UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
AS - Asia 10.917
NA - Nord America 9.786
EU - Europa 2.742
SA - Sud America 720
AF - Africa 74
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
Totale 24.254
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Nazione #
US - Stati Uniti d'America 9.691
HK - Hong Kong 7.473
SG - Singapore 1.680
CN - Cina 837
IT - Italia 817
BR - Brasile 613
UA - Ucraina 478
RU - Federazione Russa 398
VN - Vietnam 323
DE - Germania 294
TR - Turchia 215
IE - Irlanda 198
FI - Finlandia 137
KR - Corea 125
SE - Svezia 116
IN - India 74
GB - Regno Unito 69
AR - Argentina 45
PL - Polonia 43
FR - Francia 42
CA - Canada 36
JP - Giappone 34
MX - Messico 34
AT - Austria 31
NL - Olanda 28
ES - Italia 27
ZA - Sudafrica 27
BD - Bangladesh 24
PK - Pakistan 22
ID - Indonesia 20
IQ - Iraq 20
CZ - Repubblica Ceca 16
EC - Ecuador 14
GR - Grecia 13
CO - Colombia 12
UZ - Uzbekistan 12
CL - Cile 11
MA - Marocco 11
EU - Europa 10
VE - Venezuela 10
DZ - Algeria 8
IL - Israele 8
DO - Repubblica Dominicana 7
PE - Perù 7
AE - Emirati Arabi Uniti 5
BG - Bulgaria 5
JO - Giordania 5
KE - Kenya 5
LB - Libano 5
RO - Romania 5
TN - Tunisia 5
AU - Australia 4
AZ - Azerbaigian 4
EG - Egitto 4
LT - Lituania 4
NP - Nepal 4
PY - Paraguay 4
SA - Arabia Saudita 4
BO - Bolivia 3
CH - Svizzera 3
JM - Giamaica 3
KH - Cambogia 3
KZ - Kazakistan 3
NI - Nicaragua 3
PH - Filippine 3
RS - Serbia 3
TT - Trinidad e Tobago 3
BA - Bosnia-Erzegovina 2
CR - Costa Rica 2
DK - Danimarca 2
ET - Etiopia 2
GE - Georgia 2
GT - Guatemala 2
MY - Malesia 2
NO - Norvegia 2
PS - Palestinian Territory 2
PT - Portogallo 2
SN - Senegal 2
TH - Thailandia 2
AL - Albania 1
BE - Belgio 1
BJ - Benin 1
BS - Bahamas 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
CV - Capo Verde 1
DM - Dominica 1
EE - Estonia 1
GH - Ghana 1
GN - Guinea 1
HN - Honduras 1
HR - Croazia 1
IR - Iran 1
KW - Kuwait 1
LU - Lussemburgo 1
MD - Moldavia 1
MN - Mongolia 1
MW - Malawi 1
MZ - Mozambico 1
Totale 24.245
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Città #
Hong Kong 7.465
Ann Arbor 2.189
Chandler 842
Singapore 770
Houston 718
Dallas 691
Woodbridge 666
Jacksonville 633
Wilmington 627
Princeton 565
Ashburn 369
San Jose 319
Salerno 228
Beijing 197
Izmir 194
Dublin 193
Dong Ket 161
Nanjing 136
Boardman 122
Andover 120
Munich 106
The Dalles 83
Pellezzano 82
Los Angeles 70
Moscow 61
Mestre 59
Ho Chi Minh City 56
São Paulo 55
Columbus 53
Fairfield 53
New York 53
Shenyang 39
Dearborn 37
Hebei 35
Hanoi 34
Santa Clara 33
Tokyo 33
Changsha 32
Turku 32
Warsaw 31
Council Bluffs 30
Jiaxing 26
Norwalk 26
Seoul 26
Fisciano 25
Nanchang 25
Naples 25
Redwood City 25
Montreal 24
Nocera Superiore 24
Düsseldorf 22
Rome 22
Falls Church 21
Nuremberg 21
Pune 21
Tianjin 21
Washington 21
Atlanta 20
Belo Horizonte 20
Brooklyn 20
Vienna 20
Boston 19
Denver 19
Rio de Janeiro 19
Guangzhou 17
Johannesburg 17
Philadelphia 17
Chicago 16
Jakarta 15
Chennai 14
Amsterdam 13
Ankara 13
Milan 13
Phoenix 13
San Diego 13
San Francisco 13
Brasília 12
Orem 12
Seattle 12
Cambridge 11
London 11
Poplar 11
Athens 10
Hefei 10
Mexico City 10
Napoli 10
Paris 10
Sarno 10
Tashkent 10
Baronissi 9
Brno 9
Shanghai 9
Campinas 8
Da Nang 8
Kraków 8
Manchester 8
Stockholm 8
Zhengzhou 8
Guarulhos 7
Haiphong 7
Totale 19.186
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Nome #
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 1.214
Two novel SIRT1 activators, SCIC2 and SCIC2.1, enhance SIRT1-mediated effects in stress response and senescence 879
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 763
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 670
Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors 499
Combined HAT/EZH2 modulation leads to cancer-selective cell death 452
Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors 441
Successes and challenges in the development of BD1-selective BET inhibitors: a patent review 417
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 370
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 358
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 323
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 317
Identification of small molecules inhibitors of GCN5 histone acetyltransferase activity. 304
Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20 277
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 246
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 243
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor 223
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 218
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 217
FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS. 216
Arginine demethylation of G3BP1 promotes stress granule assembly 207
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 203
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 199
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 192
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 192
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 182
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 176
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 175
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 174
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 166
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 161
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 159
In Quest of Chemical Probes for DNA Methylation Reader Proteins: Nucleoside and Dimer Analogues of 5‐Methylcytosine Interact with MBD2 159
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties 156
Agenti antimicotici, antimicobatterici e antiprotozoari 156
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 154
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 151
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 148
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 147
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 147
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 147
Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23. 144
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 142
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 140
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 139
Chemical biology of Histone acetyltransferase natural compounds modulators. 137
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 137
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 136
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 136
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 136
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 134
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 133
Chemioterapici antiprotozoari 133
Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain 132
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 132
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 132
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 131
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 131
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 128
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 125
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 125
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 124
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 124
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 124
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 123
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family 121
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 119
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 118
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 118
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 118
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 118
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 117
New 6-nitroquinolones: synthesis and antimicrobial activities 116
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 116
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 116
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 116
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 114
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 114
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 112
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 112
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 112
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 111
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 111
6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase 110
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 110
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 110
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 109
The emerging role of lysine methyltransferase SETD8 in human diseases 109
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 109
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 108
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 108
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 106
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 106
ChemInform Abstract: N-[4-(1,1′-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as Non-oxazolidinone Analogues of Antimycobacterial U-100480 106
Structure-activity relationship studies on new DABOs: effect of substitutions at pyrimidine C-5 and C-6 positions on anti-HIV-1 activity 105
A novel Gcn5p inhibitor represses cell growth, gene transcription and histone acetylation in budding yeast 105
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 105
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 105
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 104
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 104
Totale 19.274
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Categoria #
all - tutte 68.538
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 68.538
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021645 0 0 0 0 0 0 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024710 62 108 64 30 42 112 38 23 7 27 38 159
2024/20252.495 94 39 45 132 210 268 377 218 423 128 314 247
2025/202611.184 2.142 3.576 3.140 498 940 471 417 0 0 0 0 0
Totale 24.748