UniSa - IRIS Institutional Research Information System

MILITE, Ciro
 Distribuzione geografica
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Continente #
AS - Asia 6.108
NA - Nord America 3.917
EU - Europa 1.165
SA - Sud America 402
AF - Africa 52
Continente sconosciuto - Info sul continente non disponibili 2
OC - Oceania 1
Totale 11.647
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Nazione #
HK - Hong Kong 4.426
US - Stati Uniti d'America 3.850
SG - Singapore 804
CN - Cina 330
IT - Italia 328
BR - Brasile 318
RU - Federazione Russa 197
VN - Vietnam 192
DE - Germania 132
UA - Ucraina 120
TR - Turchia 93
IE - Irlanda 71
FR - Francia 69
IN - India 69
FI - Finlandia 59
KR - Corea 55
SE - Svezia 50
GB - Regno Unito 46
AR - Argentina 34
MX - Messico 29
BD - Bangladesh 25
CA - Canada 25
JP - Giappone 24
IQ - Iraq 21
PL - Polonia 18
ES - Italia 14
PK - Pakistan 13
VE - Venezuela 13
ZA - Sudafrica 13
NL - Olanda 12
AT - Austria 11
ID - Indonesia 11
CO - Colombia 10
CZ - Repubblica Ceca 10
MA - Marocco 9
CL - Cile 8
EC - Ecuador 7
UZ - Uzbekistan 7
DZ - Algeria 6
GR - Grecia 6
AL - Albania 5
PA - Panama 5
PE - Perù 5
PH - Filippine 5
TN - Tunisia 5
LT - Lituania 4
MY - Malesia 4
BO - Bolivia 3
ET - Etiopia 3
JO - Giordania 3
KE - Kenya 3
PY - Paraguay 3
RO - Romania 3
SA - Arabia Saudita 3
TH - Thailandia 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
BG - Bulgaria 2
EG - Egitto 2
EU - Europa 2
IL - Israele 2
JM - Giamaica 2
LB - Libano 2
LU - Lussemburgo 2
LY - Libia 2
NI - Nicaragua 2
NP - Nepal 2
OM - Oman 2
PS - Palestinian Territory 2
SN - Senegal 2
AO - Angola 1
BE - Belgio 1
BZ - Belize 1
CG - Congo 1
CI - Costa d'Avorio 1
EE - Estonia 1
GE - Georgia 1
GH - Ghana 1
GN - Guinea 1
GT - Guatemala 1
HN - Honduras 1
KH - Cambogia 1
LV - Lettonia 1
MN - Mongolia 1
MV - Maldive 1
MZ - Mozambico 1
NO - Norvegia 1
NZ - Nuova Zelanda 1
PT - Portogallo 1
QA - Qatar 1
RS - Serbia 1
SY - Repubblica araba siriana 1
TT - Trinidad e Tobago 1
TZ - Tanzania 1
UY - Uruguay 1
Totale 11.647
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Città #
Hong Kong 4.414
Ann Arbor 707
Singapore 393
San Jose 320
Dallas 318
Chandler 314
Woodbridge 265
Ashburn 222
Princeton 187
Houston 186
Jacksonville 174
Wilmington 133
Beijing 104
Salerno 90
Council Bluffs 73
Izmir 73
The Dalles 71
Dublin 68
Munich 64
Ho Chi Minh City 59
Lauterbourg 51
Boardman 43
Dearborn 40
Andover 38
Dong Ket 38
Los Angeles 34
Nanjing 33
São Paulo 32
Hanoi 30
Santa Clara 30
New York 29
Columbus 26
Moscow 26
Tokyo 24
Turku 23
Fairfield 20
Orem 20
Pellezzano 19
Fisciano 18
Naples 16
Warsaw 16
Shenyang 15
Basingstoke 14
Hebei 14
Pune 14
Chicago 13
Helsinki 13
Montreal 13
Philadelphia 13
Rome 13
Rio de Janeiro 12
Changsha 11
Redwood City 11
Belo Horizonte 10
Mexico City 10
Norwalk 10
Nuremberg 10
Denver 9
Frankfurt am Main 9
Baghdad 8
Baronissi 8
Brno 8
Brooklyn 8
Chennai 8
Hải Dương 8
Nanchang 8
San Francisco 8
Seoul 8
Amsterdam 7
Atlanta 7
Haiphong 7
Johannesburg 7
San Diego 7
Seattle 7
Shanghai 7
Tashkent 7
Washington 7
Ankara 6
Boston 6
Caserta 6
Düsseldorf 6
Falls Church 6
Joinville 6
London 6
Munro 6
Phoenix 6
Scafati 6
Stockholm 6
Cambridge 5
Da Nang 5
Florence 5
Jakarta 5
Jiaxing 5
Lahore 5
Napoli 5
Palermo 5
Pilāni 5
Poplar 5
Sorrento 5
Tirana 5
Totale 9.316
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.240
Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell lines 710
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 685
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 522
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 432
Nutraceutical properties and polyphenolic profile of berry skin and wine of Vitis vinifera L. (cv. Aglianico) 382
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 373
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 260
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 245
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 239
Design, Synthesis, and Evaluation of New Tripeptides as COX-2 Inhibitors 235
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 228
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 218
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 196
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 190
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 179
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 173
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 165
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 162
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 157
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 156
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 155
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 153
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 151
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 150
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 147
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 147
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 145
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 145
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 143
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 141
Identification of Limonol Derivatives as Heat Shock Protein 90 (Hsp90) Inhibitors through a Multidisciplinary Approach 140
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 137
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 136
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 127
Highly Enantioselective Organocatalytic α-Amination Reactions of Aryl Oxindoles: Developing Designer Multifunctional Alkaloid Catalysts 126
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 126
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 121
The emerging role of lysine methyltransferase SETD8 in human diseases 121
Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors 121
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery. 120
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 120
Identification of new KDM4 inhibitors through a HTS and hit refinement strategy 119
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 117
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach 116
IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY 115
Synthesis and evaluation of new TSPO PET radioligands with low sensitivity to human genotype 112
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) 110
Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice 106
From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases. 105
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors 104
Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells 101
Lysine methyltransferase inhibitors: where we are now. 95
The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells 89
Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies 73
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity 65
Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization 65
Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases 62
Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues 53
The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory 50
NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors 50
Patent evaluation of WO2019209182 (A1) 2019-10-31 (Conjugated Oligoelectrolytes as Antimicrobial Agents) 49
Coactivator-associated arginine methyltransferase 1 (CARM1) inhibitors: a patenting perspective (2018-present) 29
Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5′-Terminal Oligopyrimidine Motif-Containing mRNA 17
Design, synthesis and biological evaluation of new small molecule modulators of Arginine methyltransferases 6
2‐Phenylquinolines Exhibit Anti‐Severe Acute Respiratory Syndrome Coronavirus‐2 Activity Through the Nonstructural Protein 13 Helicase Inhibition 4
Totale 11.831
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Categoria #
all - tutte 29.667
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 29.667
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021109 0 0 0 0 0 0 0 0 0 6 38 65
2021/2022371 0 2 0 6 10 15 8 19 43 53 63 152
2022/2023673 57 67 18 90 73 142 11 63 108 4 31 9
2023/2024309 16 35 26 11 17 58 15 12 1 19 12 87
2024/20251.160 21 22 22 64 109 111 192 90 166 69 155 139
2025/20267.022 988 2.169 1.831 240 403 187 483 109 281 331 0 0
Totale 11.831