UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
AS - Asia 6.154
NA - Nord America 4.060
EU - Europa 1.180
SA - Sud America 404
AF - Africa 52
Continente sconosciuto - Info sul continente non disponibili 2
OC - Oceania 1
Totale 11.853
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Nazione #
HK - Hong Kong 4.433
US - Stati Uniti d'America 3.983
SG - Singapore 809
IT - Italia 341
CN - Cina 339
BR - Brasile 319
RU - Federazione Russa 197
VN - Vietnam 192
DE - Germania 132
UA - Ucraina 120
TR - Turchia 93
IN - India 73
IE - Irlanda 71
FR - Francia 69
FI - Finlandia 59
KR - Corea 55
SE - Svezia 50
GB - Regno Unito 47
BD - Bangladesh 45
AR - Argentina 34
CA - Canada 31
MX - Messico 30
JP - Giappone 24
IQ - Iraq 21
PL - Polonia 18
ES - Italia 14
VE - Venezuela 14
PK - Pakistan 13
ZA - Sudafrica 13
NL - Olanda 12
AT - Austria 11
ID - Indonesia 11
CO - Colombia 10
CZ - Repubblica Ceca 10
MA - Marocco 9
CL - Cile 8
EC - Ecuador 7
UZ - Uzbekistan 7
DZ - Algeria 6
GR - Grecia 6
AL - Albania 5
MY - Malesia 5
PA - Panama 5
PE - Perù 5
PH - Filippine 5
TN - Tunisia 5
JM - Giamaica 4
LT - Lituania 4
RO - Romania 4
BO - Bolivia 3
ET - Etiopia 3
JO - Giordania 3
KE - Kenya 3
PY - Paraguay 3
SA - Arabia Saudita 3
TH - Thailandia 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
BG - Bulgaria 2
EG - Egitto 2
EU - Europa 2
IL - Israele 2
LB - Libano 2
LU - Lussemburgo 2
LY - Libia 2
NI - Nicaragua 2
NP - Nepal 2
OM - Oman 2
PS - Palestinian Territory 2
SN - Senegal 2
TT - Trinidad e Tobago 2
AO - Angola 1
BE - Belgio 1
BZ - Belize 1
CG - Congo 1
CI - Costa d'Avorio 1
EE - Estonia 1
GE - Georgia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
HN - Honduras 1
KH - Cambogia 1
LV - Lettonia 1
MN - Mongolia 1
MV - Maldive 1
MZ - Mozambico 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PT - Portogallo 1
QA - Qatar 1
RS - Serbia 1
SY - Repubblica araba siriana 1
TZ - Tanzania 1
UY - Uruguay 1
Totale 11.853
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Città #
Hong Kong 4.421
Ann Arbor 707
Singapore 395
San Jose 353
Dallas 320
Chandler 314
Woodbridge 265
Ashburn 226
Princeton 187
Houston 186
Jacksonville 174
Wilmington 133
Beijing 108
Salerno 90
Council Bluffs 73
Izmir 73
The Dalles 71
Dublin 68
Munich 64
Ho Chi Minh City 59
Lauterbourg 51
Boardman 43
Dearborn 40
Andover 38
Dong Ket 38
Santa Clara 37
Los Angeles 35
Nanjing 33
New York 33
São Paulo 32
Hanoi 30
Columbus 26
Moscow 26
Tokyo 24
Turku 23
Fairfield 20
Orem 20
Pellezzano 19
Fisciano 18
Naples 16
Warsaw 16
Shenyang 15
Basingstoke 14
Chicago 14
Hebei 14
Pune 14
Rome 14
Helsinki 13
Montreal 13
Philadelphia 13
Memphis 12
Rio de Janeiro 12
Brooklyn 11
Changsha 11
Mexico City 11
Redwood City 11
Belo Horizonte 10
Norwalk 10
Nuremberg 10
Atlanta 9
Denver 9
Frankfurt am Main 9
Baghdad 8
Baronissi 8
Brno 8
Chennai 8
Hải Dương 8
Nanchang 8
San Diego 8
San Francisco 8
Seoul 8
Amsterdam 7
Buffalo 7
Haiphong 7
Johannesburg 7
Seattle 7
Shanghai 7
Tashkent 7
Washington 7
Ankara 6
Boston 6
Caserta 6
Düsseldorf 6
Falls Church 6
Florence 6
Joinville 6
London 6
Munro 6
Phoenix 6
Scafati 6
Stockholm 6
Cambridge 5
Catania 5
Da Nang 5
Jakarta 5
Jiaxing 5
Lahore 5
Napoli 5
Palermo 5
Pilāni 5
Totale 9.399
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.242
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 712
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 686
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 525
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 435
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 383
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 374
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 262
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 246
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 245
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 238
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 232
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 223
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 197
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 191
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 186
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 177
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 169
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 163
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 162
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 159
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 157
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 157
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 153
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 150
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 150
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 149
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 147
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 146
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 145
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 143
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 142
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 140
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 138
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 130
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 128
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 127
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 127
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 126
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 124
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 123
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 123
The emerging role of lysine methyltransferase SETD8 in human diseases 121
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 120
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 118
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 118
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 113
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 111
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 110
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 108
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 106
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 104
Lysine methyltransferase inhibitors: where we are now. 98
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 90
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity 80
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 75
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 65
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 64
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory 61
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 56
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 54
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 49
Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5′-Terminal Oligopyrimidine Motif-Containing mRNA 31
Coactivator-associated arginine methyltransferase 1 (CARM1) inhibitors: a patenting perspective (2018-present) 30
2‐Phenylquinolines Exhibit Anti‐Severe Acute Respiratory Syndrome Coronavirus‐2 Activity Through the Nonstructural Protein 13 Helicase Inhibition 12
Design, synthesis and biological evaluation of new small molecule modulators of Arginine methyltransferases 9
Identification of 2‐Substituted‐3‐Hydroxy‐2,3‐Dihydroquinazolin‐4(1 H ) Ones as Cell‐Active Inhibitors of KDM4A Lysine Demethylase 4
Totale 12.039
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Categoria #
all - tutte 30.944
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 30.944
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/202165 0 0 0 0 0 0 0 0 0 0 0 65
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024309 16 35 26 11 17 58 15 12 1 19 12 87
2024/20251.160 21 22 22 64 109 111 192 90 166 69 155 139
2025/20267.230 988 2.169 1.831 240 403 187 483 109 281 361 117 61
Totale 12.039