UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
NA - Nord America 2.633
EU - Europa 827
AS - Asia 672
SA - Sud America 194
AF - Africa 15
Continente sconosciuto - Info sul continente non disponibili 2
OC - Oceania 1
Totale 4.344
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Nazione #
US - Stati Uniti d'America 2.617
SG - Singapore 296
IT - Italia 270
RU - Federazione Russa 186
CN - Cina 184
BR - Brasile 178
UA - Ucraina 115
TR - Turchia 78
IE - Irlanda 69
DE - Germania 58
SE - Svezia 45
VN - Vietnam 40
FI - Finlandia 27
KR - Corea 24
IN - India 18
FR - Francia 13
GB - Regno Unito 12
HK - Hong Kong 10
AT - Austria 9
CZ - Repubblica Ceca 8
AR - Argentina 7
IQ - Iraq 5
MA - Marocco 5
NL - Olanda 5
PK - Pakistan 5
CA - Canada 4
MX - Messico 4
ZA - Sudafrica 4
GR - Grecia 3
PA - Panama 3
VE - Venezuela 3
CO - Colombia 2
EU - Europa 2
JO - Giordania 2
NI - Nicaragua 2
PL - Polonia 2
TN - Tunisia 2
UZ - Uzbekistan 2
AL - Albania 1
AZ - Azerbaigian 1
BD - Bangladesh 1
BE - Belgio 1
BZ - Belize 1
CG - Congo 1
CL - Cile 1
DZ - Algeria 1
EC - Ecuador 1
GH - Ghana 1
GT - Guatemala 1
KH - Cambogia 1
LU - Lussemburgo 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PE - Perù 1
PH - Filippine 1
PS - Palestinian Territory 1
PY - Paraguay 1
RS - Serbia 1
SA - Arabia Saudita 1
SN - Senegal 1
SY - Repubblica araba siriana 1
TH - Thailandia 1
TT - Trinidad e Tobago 1
Totale 4.344
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Città #
Ann Arbor 707
Chandler 314
Woodbridge 265
Princeton 187
Houston 179
Jacksonville 173
Wilmington 132
Ashburn 99
Singapore 92
Salerno 90
Izmir 73
Dublin 66
Beijing 53
Boardman 42
Dearborn 40
Andover 38
Dong Ket 38
Nanjing 33
Moscow 25
Fairfield 20
Pellezzano 19
São Paulo 17
Shenyang 15
Hebei 14
Fisciano 13
Philadelphia 13
Council Bluffs 12
Pune 12
Rome 12
Changsha 11
Dallas 11
Redwood City 11
Norwalk 10
Brno 8
Hong Kong 8
Nanchang 8
Munich 7
New York 7
San Diego 7
Düsseldorf 6
Falls Church 6
Los Angeles 6
Munro 6
Nuremberg 6
Seattle 6
Washington 6
Cambridge 5
Florence 5
Helsinki 5
Jiaxing 5
Napoli 5
Palermo 5
Shanghai 5
Sorrento 5
The Dalles 5
Campagna 4
Joinville 4
Menlo Park 4
Mestre 4
Naples 4
Vienna 4
Campinas 3
Casoria 3
Catania 3
Guangzhou 3
Hefei 3
Jinan 3
Lahore 3
Messina 3
Mugnano del Cardinale 3
Newcastle upon Tyne 3
Néa Smýrni 3
Panama City 3
Rio de Janeiro 3
Tianjin 3
Amman 2
Aparecida de Goiânia 2
Belo Horizonte 2
Bisamberg 2
Bragança Paulista 2
Brasília 2
Caivano 2
Calvisano 2
Chicago 2
Conselheiro Lafaiete 2
Domicella 2
Duque de Caxias 2
Edinburgh 2
Embu das Artes 2
Goiânia 2
Guaratinguetá 2
Hangzhou 2
Hanover 2
Ho Chi Minh City 2
Indiana 2
Ipatinga 2
Jacareí 2
Johannesburg 2
Kolkata 2
Lappeenranta 2
Totale 3.084
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Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 166
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 146
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 135
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 123
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 120
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 118
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 117
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 115
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 115
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 114
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 108
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 108
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 105
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 104
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 99
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 99
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 96
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 95
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 95
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 94
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 94
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 91
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 86
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 85
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 82
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 82
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 79
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 77
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 76
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 76
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 75
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 72
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 72
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 71
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 70
The emerging role of lysine methyltransferase SETD8 in human diseases 69
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 69
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 63
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 60
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 60
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 59
Lysine methyltransferase inhibitors: where we are now. 56
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 54
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 54
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 54
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 44
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 44
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 43
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 39
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 38
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 32
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 31
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 31
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 28
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 26
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 21
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 21
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity 19
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory 15
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 13
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 12
Totale 4.515
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Categoria #
all - tutte 16.118
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 16.118
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/202075 0 0 0 0 0 0 0 0 0 0 71 4
2020/2021332 1 29 41 2 31 23 31 10 55 6 38 65
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024309 16 35 26 11 17 58 15 12 1 19 12 87
2024/2025866 21 22 22 64 109 111 192 90 166 69 0 0
Totale 4.515