UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
NA - Nord America 2.536
EU - Europa 562
AS - Asia 287
SA - Sud America 7
Continente sconosciuto - Info sul continente non disponibili 2
AF - Africa 1
OC - Oceania 1
Totale 3.396
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Nazione #
US - Stati Uniti d'America 2.528
IT - Italia 230
CN - Cina 158
UA - Ucraina 114
TR - Turchia 73
IE - Irlanda 69
DE - Germania 47
SE - Svezia 45
VN - Vietnam 38
FI - Finlandia 21
FR - Francia 13
IN - India 10
GB - Regno Unito 9
AR - Argentina 6
RU - Federazione Russa 5
AT - Austria 3
PA - Panama 3
CA - Canada 2
EU - Europa 2
HK - Hong Kong 2
BE - Belgio 1
BZ - Belize 1
CL - Cile 1
GH - Ghana 1
KH - Cambogia 1
KR - Corea 1
LU - Lussemburgo 1
MX - Messico 1
NL - Olanda 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PH - Filippine 1
PK - Pakistan 1
PL - Polonia 1
RS - Serbia 1
SA - Arabia Saudita 1
SG - Singapore 1
TT - Trinidad e Tobago 1
Totale 3.396
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Città #
Ann Arbor 707
Chandler 314
Woodbridge 265
Princeton 187
Houston 179
Jacksonville 173
Wilmington 132
Salerno 90
Izmir 73
Ashburn 67
Dublin 66
Beijing 53
Boardman 42
Dearborn 40
Andover 38
Dong Ket 38
Nanjing 33
Fairfield 20
Pellezzano 19
Shenyang 15
Hebei 14
Philadelphia 13
Changsha 11
Redwood City 11
Norwalk 10
Rome 10
Nanchang 8
Pune 8
Fisciano 7
San Diego 7
Düsseldorf 6
Falls Church 6
Los Angeles 6
Munro 6
Seattle 6
Washington 6
Cambridge 5
Florence 5
Jiaxing 5
Napoli 5
Palermo 5
Sorrento 5
Menlo Park 4
Mestre 4
Casoria 3
Catania 3
Jinan 3
Messina 3
Mugnano del Cardinale 3
Panama City 3
Tianjin 3
Vienna 3
Calvisano 2
Chicago 2
Edinburgh 2
Hangzhou 2
Hanover 2
Hefei 2
Hong Kong 2
Indiana 2
London 2
Maddaloni 2
Mercato San Severino 2
Munich 2
New York 2
Nocera Superiore 2
Nürnberg 2
Orange 2
Pescara 2
Spinea 2
Tappahannock 2
Yekaterinburg 2
Alexandria 1
Atlanta 1
Auckland 1
Bari 1
Belgrade 1
Belize City 1
Benevento 1
Brussels 1
Böblingen 1
Cagliari 1
Caserta 1
Castel Volturno 1
Chatham 1
Chengdu 1
Chongqing 1
Como 1
Contrada 1
Denver 1
Grammichele 1
Groningen 1
Guangzhou 1
Honolulu 1
Juarez 1
Kamampa 1
Lappeenranta 1
Laurel 1
Mainz 1
Marcianise 1
Totale 2.816
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Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 144
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 117
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 116
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 105
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 102
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 101
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 100
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 95
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 94
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 93
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 92
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 91
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 91
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 89
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 89
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 87
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 87
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 84
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 81
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 81
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 79
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 75
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 71
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 68
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 62
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 61
The emerging role of lysine methyltransferase SETD8 in human diseases 60
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 57
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 56
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 56
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 55
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 55
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 54
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 53
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 52
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 50
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 50
Lysine methyltransferase inhibitors: where we are now. 50
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 46
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 46
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 44
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 40
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 39
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 38
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 37
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 35
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 33
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 32
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 30
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 27
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 25
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 22
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 20
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 20
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 7
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 5
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 1
Totale 3.550
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Categoria #
all - tutte 9.791
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 9.791
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019143 0 0 0 0 0 0 0 0 0 0 136 7
2019/2020371 101 7 30 9 28 19 30 6 35 31 71 4
2020/2021332 1 29 41 2 31 23 31 10 55 6 38 65
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024210 16 35 26 11 17 58 15 12 1 19 0 0
Totale 3.550