UniSa - IRIS Institutional Research Information System

SBARDELLA, Gianluca
 Distribuzione geografica
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Continente #
NA - Nord America 7.880
EU - Europa 2.347
AS - Asia 1.857
SA - Sud America 403
AF - Africa 29
Continente sconosciuto - Info sul continente non disponibili 10
OC - Oceania 5
Totale 12.531
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Nazione #
US - Stati Uniti d'America 7.861
IT - Italia 749
SG - Singapore 738
CN - Cina 565
UA - Ucraina 471
RU - Federazione Russa 388
BR - Brasile 376
TR - Turchia 204
IE - Irlanda 198
DE - Germania 184
VN - Vietnam 165
SE - Svezia 109
FI - Finlandia 104
KR - Corea 67
IN - India 36
FR - Francia 25
GB - Regno Unito 25
AT - Austria 24
HK - Hong Kong 21
NL - Olanda 19
GR - Grecia 12
AR - Argentina 10
EU - Europa 10
PK - Pakistan 10
PL - Polonia 10
CZ - Repubblica Ceca 9
IQ - Iraq 9
ZA - Sudafrica 8
MA - Marocco 7
BD - Bangladesh 6
IL - Israele 6
UZ - Uzbekistan 6
VE - Venezuela 6
MX - Messico 5
AU - Australia 4
BG - Bulgaria 4
CO - Colombia 4
DO - Repubblica Dominicana 4
CA - Canada 3
CH - Svizzera 3
DZ - Algeria 3
EC - Ecuador 3
JO - Giordania 3
JP - Giappone 3
TN - Tunisia 3
AZ - Azerbaigian 2
CL - Cile 2
CR - Costa Rica 2
EG - Egitto 2
KE - Kenya 2
KH - Cambogia 2
LB - Libano 2
NO - Norvegia 2
NP - Nepal 2
PE - Perù 2
PS - Palestinian Territory 2
RO - Romania 2
RS - Serbia 2
TH - Thailandia 2
AE - Emirati Arabi Uniti 1
AL - Albania 1
BE - Belgio 1
BW - Botswana 1
BZ - Belize 1
CG - Congo 1
DK - Danimarca 1
ES - Italia 1
GE - Georgia 1
GH - Ghana 1
GT - Guatemala 1
IR - Iran 1
JM - Giamaica 1
LU - Lussemburgo 1
NI - Nicaragua 1
NZ - Nuova Zelanda 1
OM - Oman 1
PT - Portogallo 1
SA - Arabia Saudita 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
Totale 12.531
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Città #
Ann Arbor 2.189
Chandler 842
Houston 706
Woodbridge 666
Jacksonville 631
Wilmington 626
Princeton 565
Singapore 232
Salerno 228
Izmir 194
Dublin 193
Ashburn 185
Dong Ket 161
Nanjing 136
Andover 120
Beijing 120
Boardman 119
Pellezzano 82
Moscow 61
Mestre 59
Fairfield 53
Shenyang 39
Dearborn 37
Hebei 35
Changsha 31
São Paulo 29
Council Bluffs 27
Jiaxing 26
Norwalk 26
Nanchang 25
Redwood City 25
Fisciano 24
Nocera Superiore 24
Düsseldorf 22
Falls Church 21
Pune 21
Tianjin 21
Rome 20
Hong Kong 19
Naples 18
Washington 18
Dallas 17
Philadelphia 17
Vienna 17
Guangzhou 15
San Diego 13
Los Angeles 12
Nuremberg 12
Cambridge 11
New York 11
Rio de Janeiro 11
Napoli 10
Athens 9
Belo Horizonte 9
Brno 9
The Dalles 9
Hefei 8
Kraków 8
Sarno 8
Seattle 8
Amsterdam 7
Jinan 7
Munich 7
Shanghai 7
Zhengzhou 7
Bari 6
Brasília 6
Catania 6
Indiana 6
London 6
Milan 6
Munro 6
Renton 6
Bologna 5
Cagliari 5
Campagna 5
Florence 5
Palermo 5
Sorrento 5
Tappahannock 5
Tashkent 5
Venezia 5
Wuhan 5
Yubileyny 5
Atlanta 4
Baghdad 4
Campinas 4
Curitiba 4
Dhaka 4
Groningen 4
Hamburg 4
Joinville 4
Kolkata 4
Lappeenranta 4
Lucknow 4
Maringá 4
Recife 4
Ribeirão Preto 4
San Francisco 4
Spinea 4
Totale 9.092
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Nome #
Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. 177
A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach 166
The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme 155
CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli 146
Agenti antimicotici, antimicobatterici e antiprotozoari 138
Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors 136
A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery 135
Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS 134
Developing Spindlin1 small-molecule inhibitors by using protein microarrays 126
A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems 125
Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 123
Arginine demethylation of G3BP1 promotes stress granule assembly 122
3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A 121
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation 120
Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) 118
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors 118
Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) 117
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. 116
Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions 115
Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF 115
ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction 114
ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 114
A TR-FRET-Based Functional Assay for Screening Activators of CARM1 113
Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors 113
Preparation of oxo-​pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection 110
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 110
Preparation of substituted 6-​benzyl-​4-​oxopyrimidines for prevention and treatment of HIV infection 109
Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans 108
Preparation of 6-​benzyl-​4-​oxopyrimidines as antiviral agents 108
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation 107
