UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
AS - Asia 7.971
NA - Nord America 7.137
EU - Europa 2.118
SA - Sud America 632
AF - Africa 98
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 3
Totale 17.965
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Nazione #
US - Stati Uniti d'America 7.027
HK - Hong Kong 4.856
SG - Singapore 1.364
CN - Cina 649
IT - Italia 519
BR - Brasile 476
VN - Vietnam 460
UA - Ucraina 321
RU - Federazione Russa 309
DE - Germania 225
TR - Turchia 189
FR - Francia 142
IE - Irlanda 137
FI - Finlandia 105
KR - Corea 104
IN - India 102
SE - Svezia 102
GB - Regno Unito 88
AR - Argentina 57
MX - Messico 45
CA - Canada 39
BD - Bangladesh 37
JP - Giappone 36
PL - Polonia 35
IQ - Iraq 32
PK - Pakistan 27
ZA - Sudafrica 26
ID - Indonesia 25
ES - Italia 23
NL - Olanda 22
CO - Colombia 21
EC - Ecuador 19
AT - Austria 18
CZ - Repubblica Ceca 17
UZ - Uzbekistan 15
VE - Venezuela 15
MA - Marocco 14
CL - Cile 13
PE - Perù 13
DZ - Algeria 11
PH - Filippine 11
IL - Israele 10
PY - Paraguay 10
GR - Grecia 9
TN - Tunisia 8
MY - Malesia 7
SA - Arabia Saudita 7
AE - Emirati Arabi Uniti 6
AL - Albania 6
BO - Bolivia 6
EG - Egitto 6
ET - Etiopia 6
EU - Europa 6
JO - Giordania 6
KE - Kenya 6
RO - Romania 6
AZ - Azerbaigian 5
HU - Ungheria 5
PA - Panama 5
BG - Bulgaria 4
HN - Honduras 4
LY - Libia 4
BE - Belgio 3
CH - Svizzera 3
DO - Repubblica Dominicana 3
HR - Croazia 3
IR - Iran 3
JM - Giamaica 3
LB - Libano 3
LT - Lituania 3
TT - Trinidad e Tobago 3
CG - Congo 2
GT - Guatemala 2
KZ - Kazakistan 2
LU - Lussemburgo 2
NG - Nigeria 2
NI - Nicaragua 2
NO - Norvegia 2
NP - Nepal 2
NZ - Nuova Zelanda 2
OM - Oman 2
PS - Palestinian Territory 2
RS - Serbia 2
UY - Uruguay 2
AM - Armenia 1
AO - Angola 1
AU - Australia 1
BA - Bosnia-Erzegovina 1
BW - Botswana 1
BZ - Belize 1
CI - Costa d'Avorio 1
CM - Camerun 1
CR - Costa Rica 1
CY - Cipro 1
DK - Danimarca 1
DM - Dominica 1
EE - Estonia 1
GH - Ghana 1
GN - Guinea 1
IS - Islanda 1
Totale 17.947
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Città #
Hong Kong 4.842
Ann Arbor 1.456
Singapore 697
Chandler 527
San Jose 527
Woodbridge 503
Houston 425
Jacksonville 421
Princeton 384
Ashburn 361
Dallas 325
Wilmington 311
Beijing 177
Dong Ket 177
Salerno 167
Izmir 160
Council Bluffs 132
Dublin 130
The Dalles 119
Ho Chi Minh City 105
Lauterbourg 95
Munich 87
Nanjing 82
Boardman 79
Andover 78
Los Angeles 65
Hanoi 61
Moscow 53
Pellezzano 51
New York 47
São Paulo 44
Santa Clara 43
Dearborn 41
Fairfield 40
Columbus 34
Hebei 34
Tokyo 33
Warsaw 31
Shenyang 26
Turku 26
Rome 23
Pune 22
Fisciano 21
Mestre 21
Montreal 21
Nanchang 20
Orem 20
Basingstoke 19
Frankfurt am Main 19
Atlanta 18
Denver 18
Philadelphia 18
Chicago 17
Rio de Janeiro 17
Boston 16
Brooklyn 16
Changsha 16
Jiaxing 16
Norwalk 16
Seattle 16
Seoul 16
Helsinki 15
Johannesburg 15
Nuremberg 15
Redwood City 15
Tashkent 15
Chennai 14
Guangzhou 14
Mexico City 14
Naples 14
Amsterdam 13
Düsseldorf 13
Falls Church 13
Jakarta 13
Shanghai 13
Washington 13
Baghdad 12
Belo Horizonte 12
Haiphong 12
London 12
San Francisco 12
Tianjin 12
Brno 11
Da Nang 11
Hải Dương 11
Phoenix 11
Poplar 11
Stockholm 11
Ankara 10
Baronissi 9
Cambridge 9
Campinas 9
Lahore 9
Scafati 9
City of London 8
Karachi 8
Manchester 8
Vienna 8
Guarulhos 7
Jinan 7
Totale 13.830
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.240
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 685
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 522
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 457
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 432
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 375
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 373
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 292
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 260
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 258
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 245
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 239
Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors 239
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 228
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 227
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 218
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 206
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 196
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 191
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 190
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 179
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 178
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 173
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 167
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 166
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 165
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 162
Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold 160
Microbiologia Molecolare e Cellulare 157
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 157
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 156
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 155
Chemical biology of Histone acetyltransferase natural compounds modulators. 151
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 151
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 150
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 147
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 147
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 145
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 145
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 145
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 144
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 143
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 140
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 140
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 140
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 137
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 136
Azole antifungal agents related to naftifine and butenafine 135
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 127
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 127
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 127
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 126
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 125
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 123
N-Pyrrylarylsulfones with High Therapeutic Potential 122
Antimycobacterial activity of ionic fullerene derivatives. 121
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 121
The emerging role of lysine methyltransferase SETD8 in human diseases 121
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 121
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 120
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 120
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 119
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 119
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 117
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 117
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 116
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 115
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 115
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 114
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 113
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 113
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 113
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 113
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 112
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 112
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 112
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 112
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 111
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 110
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 107
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 106
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 105
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 104
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 104
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 102
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 100
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 100
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 98
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 96
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 95
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 95
Lysine methyltransferase inhibitors: where we are now. 95
Discovery of new chemical probes for the MRG15 chromo domain. 93
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 92
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 91
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 89
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 89
Enhancement of lysine acetylation accelerates wound repair 88
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 88
Synthesis and pharmacological characterization of new analogs of broxaterol. 86
Totale 17.021
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Categoria #
all - tutte 51.824
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 51.824
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021310 0 0 0 0 0 0 0 0 0 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/20269.139 1.139 2.239 2.228 439 719 324 895 234 406 516 0 0
Totale 18.261