UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
NA - Nord America 7.701
EU - Europa 1.819
AS - Asia 876
SA - Sud America 11
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
AF - Africa 2
Totale 10.424
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Nazione #
US - Stati Uniti d'America 7.694
IT - Italia 661
CN - Cina 481
UA - Ucraina 469
IE - Irlanda 198
TR - Turchia 194
DE - Germania 164
VN - Vietnam 163
SE - Svezia 109
FI - Finlandia 101
FR - Francia 25
GB - Regno Unito 21
IN - India 19
RU - Federazione Russa 17
AT - Austria 12
EU - Europa 10
NL - Olanda 9
PL - Polonia 9
AR - Argentina 6
GR - Grecia 5
IL - Israele 5
AU - Australia 4
BG - Bulgaria 4
KR - Corea 4
CH - Svizzera 3
JP - Giappone 3
MX - Messico 3
BR - Brasile 2
NO - Norvegia 2
RO - Romania 2
RS - Serbia 2
BE - Belgio 1
BZ - Belize 1
CA - Canada 1
CL - Cile 1
CO - Colombia 1
CR - Costa Rica 1
DK - Danimarca 1
EG - Egitto 1
ES - Italia 1
GH - Ghana 1
IR - Iran 1
KH - Cambogia 1
LU - Lussemburgo 1
NZ - Nuova Zelanda 1
PE - Perù 1
PK - Pakistan 1
PT - Portogallo 1
SA - Arabia Saudita 1
SG - Singapore 1
SK - Slovacchia (Repubblica Slovacca) 1
TH - Thailandia 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
Totale 10.424
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Città #
Ann Arbor 2.189
Chandler 842
Houston 706
Woodbridge 666
Jacksonville 631
Wilmington 626
Princeton 565
Salerno 226
Izmir 194
Dublin 193
Dong Ket 161
Ashburn 136
Nanjing 135
Andover 120
Beijing 119
Boardman 119
Pellezzano 82
Mestre 59
Fairfield 53
Shenyang 39
Dearborn 37
Hebei 35
Changsha 29
Norwalk 26
Nanchang 25
Redwood City 25
Nocera Superiore 24
Jiaxing 23
Düsseldorf 22
Falls Church 21
Tianjin 19
Rome 18
Washington 18
Philadelphia 17
Pune 17
San Diego 13
Fisciano 12
Vienna 12
Cambridge 11
Napoli 10
Guangzhou 9
Kraków 8
Seattle 8
Hefei 7
Jinan 7
Los Angeles 7
Catania 6
Indiana 6
Milan 6
Munro 6
New York 6
Renton 6
Zhengzhou 6
Athens 5
Bologna 5
Cagliari 5
Florence 5
London 5
Naples 5
Palermo 5
Sorrento 5
Tappahannock 5
Venezia 5
Amsterdam 4
Atlanta 4
Groningen 4
Spinea 4
Casoria 3
Hangzhou 3
Lappeenranta 3
Marcianise 3
Messina 3
Mugnano del Cardinale 3
Paris 3
Pavia 3
Altavilla Silentina 2
Bari 2
Calvisano 2
Caserta 2
Cattolica 2
Chicago 2
Chongqing 2
Cinisello Balsamo 2
Contrada 2
Durham 2
Edinburgh 2
Forlì 2
Frankfurt am Main 2
Hanover 2
Kunming 2
Maddaloni 2
Magdeburg 2
Manassas 2
Melbourne 2
Mexico City 2
Munich 2
Novi Sad 2
Orange 2
Perugia 2
Pescara 2
Totale 8.503
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Nome #
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 168
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 145
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 144
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 131
Agenti antimicotici, antimicobatterici e antiprotozoari 131
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 127
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 117
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 116
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 115
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 114
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 106
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 105
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 105
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 105
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 102
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 102
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 101
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 100
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 98
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 97
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 97
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 97
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 97
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 97
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 95
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 95
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 95
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 94
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 94
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 93
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 93
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 92
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 92
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 91
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 91
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 91
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 91
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 90
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 90
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 89
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 89
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 89
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 89
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 89
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 87
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 87
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 86
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 86
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 86
Arginine demethylation of G3BP1 promotes stress granule assembly 86
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 86
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 85
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 84
DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors 84
Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian 84
SELECTIVE INHIBITORS FOR TRANSFERASES 82
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 82
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 81
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 81
Chemical biology of Histone acetyltransferase natural compounds modulators. 80
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 80
The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) 80
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 79
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 79
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 78
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 77
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. 77
N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 76
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 76
Methods for inhibiting the transmission of HIV using topically applied substituted 6-​benzyl-​4-​oxopyrimidines 75
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 75
Chemioterapici antiprotozoari 73
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 71
ChemInform Abstract: A Simplified Synthesis of Ethyl 5-Chloro-4-fluoro-1H-indole-2-carboxylate and Ethyl 5-Chloro-6-fluoro-1H-indole-2-carboxylate 71
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 71
Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity 70
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 70
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 69
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 68
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 67
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 67
Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases 67
New 6-nitroquinolones: synthesis and antimicrobial activities 66
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 66
Does the 2-methylthiomethyl substituent really confer high anti-HIV-1 activity to S-DABOs ? 65
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties 65
Synthesis and Antiviral Activity of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs), New Potent and Selective HIV-1 Inhibitors. 65
ChemInform Abstract: N-[4-(1,1′-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as Non-oxazolidinone Analogues of Antimycobacterial U-100480 65
6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase 64
CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. 64
Anti-HIV-1 Activity of Arylthiazolylcarboxyamides, a novel class of NNRTIs as Hybrid Congeners between PETT, UC781 and TDA 63
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 63
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 62
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 62
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family 61
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 61
Enhancement of lysine acetylation accelerates wound repair 60
The emerging role of lysine methyltransferase SETD8 in human diseases 60
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. 60
A simplified synthesis of ethyl 5-chloro-6-fluoro-1H-indole-2-carboxylate and ethyl 5-chloro-4-fluoro-1H-indole-2-carboxylate 57
Totale 8.641
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Categoria #
all - tutte 27.450
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 27.450
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019304 0 0 0 0 0 0 0 0 0 0 288 16
2019/20201.091 311 10 116 14 85 31 114 21 111 77 188 13
2020/20211.055 9 99 130 11 119 42 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024515 62 108 64 30 42 112 38 23 7 27 2 0
Totale 10.874