UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
AS - Asia 8.773
NA - Nord America 8.732
EU - Europa 2.584
SA - Sud America 514
AF - Africa 50
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
Totale 20.668
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Nazione #
US - Stati Uniti d'America 8.679
HK - Hong Kong 6.596
SG - Singapore 804
IT - Italia 763
CN - Cina 687
BR - Brasile 477
UA - Ucraina 473
RU - Federazione Russa 393
DE - Germania 286
TR - Turchia 211
IE - Irlanda 198
VN - Vietnam 195
FI - Finlandia 135
SE - Svezia 111
KR - Corea 108
IN - India 54
GB - Regno Unito 45
FR - Francia 39
AT - Austria 30
PL - Polonia 24
CA - Canada 23
NL - Olanda 21
JP - Giappone 20
ZA - Sudafrica 19
PK - Pakistan 16
BD - Bangladesh 15
CZ - Repubblica Ceca 15
IQ - Iraq 15
ES - Italia 14
MX - Messico 14
GR - Grecia 13
AR - Argentina 11
EU - Europa 10
UZ - Uzbekistan 10
IL - Israele 8
MA - Marocco 8
EC - Ecuador 6
VE - Venezuela 6
CO - Colombia 5
DZ - Algeria 5
PE - Perù 5
AU - Australia 4
BG - Bulgaria 4
DO - Repubblica Dominicana 4
TN - Tunisia 4
AZ - Azerbaigian 3
CH - Svizzera 3
CL - Cile 3
ID - Indonesia 3
JO - Giordania 3
KE - Kenya 3
PH - Filippine 3
RO - Romania 3
TT - Trinidad e Tobago 3
AE - Emirati Arabi Uniti 2
CR - Costa Rica 2
EG - Egitto 2
GE - Georgia 2
JM - Giamaica 2
KH - Cambogia 2
KZ - Kazakistan 2
LB - Libano 2
LT - Lituania 2
NO - Norvegia 2
NP - Nepal 2
PS - Palestinian Territory 2
RS - Serbia 2
SA - Arabia Saudita 2
TH - Thailandia 2
AL - Albania 1
BA - Bosnia-Erzegovina 1
BE - Belgio 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
CV - Capo Verde 1
DK - Danimarca 1
DM - Dominica 1
ET - Etiopia 1
GH - Ghana 1
GT - Guatemala 1
IR - Iran 1
LU - Lussemburgo 1
MD - Moldavia 1
MN - Mongolia 1
MZ - Mozambico 1
NA - Namibia 1
NG - Nigeria 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
OM - Oman 1
PA - Panama 1
PT - Portogallo 1
PY - Paraguay 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
TW - Taiwan 1
Totale 20.668
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Città #
Hong Kong 6.589
Ann Arbor 2.189
Chandler 842
Houston 707
Woodbridge 666
Jacksonville 633
Wilmington 627
Princeton 565
Dallas 431
Singapore 291
Salerno 228
Ashburn 227
Izmir 194
Dublin 193
Beijing 161
Dong Ket 161
Nanjing 136
Andover 120
Boardman 120
Munich 101
Pellezzano 82
Moscow 61
Mestre 59
The Dalles 58
Columbus 53
Fairfield 53
Los Angeles 41
Shenyang 39
São Paulo 38
Dearborn 37
Hebei 35
Changsha 31
Council Bluffs 30
Turku 30
Jiaxing 26
Norwalk 26
Fisciano 25
Nanchang 25
New York 25
Redwood City 25
Nocera Superiore 24
Santa Clara 24
Düsseldorf 22
Falls Church 21
Pune 21
Tianjin 21
Washington 21
Naples 20
Nuremberg 20
Rome 20
Vienna 20
Tokyo 19
Philadelphia 17
Rio de Janeiro 17
Boston 15
Guangzhou 15
Belo Horizonte 14
Montreal 14
Warsaw 14
Brooklyn 13
San Diego 13
San Francisco 13
Cambridge 11
Chicago 11
Johannesburg 11
Athens 10
Napoli 10
Ankara 9
Brasília 9
Brno 9
Ho Chi Minh City 9
London 9
Paris 9
Seattle 9
Seoul 9
Amsterdam 8
Atlanta 8
Hefei 8
Kraków 8
Sarno 8
Tashkent 8
Chennai 7
Jinan 7
Scafati 7
Shanghai 7
Zhengzhou 7
Bari 6
Catania 6
Hanoi 6
Indiana 6
Joinville 6
Manchester 6
Milan 6
Munro 6
Olomouc 6
Renton 6
Baghdad 5
Bologna 5
Cagliari 5
Campagna 5
Totale 16.666
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.137
Two novel SIRT1 activators, SCIC2 and SCIC2.1, enhance SIRT1-mediated effects in stress response and senescence 852
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 685
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 587
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 424
Combined HAT/EZH2 modulation leads to cancer-selective cell death 383
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 369
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 355
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 313
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 313
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 301
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 296
Identification of small molecules inhibitors of GCN5 histone acetyltransferase activity. 289
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 243
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 226
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 200
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 191
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 182
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 180
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 178
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 168
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 163
Arginine demethylation of G3BP1 promotes stress granule assembly 160
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 157
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 157
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 154
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 151
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 150
In Quest of Chemical Probes for DNA Methylation Reader Proteins: Nucleoside and Dimer Analogues of 5‐Methylcytosine Interact with MBD2 150
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 144
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 142
Agenti antimicotici, antimicobatterici e antiprotozoari 142
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 140
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 130
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 130
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 128
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 127
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 126
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 125
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 124
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 124
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 121
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties 121
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 121
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 119
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 119
Chemical biology of Histone acetyltransferase natural compounds modulators. 118
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 117
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 116
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 113
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 113
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 113
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 112
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 111
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 110
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 110
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 110
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 109
New 6-nitroquinolones: synthesis and antimicrobial activities 108
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 108
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 108
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 107
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 107
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 107
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 106
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 105
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 104
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 104
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 104
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 104
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 103
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 103
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 103
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 102
Chemioterapici antiprotozoari 102
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 101
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 101
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 100
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 100
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 99
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 99
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 98
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 97
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 97
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 96
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 96
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 96
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 94
DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors 94
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 94
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 93
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 93
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 93
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 91
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 91
The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) 90
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. 90
N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 89
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 89
ChemInform Abstract: N-[4-(1,1′-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as Non-oxazolidinone Analogues of Antimycobacterial U-100480 89
Totale 16.804
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Categoria #
all - tutte 58.022
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 58.022
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021947 0 0 130 11 119 42 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024710 62 108 64 30 42 112 38 23 7 27 38 159
2024/20252.495 94 39 45 132 210 268 377 218 423 128 314 247
2025/20267.591 2.142 3.576 1.873 0 0 0 0 0 0 0 0 0
Totale 21.155