UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
NA - Nord America 2.756
EU - Europa 911
AS - Asia 776
SA - Sud America 232
AF - Africa 19
Continente sconosciuto - Info sul continente non disponibili 2
OC - Oceania 1
Totale 4.697
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Nazione #
US - Stati Uniti d'America 2.729
SG - Singapore 305
IT - Italia 273
BR - Brasile 214
CN - Cina 205
RU - Federazione Russa 189
UA - Ucraina 115
DE - Germania 102
TR - Turchia 79
IE - Irlanda 69
FI - Finlandia 48
HK - Hong Kong 46
SE - Svezia 46
KR - Corea 45
VN - Vietnam 42
IN - India 22
GB - Regno Unito 15
FR - Francia 14
CA - Canada 10
CZ - Repubblica Ceca 10
AT - Austria 9
MX - Messico 9
AR - Argentina 7
IQ - Iraq 7
PK - Pakistan 7
NL - Olanda 6
BD - Bangladesh 5
MA - Marocco 5
ZA - Sudafrica 5
PL - Polonia 4
CO - Colombia 3
DZ - Algeria 3
ES - Italia 3
GR - Grecia 3
PA - Panama 3
VE - Venezuela 3
CL - Cile 2
EU - Europa 2
JO - Giordania 2
NI - Nicaragua 2
PS - Palestinian Territory 2
TN - Tunisia 2
UZ - Uzbekistan 2
AL - Albania 1
AZ - Azerbaigian 1
BE - Belgio 1
BZ - Belize 1
CG - Congo 1
EC - Ecuador 1
GH - Ghana 1
GT - Guatemala 1
IL - Israele 1
KE - Kenya 1
KH - Cambogia 1
LU - Lussemburgo 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PE - Perù 1
PH - Filippine 1
PY - Paraguay 1
RS - Serbia 1
SA - Arabia Saudita 1
SN - Senegal 1
SY - Repubblica araba siriana 1
TH - Thailandia 1
TT - Trinidad e Tobago 1
Totale 4.697
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Città #
Ann Arbor 707
Chandler 314
Woodbridge 265
Princeton 187
Houston 179
Jacksonville 174
Wilmington 133
Ashburn 104
Singapore 100
Salerno 90
Beijing 73
Izmir 73
Dublin 66
Munich 48
Hong Kong 44
Boardman 42
Dearborn 40
Andover 38
Dong Ket 38
Nanjing 33
Columbus 25
Moscow 25
The Dalles 21
Turku 21
Fairfield 20
Pellezzano 19
São Paulo 18
Dallas 16
Shenyang 15
Hebei 14
Fisciano 13
Philadelphia 13
Council Bluffs 12
Pune 12
Rome 12
Changsha 11
Los Angeles 11
Redwood City 11
Norwalk 10
Nuremberg 9
Brno 8
Nanchang 8
New York 7
San Diego 7
Seattle 7
Düsseldorf 6
Falls Church 6
Munro 6
San Francisco 6
Washington 6
Belo Horizonte 5
Cambridge 5
Chicago 5
Florence 5
Helsinki 5
Jiaxing 5
Joinville 5
Mexico City 5
Naples 5
Napoli 5
Palermo 5
Rio de Janeiro 5
Shanghai 5
Sorrento 5
Campagna 4
Lahore 4
Menlo Park 4
Mestre 4
Santa Clara 4
Vienna 4
Warsaw 4
Campinas 3
Casoria 3
Catania 3
Guangzhou 3
Hefei 3
Jinan 3
Johannesburg 3
London 3
Messina 3
Montreal 3
Mugnano del Cardinale 3
Newcastle upon Tyne 3
Néa Smýrni 3
Panama City 3
Tianjin 3
Amman 2
Amsterdam 2
Aparecida de Goiânia 2
Baghdad 2
Bisamberg 2
Bom Despacho 2
Boston 2
Bragança Paulista 2
Brasília 2
Brooklyn 2
Buffalo 2
Caivano 2
Calvisano 2
Chennai 2
Totale 3.294
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Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 177
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 152
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 145
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 128
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 124
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 124
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 123
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 123
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 119
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 119
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 117
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 111
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 109
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 109
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 109
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 107
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 104
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 102
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 99
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 97
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 97
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 96
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 90
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 89
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 89
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 89
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 88
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 87
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 87
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 86
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 82
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 81
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 76
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 76
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 75
The emerging role of lysine methyltransferase SETD8 in human diseases 74
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 72
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 68
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 67
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 65
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 64
Lysine methyltransferase inhibitors: where we are now. 61
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 60
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 58
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 58
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 51
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 51
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 50
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 50
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 44
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 37
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 35
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 32
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 31
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 29
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 28
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity 25
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 23
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory 18
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 16
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 16
Totale 4.869
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Categoria #
all - tutte 17.443
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 17.443
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021332 1 29 41 2 31 23 31 10 55 6 38 65
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024309 16 35 26 11 17 58 15 12 1 19 12 87
2024/20251.160 21 22 22 64 109 111 192 90 166 69 155 139
2025/202660 60 0 0 0 0 0 0 0 0 0 0 0
Totale 4.869