UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 7.283
NA - Nord America 6.494
EU - Europa 1.881
SA - Sud America 519
AF - Africa 64
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 2
Totale 16.249
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Nazione #
US - Stati Uniti d'America 6.410
HK - Hong Kong 4.743
SG - Singapore 1.192
CN - Cina 600
IT - Italia 491
BR - Brasile 428
UA - Ucraina 312
RU - Federazione Russa 303
VN - Vietnam 301
DE - Germania 202
TR - Turchia 176
IE - Irlanda 135
SE - Svezia 102
FI - Finlandia 97
KR - Corea 88
GB - Regno Unito 59
IN - India 59
FR - Francia 42
AR - Argentina 36
CA - Canada 36
MX - Messico 32
PL - Polonia 32
JP - Giappone 26
ES - Italia 19
ID - Indonesia 17
ZA - Sudafrica 17
AT - Austria 16
BD - Bangladesh 16
CZ - Repubblica Ceca 16
NL - Olanda 15
EC - Ecuador 13
IQ - Iraq 13
PK - Pakistan 13
CO - Colombia 11
PE - Perù 11
DZ - Algeria 9
MA - Marocco 9
UZ - Uzbekistan 8
PY - Paraguay 7
CL - Cile 6
EU - Europa 6
GR - Grecia 6
RO - Romania 6
TN - Tunisia 6
HU - Ungheria 5
SA - Arabia Saudita 5
EG - Egitto 4
IL - Israele 4
KE - Kenya 4
VE - Venezuela 4
AE - Emirati Arabi Uniti 3
BG - Bulgaria 3
JO - Giordania 3
LT - Lituania 3
PA - Panama 3
TT - Trinidad e Tobago 3
AL - Albania 2
AZ - Azerbaigian 2
BE - Belgio 2
BO - Bolivia 2
CG - Congo 2
CH - Svizzera 2
DO - Repubblica Dominicana 2
HR - Croazia 2
IR - Iran 2
JM - Giamaica 2
KZ - Kazakistan 2
LB - Libano 2
LY - Libia 2
NO - Norvegia 2
NZ - Nuova Zelanda 2
PH - Filippine 2
PS - Palestinian Territory 2
RS - Serbia 2
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CM - Camerun 1
CR - Costa Rica 1
DM - Dominica 1
EE - Estonia 1
ET - Etiopia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
HN - Honduras 1
IS - Islanda 1
KH - Cambogia 1
KW - Kuwait 1
LU - Lussemburgo 1
MW - Malawi 1
MY - Malesia 1
MZ - Mozambico 1
NA - Namibia 1
NG - Nigeria 1
NI - Nicaragua 1
NP - Nepal 1
PT - Portogallo 1
SC - Seychelles 1
SN - Senegal 1
Totale 16.248
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Città #
Hong Kong 4.735
Ann Arbor 1.456
Singapore 573
Chandler 527
Woodbridge 503
Houston 425
Jacksonville 421
Princeton 384
Dallas 325
Wilmington 311
Ashburn 297
San Jose 246
Dong Ket 177
Salerno 167
Beijing 165
Izmir 160
Dublin 128
Munich 87
Nanjing 82
Boardman 79
Andover 78
Los Angeles 63
The Dalles 62
Moscow 52
Pellezzano 51
Ho Chi Minh City 43
New York 43
Dearborn 41
São Paulo 41
Fairfield 40
Columbus 34
Hebei 34
Warsaw 30
Santa Clara 28
Shenyang 26
Turku 26
Tokyo 24
Hanoi 22
Mestre 21
Montreal 20
Nanchang 20
Pune 20
Rome 20
Council Bluffs 18
Denver 18
Atlanta 17
Philadelphia 17
Brooklyn 16
Changsha 16
Chicago 16
Fisciano 16
Norwalk 16
Seattle 16
Seoul 16
Boston 15
Jiaxing 15
Redwood City 15
Guangzhou 14
Düsseldorf 13
Falls Church 13
Washington 13
Belo Horizonte 12
Chennai 12
Mexico City 12
Nuremberg 12
San Francisco 12
Tianjin 12
Brno 11
Johannesburg 11
Phoenix 11
Poplar 11
Rio de Janeiro 11
Shanghai 11
Stockholm 11
Jakarta 10
London 10
Ankara 9
Baronissi 9
Cambridge 9
Orem 9
Scafati 9
Amsterdam 8
Campinas 8
Tashkent 8
Helsinki 7
Jinan 7
Manchester 7
Naples 7
Napoli 7
San Diego 7
Santo André 7
Vienna 7
Da Nang 6
Guarulhos 6
Indiana 6
Joinville 6
Munro 6
Renton 6
Tappahannock 6
Brasília 5
Totale 12.708
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.215
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 671
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 499
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 441
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 417
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 370
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 358
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 277
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 246
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 243
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 230
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 223
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 217
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 216
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 204
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 193
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 182
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 175
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 175
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 166
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 159
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 155
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 155
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 151
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 147
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 147
Microbiologia Molecolare e Cellulare 146
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 145
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 142
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 140
Chemical biology of Histone acetyltransferase natural compounds modulators. 137
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 137
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 137
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 137
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 136
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 135
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 132
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 131
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 131
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 125
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 125
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 125
Azole antifungal agents related to naftifine and butenafine 121
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 121
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 120
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 119
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 117
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 116
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 116
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 116
N-Pyrrylarylsulfones with High Therapeutic Potential 115
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 114
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 112
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 112
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 111
The emerging role of lysine methyltransferase SETD8 in human diseases 109
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 109
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 107
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 106
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 106
Antimycobacterial activity of ionic fullerene derivatives. 105
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 105
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 105
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 105
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 104
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 103
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 102
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 101
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 101
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 101
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 101
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 100
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 100
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 98
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 98
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 95
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 95
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 95
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 95
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 94
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 92
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 92
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 91
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 91
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 89
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 88
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 87
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 87
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 87
Lysine methyltransferase inhibitors: where we are now. 87
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 85
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 82
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 82
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 81
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 80
Discovery of new chemical probes for the MRG15 chromo domain. 79
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 78
Enhancement of lysine acetylation accelerates wound repair 78
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 78
Synthesis and pharmacological characterization of new analogs of broxaterol. 77
Totale 15.534
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Categoria #
all - tutte 49.318
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 49.318
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021500 0 0 0 0 0 0 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/20267.421 1.139 2.239 2.228 439 719 324 333 0 0 0 0 0
Totale 16.543