UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
NA - Nord America 8.074
EU - Europa 2.498
AS - Asia 2.007
SA - Sud America 453
AF - Africa 36
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
Totale 13.083
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Nazione #
US - Stati Uniti d'America 8.044
SG - Singapore 755
IT - Italia 754
CN - Cina 589
UA - Ucraina 471
BR - Brasile 421
RU - Federazione Russa 390
DE - Germania 258
TR - Turchia 206
IE - Irlanda 198
VN - Vietnam 168
FI - Finlandia 134
SE - Svezia 110
KR - Corea 101
HK - Hong Kong 74
IN - India 40
FR - Francia 38
GB - Regno Unito 33
AT - Austria 27
NL - Olanda 19
CZ - Repubblica Ceca 15
PL - Polonia 14
IQ - Iraq 13
GR - Grecia 12
ZA - Sudafrica 12
PK - Pakistan 11
AR - Argentina 10
BD - Bangladesh 10
CA - Canada 10
EU - Europa 10
MX - Messico 8
MA - Marocco 7
UZ - Uzbekistan 7
IL - Israele 6
VE - Venezuela 6
CO - Colombia 5
DZ - Algeria 5
ES - Italia 5
AU - Australia 4
BG - Bulgaria 4
DO - Repubblica Dominicana 4
EC - Ecuador 4
PE - Perù 4
CH - Svizzera 3
CL - Cile 3
JO - Giordania 3
JP - Giappone 3
KE - Kenya 3
TN - Tunisia 3
AE - Emirati Arabi Uniti 2
AZ - Azerbaigian 2
CR - Costa Rica 2
EG - Egitto 2
KH - Cambogia 2
LB - Libano 2
NO - Norvegia 2
NP - Nepal 2
PS - Palestinian Territory 2
RO - Romania 2
RS - Serbia 2
SA - Arabia Saudita 2
TH - Thailandia 2
AL - Albania 1
BE - Belgio 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
DK - Danimarca 1
GE - Georgia 1
GH - Ghana 1
GT - Guatemala 1
IR - Iran 1
JM - Giamaica 1
KZ - Kazakistan 1
LT - Lituania 1
LU - Lussemburgo 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
OM - Oman 1
PA - Panama 1
PT - Portogallo 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
Totale 13.083
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Città #
Ann Arbor 2.189
Chandler 842
Houston 706
Woodbridge 666
Jacksonville 631
Wilmington 627
Princeton 565
Singapore 246
Salerno 228
Izmir 194
Dublin 193
Ashburn 188
Dong Ket 161
Beijing 141
Nanjing 136
Andover 120
Boardman 119
Pellezzano 82
Munich 76
Hong Kong 72
Moscow 61
Mestre 59
The Dalles 58
Fairfield 53
Shenyang 39
Dearborn 37
Hebei 35
Changsha 31
São Paulo 30
Turku 30
Council Bluffs 27
Jiaxing 26
Los Angeles 26
Norwalk 26
Nanchang 25
Redwood City 25
Fisciano 24
Nocera Superiore 24
Dallas 23
Düsseldorf 22
Falls Church 21
Pune 21
Tianjin 21
Rome 20
Naples 19
Vienna 18
Washington 18
Nuremberg 17
Philadelphia 17
Guangzhou 15
New York 15
Belo Horizonte 13
San Diego 13
Rio de Janeiro 12
Cambridge 11
Napoli 10
Athens 9
Brno 9
Columbus 9
Paris 9
San Francisco 9
Seattle 9
Hefei 8
Kraków 8
London 8
Sarno 8
Amsterdam 7
Brasília 7
Jinan 7
Shanghai 7
Zhengzhou 7
Bari 6
Catania 6
Indiana 6
Joinville 6
Milan 6
Munro 6
Olomouc 6
Renton 6
Santa Clara 6
Tashkent 6
Warsaw 6
Baghdad 5
Bologna 5
Boston 5
Brooklyn 5
Cagliari 5
Campagna 5
Campinas 5
Chicago 5
Dhaka 5
Florence 5
Guarulhos 5
Johannesburg 5
Palermo 5
Recife 5
Sorrento 5
Tappahannock 5
Venezia 5
Wuhan 5
Totale 9.401
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Nome #
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 179
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 177
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 158
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 152
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 143
Agenti antimicotici, antimicobatterici e antiprotozoari 138
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 136
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 136
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 129
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 129
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 127
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 126
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 124
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 123
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 122
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 122
Arginine demethylation of G3BP1 promotes stress granule assembly 122
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 122
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 120
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 119
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 118
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 118
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 116
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 115
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 114
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 113
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 111
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 110
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 110
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 110
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 109
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 108
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 108
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 108
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 106
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 106
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 105
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 103
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 103
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 103
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 103
New 6-nitroquinolones: synthesis and antimicrobial activities 102
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 102
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 101
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 101
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 101
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 99
Chemical biology of Histone acetyltransferase natural compounds modulators. 99
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 99
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 97
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 97
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 97
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 97
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 97
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 97
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 96
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 96
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 94
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 94
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 94
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 94
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 93
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 93
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 93
DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors 90
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 89
Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian 89
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 89
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 88
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 88
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 88
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 88
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 88
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 88
SELECTIVE INHIBITORS FOR TRANSFERASES 87
The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) 86
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. 86
N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 85
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 85
Methods for inhibiting the transmission of HIV using topically applied substituted 6-​benzyl-​4-​oxopyrimidines 85
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 84
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 84
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 84
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 82
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family 81
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 80
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure 80
6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase 79
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 78
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 78
Chemioterapici antiprotozoari 78
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 78
A simplified synthesis of ethyl 5-chloro-6-fluoro-1H-indole-2-carboxylate and ethyl 5-chloro-4-fluoro-1H-indole-2-carboxylate 77
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 77
ChemInform Abstract: A Simplified Synthesis of Ethyl 5-Chloro-4-fluoro-1H-indole-2-carboxylate and Ethyl 5-Chloro-6-fluoro-1H-indole-2-carboxylate 77
Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity 76
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties 75
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 75
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 75
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 75
Totale 10.206
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Categoria #
all - tutte 45.100
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 45.100
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/20211.055 9 99 130 11 119 42 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024710 62 108 64 30 42 112 38 23 7 27 38 159
2024/20252.495 94 39 45 132 210 268 377 218 423 128 314 247
2025/20264 4 0 0 0 0 0 0 0 0 0 0 0
Totale 13.568