UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
NA - Nord America 8.155
EU - Europa 2.535
AS - Asia 2.061
SA - Sud America 476
AF - Africa 40
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
Totale 13.282
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Nazione #
US - Stati Uniti d'America 8.121
SG - Singapore 781
IT - Italia 754
CN - Cina 589
UA - Ucraina 472
BR - Brasile 443
RU - Federazione Russa 390
DE - Germania 285
TR - Turchia 207
IE - Irlanda 198
VN - Vietnam 172
FI - Finlandia 134
SE - Svezia 110
KR - Corea 101
HK - Hong Kong 80
IN - India 44
FR - Francia 38
GB - Regno Unito 36
AT - Austria 28
NL - Olanda 20
CZ - Repubblica Ceca 15
IQ - Iraq 15
PK - Pakistan 15
PL - Polonia 14
ZA - Sudafrica 14
BD - Bangladesh 13
CA - Canada 13
GR - Grecia 12
AR - Argentina 10
EU - Europa 10
UZ - Uzbekistan 9
ES - Italia 8
MA - Marocco 8
MX - Messico 8
IL - Israele 7
VE - Venezuela 6
CO - Colombia 5
DZ - Algeria 5
EC - Ecuador 5
AU - Australia 4
BG - Bulgaria 4
DO - Repubblica Dominicana 4
JP - Giappone 4
PE - Perù 4
CH - Svizzera 3
CL - Cile 3
JO - Giordania 3
KE - Kenya 3
RO - Romania 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
CR - Costa Rica 2
EG - Egitto 2
KH - Cambogia 2
LB - Libano 2
NO - Norvegia 2
NP - Nepal 2
PS - Palestinian Territory 2
RS - Serbia 2
SA - Arabia Saudita 2
TH - Thailandia 2
TT - Trinidad e Tobago 2
AL - Albania 1
BE - Belgio 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
DK - Danimarca 1
ET - Etiopia 1
GE - Georgia 1
GH - Ghana 1
GT - Guatemala 1
IR - Iran 1
JM - Giamaica 1
KZ - Kazakistan 1
LT - Lituania 1
LU - Lussemburgo 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
OM - Oman 1
PA - Panama 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
TW - Taiwan 1
Totale 13.282
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Città #
Ann Arbor 2.189
Chandler 842
Houston 707
Woodbridge 666
Jacksonville 633
Wilmington 627
Princeton 565
Singapore 269
Salerno 228
Ashburn 194
Izmir 194
Dublin 193
Dong Ket 161
Beijing 141
Nanjing 136
Andover 120
Boardman 119
Munich 101
Pellezzano 82
Hong Kong 78
Moscow 61
Mestre 59
The Dalles 58
Columbus 53
Fairfield 53
Shenyang 39
Dearborn 37
Hebei 35
São Paulo 33
Changsha 31
Turku 30
Los Angeles 29
Council Bluffs 27
Jiaxing 26
Norwalk 26
Nanchang 25
Redwood City 25
Fisciano 24
Nocera Superiore 24
Dallas 23
Düsseldorf 22
Falls Church 21
Pune 21
Tianjin 21
Rome 20
Naples 19
Nuremberg 19
Vienna 19
Washington 19
Philadelphia 17
New York 16
Guangzhou 15
Rio de Janeiro 14
Belo Horizonte 13
San Diego 13
Cambridge 11
Napoli 10
San Francisco 10
Athens 9
Brno 9
Brooklyn 9
Paris 9
Seattle 9
Amsterdam 8
Hefei 8
Kraków 8
London 8
Sarno 8
Tashkent 8
Boston 7
Brasília 7
Jinan 7
Shanghai 7
Zhengzhou 7
Bari 6
Catania 6
Chicago 6
Indiana 6
Johannesburg 6
Joinville 6
Milan 6
Montreal 6
Munro 6
Olomouc 6
Renton 6
Santa Clara 6
Warsaw 6
Ankara 5
Baghdad 5
Bologna 5
Cagliari 5
Campagna 5
Campinas 5
Dhaka 5
Florence 5
Guarulhos 5
Kolkata 5
Palermo 5
Recife 5
Sorrento 5
Totale 9.534
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Nome #
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 179
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 179
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 160
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 154
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 147
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 138
Agenti antimicotici, antimicobatterici e antiprotozoari 138
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 137
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 132
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 130
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 130
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 129
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 129
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 124
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 124
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 124
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 124
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 123
Arginine demethylation of G3BP1 promotes stress granule assembly 123
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 122
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 119
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 119
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 118
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 116
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 115
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 114
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 113
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 111
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 110
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 110
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 110
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 110
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 110
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 109
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 109
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 108
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 105
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 104
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 103
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 103
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 103
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 103
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 103
New 6-nitroquinolones: synthesis and antimicrobial activities 102
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 102
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 102
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 101
Chemical biology of Histone acetyltransferase natural compounds modulators. 101
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 101
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 100
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 100
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 98
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 97
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 97
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 97
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 97
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 96
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 96
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 96
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 96
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 95
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 94
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 94
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 94
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 93
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 91
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 90
DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors 90
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 90
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 89
Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian 89
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 89
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 89
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 88
The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) 88
SELECTIVE INHIBITORS FOR TRANSFERASES 87
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 87
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 86
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 86
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. 86
N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 85
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 85
Methods for inhibiting the transmission of HIV using topically applied substituted 6-​benzyl-​4-​oxopyrimidines 85
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 84
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 84
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family 83
6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase 82
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 82
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 80
A simplified synthesis of ethyl 5-chloro-6-fluoro-1H-indole-2-carboxylate and ethyl 5-chloro-4-fluoro-1H-indole-2-carboxylate 79
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 79
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 78
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 78
Chemioterapici antiprotozoari 78
A novel Gcn5p inhibitor represses cell growth, gene transcription and histone acetylation in budding yeast 77
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 77
ChemInform Abstract: A Simplified Synthesis of Ethyl 5-Chloro-4-fluoro-1H-indole-2-carboxylate and Ethyl 5-Chloro-6-fluoro-1H-indole-2-carboxylate 77
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 77
Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity 76
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 76
Totale 10.347
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Categoria #
all - tutte 46.045
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 46.045
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/20211.055 9 99 130 11 119 42 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024710 62 108 64 30 42 112 38 23 7 27 38 159
2024/20252.495 94 39 45 132 210 268 377 218 423 128 314 247
2025/2026203 203 0 0 0 0 0 0 0 0 0 0 0
Totale 13.767