UniSa - IRIS Institutional Research Information System

CASTELLANO, Sabrina
 Distribuzione geografica
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Continente #
NA - Nord America 5.407
EU - Europa 1.724
AS - Asia 1.496
SA - Sud America 294
AF - Africa 30
Continente sconosciuto - Info sul continente non disponibili 6
OC - Oceania 1
Totale 8.958
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Nazione #
US - Stati Uniti d'America 5.373
SG - Singapore 504
IT - Italia 460
CN - Cina 408
UA - Ucraina 306
RU - Federazione Russa 298
BR - Brasile 265
DE - Germania 188
VN - Vietnam 182
TR - Turchia 169
IE - Irlanda 135
SE - Svezia 95
FI - Finlandia 92
HK - Hong Kong 75
KR - Corea 74
FR - Francia 39
GB - Regno Unito 34
IN - India 32
AT - Austria 15
CZ - Repubblica Ceca 15
CA - Canada 14
PK - Pakistan 11
AR - Argentina 10
MX - Messico 10
IQ - Iraq 9
NL - Olanda 8
PE - Perù 8
PL - Polonia 7
ZA - Sudafrica 7
BD - Bangladesh 6
EU - Europa 6
MA - Marocco 6
DZ - Algeria 5
ES - Italia 5
GR - Grecia 5
HU - Ungheria 5
IL - Israele 4
RO - Romania 4
UZ - Uzbekistan 4
BG - Bulgaria 3
CL - Cile 3
CO - Colombia 3
EC - Ecuador 3
JO - Giordania 3
JP - Giappone 3
PA - Panama 3
TN - Tunisia 3
AZ - Azerbaigian 2
BE - Belgio 2
DO - Repubblica Dominicana 2
HR - Croazia 2
IR - Iran 2
KE - Kenya 2
NO - Norvegia 2
PS - Palestinian Territory 2
SA - Arabia Saudita 2
TT - Trinidad e Tobago 2
VE - Venezuela 2
AL - Albania 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
CH - Svizzera 1
CM - Camerun 1
EG - Egitto 1
ET - Etiopia 1
GH - Ghana 1
GT - Guatemala 1
ID - Indonesia 1
KH - Cambogia 1
KZ - Kazakistan 1
LU - Lussemburgo 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
PH - Filippine 1
RS - Serbia 1
SC - Seychelles 1
Totale 8.958
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Città #
Ann Arbor 1.456
Chandler 527
Woodbridge 503
Jacksonville 421
Houston 418
Princeton 384
Wilmington 311
Singapore 183
Dong Ket 177
Ashburn 169
Salerno 167
Izmir 160
Dublin 128
Beijing 119
Nanjing 82
Andover 78
Boardman 78
Munich 77
Hong Kong 73
Moscow 52
Pellezzano 51
Dearborn 41
Fairfield 40
The Dalles 36
Columbus 34
Hebei 34
Los Angeles 28
Shenyang 25
Turku 23
Mestre 21
Nanchang 20
Pune 20
São Paulo 20
Dallas 18
Philadelphia 17
Rome 17
Changsha 16
Fisciano 16
Norwalk 16
Council Bluffs 15
Jiaxing 15
New York 15
Redwood City 15
Düsseldorf 13
Falls Church 13
Guangzhou 12
Nuremberg 12
Tianjin 12
Washington 12
Brno 11
Seattle 11
Cambridge 9
San Francisco 9
Shanghai 9
Brooklyn 7
Jinan 7
London 7
Napoli 7
San Diego 7
Warsaw 7
Belo Horizonte 6
Boston 6
Chicago 6
Helsinki 6
Indiana 6
Joinville 6
Munro 6
Renton 6
Santa Clara 6
Tappahannock 6
Vienna 6
Campinas 5
Florence 5
Manchester 5
Mexico City 5
Palermo 5
Rio de Janeiro 5
Sarno 5
Sorrento 5
Spinea 5
Stockholm 5
Atlanta 4
Edinburgh 4
Johannesburg 4
Menlo Park 4
Montreal 4
Naples 4
Olomouc 4
Tashkent 4
Amman 3
Cagliari 3
Casoria 3
Catania 3
Clifton 3
Durham 3
Fortaleza 3
Guarulhos 3
Hefei 3
Lahore 3
Lappeenranta 3
Totale 6.462
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Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 179
11C-ER176, a radioligand for 18-kDa translocator protein (TSPO), has adequate sensitivity to robustly image all three affinity genotypes in human brain 170
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 153
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 147
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 131
Unexpected fungicidal activity against Candida albicans of CPA18 and CPA109, novel azole compounds 130
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 130
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 129
Microbiologia Molecolare e Cellulare 127
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 124
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 124
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 124
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 124
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 123
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 119
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 119
Diversity through a branched reaction pathway: Generation of multicyclic scaffolds and identification of antimigratory agents 119
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 118
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 116
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 110
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 109
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 109
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 108
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 104
Azole antifungal agents related to naftifine and butenafine 103
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 103
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 101
Small-Molecule Inhibitors of Protein Geranylgeranyltransferase Type I 100
Chemical biology of Histone acetyltransferase natural compounds modulators. 100
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 100
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 97
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 96
Unprecedented synthesis of a novel amino quinone ring system via oxidative decarboxylation of quinone-based alpha,alpha-amino esters 95
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 94
