UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
AS - Asia 6.190
NA - Nord America 4.223
EU - Europa 1.543
SA - Sud America 411
Continente sconosciuto - Info sul continente non disponibili 191
AF - Africa 52
OC - Oceania 1
Totale 12.611
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Nazione #
HK - Hong Kong 4.446
US - Stati Uniti d'America 4.120
SG - Singapore 817
IT - Italia 697
CN - Cina 350
BR - Brasile 324
RU - Federazione Russa 197
VN - Vietnam 193
DE - Germania 132
UA - Ucraina 120
TR - Turchia 93
IN - India 74
IE - Irlanda 71
FR - Francia 69
FI - Finlandia 59
KR - Corea 55
SE - Svezia 52
GB - Regno Unito 48
BD - Bangladesh 45
CA - Canada 38
AR - Argentina 34
MX - Messico 32
JP - Giappone 24
IQ - Iraq 21
PL - Polonia 19
ES - Italia 15
VE - Venezuela 15
NL - Olanda 13
PK - Pakistan 13
ZA - Sudafrica 13
JM - Giamaica 12
AT - Austria 11
ID - Indonesia 11
CO - Colombia 10
CZ - Repubblica Ceca 10
MA - Marocco 9
CL - Cile 8
EC - Ecuador 8
UZ - Uzbekistan 7
DZ - Algeria 6
GR - Grecia 6
AL - Albania 5
MY - Malesia 5
PA - Panama 5
PE - Perù 5
PH - Filippine 5
TN - Tunisia 5
LT - Lituania 4
RO - Romania 4
SA - Arabia Saudita 4
BO - Bolivia 3
CR - Costa Rica 3
ET - Etiopia 3
IL - Israele 3
JO - Giordania 3
KE - Kenya 3
PR - Porto Rico 3
PY - Paraguay 3
TH - Thailandia 3
TT - Trinidad e Tobago 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
BG - Bulgaria 2
EG - Egitto 2
EU - Europa 2
LB - Libano 2
LU - Lussemburgo 2
LY - Libia 2
NI - Nicaragua 2
NP - Nepal 2
OM - Oman 2
PS - Palestinian Territory 2
PT - Portogallo 2
SN - Senegal 2
AO - Angola 1
BB - Barbados 1
BE - Belgio 1
BZ - Belize 1
CG - Congo 1
CI - Costa d'Avorio 1
EE - Estonia 1
GE - Georgia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
HN - Honduras 1
KH - Cambogia 1
LV - Lettonia 1
MN - Mongolia 1
MV - Maldive 1
MZ - Mozambico 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
QA - Qatar 1
RS - Serbia 1
SV - El Salvador 1
SY - Repubblica araba siriana 1
TZ - Tanzania 1
UY - Uruguay 1
Totale 12.422
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Città #
Hong Kong 4.434
Ann Arbor 707
Singapore 403
San Jose 353
Dallas 323
Chandler 314
Woodbridge 265
Ashburn 235
Milan 213
Princeton 187
Houston 186
Jacksonville 174
Wilmington 133
Beijing 119
Salerno 115
Council Bluffs 84
Izmir 73
The Dalles 71
Dublin 68
Munich 64
Ho Chi Minh City 59
Rome 55
Lauterbourg 51
Santa Clara 51
Boardman 43
Dearborn 40
Andover 38
Dong Ket 38
Los Angeles 37
New York 35
Nanjing 33
São Paulo 32
Hanoi 30
Columbus 27
Moscow 26
Tokyo 24
Turku 23
Orem 21
Fairfield 20
Figino 19
Naples 19
Pellezzano 19
Fisciano 18
Chicago 17
Warsaw 17
Philadelphia 15
Shenyang 15
Basingstoke 14
Hebei 14
Montreal 14
Pune 14
Brooklyn 13
Helsinki 13
Mexico City 13
Memphis 12
Rio de Janeiro 12
Changsha 11
Redwood City 11
San Francisco 11
Belo Horizonte 10
Norwalk 10
Nuremberg 10
Atlanta 9
Denver 9
Frankfurt am Main 9
Baghdad 8
Baronissi 8
Brno 8
Buffalo 8
Chennai 8
Hải Dương 8
Nanchang 8
San Diego 8
Seattle 8
Seoul 8
Stockholm 8
Turin 8
Amsterdam 7
Caserta 7
Florence 7
Haiphong 7
Johannesburg 7
Shanghai 7
Tashkent 7
Washington 7
Ankara 6
Boston 6
Charlotte 6
Düsseldorf 6
Falls Church 6
Joinville 6
Kingston 6
London 6
Munro 6
Palermo 6
Phoenix 6
Scafati 6
Cambridge 5
Catania 5
Da Nang 5
Totale 9.791
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.249
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 723
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 690
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 533
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 443
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 386
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 379
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 271
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 259
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 254
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 243
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 242
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 229
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 203
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 199
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 193
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 183
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 178
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 175
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 171
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 166
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 164
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 163
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 162
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 159
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 158
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 156
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 156
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 155
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 151
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 150
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 149
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 149
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 144
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 143
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 138
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 136
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 133
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 131
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 131
The emerging role of lysine methyltransferase SETD8 in human diseases 129
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 127
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 126
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 126
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 126
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 124
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 120
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 120
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 114
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 113
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 112
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 110
Lysine methyltransferase inhibitors: where we are now. 110
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 99
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity 91
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 87
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 71
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory 69
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 67
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 65
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 64
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 58
Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5′-Terminal Oligopyrimidine Motif-Containing mRNA 56
Coactivator-associated arginine methyltransferase 1 (CARM1) inhibitors: a patenting perspective (2018-present) 40
2‐Phenylquinolines Exhibit Anti‐Severe Acute Respiratory Syndrome Coronavirus‐2 Activity Through the Nonstructural Protein 13 Helicase Inhibition 32
Identification of 2‐Substituted‐3‐Hydroxy‐2,3‐Dihydroquinazolin‐4(1 H ) Ones as Cell‐Active Inhibitors of KDM4A Lysine Demethylase 30
Design, synthesis and biological evaluation of new small molecule modulators of Arginine methyltransferases 20
Targeting Copper in Cancer: Chelators to Counteract Cuproplasia and Ionophores to Promote Cuproptosis 4
Discovery of High-Affinity Peptide Ligands Targeting the SPIN1 Tudor 3 Domain Via a Minimalist Pruning Strategy 3
Targeting PRMTs with Small-Molecule Inhibitors: A Comprehensive Review 1
Totale 12.611
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Categoria #
all - tutte 33.014
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 33.014
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024309 16 35 26 11 17 58 15 12 1 19 12 87
2024/20251.160 21 22 22 64 109 111 192 90 166 69 155 139
2025/20267.558 988 2.169 1.831 240 403 187 483 109 281 361 117 389
2026/2027244 170 74 0 0 0 0 0 0 0 0 0 0
Totale 12.611