A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. 106
Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. 105
3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 105
Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant 104
N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. 103
Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) 103
Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors 102
New 6-nitroquinolones: synthesis and antimicrobial activities 101
ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro 101
Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins 100
Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. 99
Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) 99
Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors 99
MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS 98
Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation 97
Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. 96
Chemical biology of Histone acetyltransferase natural compounds modulators. 96
Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein 96
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells 96
Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors 95
Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids 95
ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery 95
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. 94
Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains 94
p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear 94
Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors 94
ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators 93
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase 93
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors 92
STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA 92
ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation 92
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. 92
Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. 90
Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells 90
DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors 90
Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian 89
Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations 88
SELECTIVE INHIBITORS FOR TRANSFERASES 87
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells 87
The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients 85
Methods for inhibiting the transmission of HIV using topically applied substituted 6-​benzyl-​4-​oxopyrimidines 85
The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) 85
Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. 85
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart 84
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer 84
N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 83
Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach 82
Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. 82
Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins 80
3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors 79
P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins 79
Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach 79
Chemioterapici antiprotozoari 78
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases 77
ChemInform Abstract: A Simplified Synthesis of Ethyl 5-Chloro-4-fluoro-1H-indole-2-carboxylate and Ethyl 5-Chloro-6-fluoro-1H-indole-2-carboxylate 77
6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase 76
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors 76
Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery. 76
DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH 76
5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family 75
Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity 75
Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors 75
A simplified synthesis of ethyl 5-chloro-6-fluoro-1H-indole-2-carboxylate and ethyl 5-chloro-4-fluoro-1H-indole-2-carboxylate 74
6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation 74
Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 74
Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties 73
ChemInform Abstract: N-[4-(1,1′-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as Non-oxazolidinone Analogues of Antimycobacterial U-100480 73
Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells 73
Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. 72
Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients 72
Totale 9.889
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Categoria #
all - tutte 42.785
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 42.785
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020201 0 0 0 0 0 0 0 0 0 0 188 13
2020/20211.055 9 99 130 11 119 42 120 25 141 14 126 219
2021/20221.058 3 6 6 8 26 32 20 45 130 142 164 476
2022/20231.823 173 169 56 261 220 355 16 175 285 8 72 33
2023/2024710 62 108 64 30 42 112 38 23 7 27 38 159
2024/20251.944 94 39 45 132 210 268 377 218 423 128 10 0
Totale 13.013