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 94
Effects of azole treatments on the physical properties of Candida albicans plasma membrane: A spin probe EPR study 92
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 91
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 90
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 90
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 90
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 89
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 89
Interaction of Azole Compounds with DOPC and DOPC/Ergosterol Bilayers by Spin Probe EPR Spectroscopy: Implications for Antifungal Activity 88
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 88
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 88
Antimycobacterial activity of ionic fullerene derivatives. 87
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 87
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 87
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 86
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 85
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 84
Luminometric sub-nanoliter droplet-to-droplet array (LUMDA) and its application to drug screening by phase I metabolism enzymes 84
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 84
A chemoenzymatic approach to the synthesis of the stereoisomers of a b-adrenergic receptor antagonist. 83
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 82
Synthesis of 11-aryl-5H-imidazo[2,1-c][1,4]benzodiazepines and their benzodiazepine and A1 adenosine binding activity. 79
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 79
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 78
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 77
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 77
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 77
A new class of antifungal agents. Synthesis and antimycotic activity of disubstituted N-azolylamines. 76
The emerging role of lysine methyltransferase SETD8 in human diseases 76
N-Pyrrylarylsulfones with High Therapeutic Potential 76
New structural analogues of tubulozole induce apoptosis, [Ca2+]i modifications and cytoskeletal disorganization in glial (GL15) and neuronal-like (PC12) cell lines. 75
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 75
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 75
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 75
5-Aryl-imidazo[2,1-c][1,4]benzodiazepine derivatives as tricyclic constrained analogues of diazepam and Ro5-4864. Synthesis and binding properties at peripheral and central benzodiazepine receptors. 73
Synthesis and antimicrobial properties of 3-aryl-1-(1,1'-biphenyl-4-yl)-2-(1H-imidazol-1-yl)propanes as 'carba-analogues' of the N-arylmethyl-N-[(1,1'-biphenyl)-4-ylmethyl])-1H-imidazol-1-amines, a new class of antifungal agents. 72
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 72
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 72
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 70
TRANSLOCATOR PROTEIN IMAGING AGENTS; METHODS OF MANUFACTURE, AND METHODS OF USE THEREOF 69
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 69
Enhancement of lysine acetylation accelerates wound repair 68
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 68
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 67
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 67
Synthesis of tricyclic triazepinones related to nevirapine. 65
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 65
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 64
Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20. 63
Synthesis and pharmacological characterization of new analogs of broxaterol. 62
Lysine methyltransferase inhibitors: where we are now. 62
Design and Synthesis of Novel [60]Fullerene Derivatives as Potential HIV Aspartic Protease Inhibitors. 60
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 60
Discovery of new chemical probes for the MRG15 chromo domain. 59
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 58
Synthesis and antifungal properties of N-[(1,1'-biphenyl)-4-ylmethyl]-1H-imidazol-1-amine derivatives. 57
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 56
Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain 56
Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 56
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 53
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 51
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 51
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 51
DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 44
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 44
Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging 42
Totale 8.814
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Categoria #
all - tutte 33.438
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 33.438
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021785 5 71 88 4 81 36 79 15 96 6 82 222
2021/2022737 6 5 4 7 23 27 11 30 93 108 107 316
2022/20231.192 117 106 27 159 141 240 12 123 182 5 59 21
2023/2024540 41 67 38 14 39 94 28 40 5 23 24 127
2024/20251.701 66 25 31 69 121 171 263 148 280 78 249 200
2025/2026128 128 0 0 0 0 0 0 0 0 0 0 0
Totale 9.250