
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 110
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 107
Discovery of new chemical probes for the MRG15 chromo domain. 106
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 105
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 105
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 105
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 104
Synthesis and pharmacological characterization of new analogs of broxaterol. 102
Enhancement of lysine acetylation accelerates wound repair 102
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 101
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 100
Totale 18.287
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Categoria #
all - tutte 58.960
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 58.960
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022726 0 0 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/202610.024 1.139 2.239 2.228 439 719 324 895 234 406 562 159 680
2026/2027747 242 208 297 0 0 0 0 0 0 0 0 0
Totale 19.893